ES2396723T3 - Composición farmacéutica auto-emulsionante con biodisponibilidad mejorada - Google Patents
Composición farmacéutica auto-emulsionante con biodisponibilidad mejorada Download PDFInfo
- Publication number
- ES2396723T3 ES2396723T3 ES08020342T ES08020342T ES2396723T3 ES 2396723 T3 ES2396723 T3 ES 2396723T3 ES 08020342 T ES08020342 T ES 08020342T ES 08020342 T ES08020342 T ES 08020342T ES 2396723 T3 ES2396723 T3 ES 2396723T3
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- pharmaceutical composition
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
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- A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US944239 | 2007-11-21 | ||
| US11/944,239 US20090130198A1 (en) | 2007-11-21 | 2007-11-21 | Pharmaceutical composition with enhanced bioavailability |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2396723T3 true ES2396723T3 (es) | 2013-02-25 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES08020342T Active ES2396723T3 (es) | 2007-11-21 | 2008-11-21 | Composición farmacéutica auto-emulsionante con biodisponibilidad mejorada |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20090130198A1 (enExample) |
| EP (1) | EP2062571B8 (enExample) |
| JP (3) | JP5491724B2 (enExample) |
| CN (1) | CN101439015B (enExample) |
| ES (1) | ES2396723T3 (enExample) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ592970A (en) * | 2008-12-03 | 2013-05-31 | Astellas Deutschland Gmbh | Oral dosage forms of bendamustine |
| DK2519261T3 (da) | 2009-12-28 | 2014-02-03 | Reig Jofre S A Lab | Flydende oralt farmaceutisk præparat, som er en opløsning omfattende nifedipin. |
| SG10201503234SA (en) | 2010-05-03 | 2015-06-29 | Teikoku Pharma Usa Inc | Non-Aqueous Taxane Pro-Emulsion Formulations and Methods of Making and Using the Same |
| MY158809A (en) * | 2010-09-22 | 2016-11-15 | Craun Res Sdn Bhd | Pharmaceutical compositions for calanolides, their derivatives and analogues, and process for producing the same |
| CN102389401B (zh) * | 2011-11-22 | 2013-05-22 | 陆荣政 | 一种右旋布洛芬颗粒及其制备方法 |
| KR101211902B1 (ko) * | 2012-04-30 | 2012-12-13 | 주식회사 휴온스 | 사이클로스포린 함유 무자극성 나노에멀젼 안약 조성물 |
| JO3685B1 (ar) | 2012-10-01 | 2020-08-27 | Teikoku Pharma Usa Inc | صيغ التشتيت الجسيمي للتاكسين غير المائي وطرق استخدامها |
| CN109953954A (zh) | 2013-08-27 | 2019-07-02 | V·沃道里斯 | 苯达莫司汀医药组合物 |
| RU2746548C2 (ru) * | 2014-11-04 | 2021-04-15 | Иннофармакс, Инк. | Пероральное введение неустойчивых или плохо всасывающихся лекарственных средств |
| EP3337463A4 (en) * | 2015-08-19 | 2019-04-03 | Vivus, Inc. | PHARMACEUTICAL FORMULATIONS |
| JP6103111B1 (ja) | 2016-05-24 | 2017-03-29 | 三生医薬株式会社 | 経口医薬組成物及び該組成物からなる粒子状製剤の製造方法 |
| JP2020152674A (ja) * | 2019-03-20 | 2020-09-24 | 株式会社リコー | 難水溶性化合物の可溶化物の製造方法 |
| KR102676428B1 (ko) * | 2019-07-08 | 2024-06-19 | 가부시키가이샤 모레스코 | 마이크로에멀션을 조제하기 위한 조성물, 마이크로에멀션, 이들의 제조 방법, 및 마이크로에멀션의 이용 |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8630273D0 (en) * | 1986-12-18 | 1987-01-28 | Til Medical Ltd | Pharmaceutical delivery systems |
| AU1766592A (en) * | 1991-06-03 | 1993-01-08 | Merck Sharp & Dohme Limited | Pharmaceutical formulations of a benzodiazepine |
| US6312704B1 (en) * | 1993-09-30 | 2001-11-06 | Gattefosse, S.A. | Orally administrable composition capable of providing enhanced bioavailability when ingested |
| US6054136A (en) * | 1993-09-30 | 2000-04-25 | Gattefosse S.A. | Orally administrable composition capable of providing enhanced bioavailability when ingested |
| US5965160A (en) * | 1995-04-24 | 1999-10-12 | Yissum Research Development Company Of The Hebrew University Of Jerusalem | Self-emulsifiable formulation producing an oil-in-water emulsion |
| JP3009742B2 (ja) * | 1995-08-25 | 2000-02-14 | サングスタット メディカル コーポレイション | 経口用シクロスポリン製剤 |
| KR970064620A (ko) * | 1996-03-05 | 1997-10-13 | 임성기 | 사이클로스포린-함유 외용약제 조성물 |
| US5993858A (en) * | 1996-06-14 | 1999-11-30 | Port Systems L.L.C. | Method and formulation for increasing the bioavailability of poorly water-soluble drugs |
| US6458373B1 (en) * | 1997-01-07 | 2002-10-01 | Sonus Pharmaceuticals, Inc. | Emulsion vehicle for poorly soluble drugs |
| KR20040004416A (ko) * | 1997-01-30 | 2004-01-13 | 노파르티스 아게 | 오일을 함유하지 않은 사이클로스포린 ａ 함유 제약 조성물 |
| NZ337316A (en) * | 1997-03-12 | 2001-06-29 | Abbott Lab | Hydrophilic binary systems comprising cyclosporine, hydrophilic phase and a surfactant for the administration of cyclosporine |
| ID25908A (id) * | 1998-03-06 | 2000-11-09 | Novartis Ag | Prakonsentrat-prakonsentrat emulsi yang mengandung siklosporin atau makrolida |
| AU3843999A (en) * | 1998-05-07 | 1999-11-23 | Elan Corporation, Plc | Solvent/cosolvent free microemulsion and emulsion preconcentrate drug delivery systems |
| DE69822814T2 (de) * | 1998-08-18 | 2005-01-27 | Panacea Biotec Ltd. | Zusammensetzung enthaltend Cyclosporin in einem hydrophilen Träger |
| CN1236813C (zh) * | 1998-12-11 | 2006-01-18 | 药品处理公司 | 水难溶性药物的自乳化组合物 |
| US6294192B1 (en) * | 1999-02-26 | 2001-09-25 | Lipocine, Inc. | Triglyceride-free compositions and methods for improved delivery of hydrophobic therapeutic agents |
| US6057289A (en) * | 1999-04-30 | 2000-05-02 | Pharmasolutions, Inc. | Pharmaceutical composition comprising cyclosporin in association with a carrier in a self-emulsifying drug delivery system |
| US6596306B1 (en) * | 2000-07-07 | 2003-07-22 | David Ho Sue San Ho | Drug delivery system:formulation for fat-soluble drugs |
| DE10133305B4 (de) * | 2001-07-12 | 2004-06-03 | Aquanova German Solubilisate Technologies (Agt) Gmbh | Ubichinon Konzentrat |
| US6960563B2 (en) * | 2001-08-31 | 2005-11-01 | Morton Grove Pharmaceuticals, Inc. | Spontaneous emulsions containing cyclosporine |
| JP2005343799A (ja) * | 2004-05-31 | 2005-12-15 | Nisshin Oillio Group Ltd | 水分散性植物ステロース製剤と油脂含有水分散性植物ステロール製剤 |
| KR100678829B1 (ko) * | 2004-12-06 | 2007-02-05 | 한미약품 주식회사 | 타크로리무스의 경구용 마이크로에멀젼 조성물 |
-
2007
- 2007-11-21 US US11/944,239 patent/US20090130198A1/en not_active Abandoned
-
2008
- 2008-11-21 EP EP08020342A patent/EP2062571B8/en active Active
- 2008-11-21 JP JP2008298513A patent/JP5491724B2/ja not_active Expired - Fee Related
- 2008-11-21 CN CN2008101811022A patent/CN101439015B/zh not_active Expired - Fee Related
- 2008-11-21 ES ES08020342T patent/ES2396723T3/es active Active
-
2014
- 2014-02-28 JP JP2014038075A patent/JP2014098039A/ja active Pending
-
2016
- 2016-03-17 JP JP2016053870A patent/JP2016106152A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| US20090130198A1 (en) | 2009-05-21 |
| EP2062571B1 (en) | 2012-11-14 |
| CN101439015B (zh) | 2013-02-13 |
| CN101439015A (zh) | 2009-05-27 |
| JP2016106152A (ja) | 2016-06-16 |
| EP2062571A1 (en) | 2009-05-27 |
| JP5491724B2 (ja) | 2014-05-14 |
| EP2062571B8 (en) | 2012-12-19 |
| JP2014098039A (ja) | 2014-05-29 |
| JP2009132712A (ja) | 2009-06-18 |
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