ES2342181T3 - Compuestos quimicos i. - Google Patents

Compuestos quimicos i. Download PDF

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Publication number
ES2342181T3
ES2342181T3 ES05753676T ES05753676T ES2342181T3 ES 2342181 T3 ES2342181 T3 ES 2342181T3 ES 05753676 T ES05753676 T ES 05753676T ES 05753676 T ES05753676 T ES 05753676T ES 2342181 T3 ES2342181 T3 ES 2342181T3
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ES
Spain
Prior art keywords
compound
pharmaceutically acceptable
piperidin
salt
methylsulfonyl
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ES05753676T
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English (en)
Spanish (es)
Inventor
Howard Tucker
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AstraZeneca AB
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AstraZeneca AB
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Application filed by AstraZeneca AB filed Critical AstraZeneca AB
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Publication of ES2342181T3 publication Critical patent/ES2342181T3/es
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Dermatology (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Molecular Biology (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
ES05753676T 2004-06-24 2005-06-20 Compuestos quimicos i. Active ES2342181T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE2004101657 2004-06-24
SE0401657A SE0401657D0 (sv) 2004-06-24 2004-06-24 Chemical compounds

Publications (1)

Publication Number Publication Date
ES2342181T3 true ES2342181T3 (es) 2010-07-02

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ES05753676T Active ES2342181T3 (es) 2004-06-24 2005-06-20 Compuestos quimicos i.

Country Status (22)

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US (1) US20070259914A1 (xx)
EP (1) EP1761494B1 (xx)
JP (1) JP5147393B2 (xx)
CN (1) CN101006058A (xx)
AR (1) AR049830A1 (xx)
AT (1) ATE465148T1 (xx)
AU (1) AU2005257707B2 (xx)
BR (1) BRPI0512420A (xx)
CA (1) CA2571087A1 (xx)
DE (1) DE602005020787D1 (xx)
ES (1) ES2342181T3 (xx)
IL (1) IL179729A0 (xx)
MX (1) MXPA06014413A (xx)
MY (1) MY139268A (xx)
NO (1) NO20070431L (xx)
RU (1) RU2381216C2 (xx)
SE (1) SE0401657D0 (xx)
TW (1) TW200610759A (xx)
UA (1) UA88303C2 (xx)
UY (1) UY28974A1 (xx)
WO (1) WO2006001751A1 (xx)
ZA (1) ZA200610526B (xx)

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Publication number Priority date Publication date Assignee Title
TW200610761A (en) * 2004-04-23 2006-04-01 Astrazeneca Ab Chemical compounds
EP2066674B1 (en) 2006-09-18 2010-06-30 F.Hoffmann-La Roche Ag Octahydropyrrolo [3, 4-c] pyrrole derivatives and their use as antiviral agents
EP2173715A2 (en) * 2007-07-13 2010-04-14 Euroscreen S.A. Use of piperidine derivatives as agonists of chemokine receptor activity
WO2009151910A2 (en) * 2008-05-25 2009-12-17 Wyeth Combination product of receptor tyrosine kinase inhibitor and fatty acid synthase inhibitor for treating cancer
WO2012113103A1 (en) 2011-02-25 2012-08-30 Helsinn Healthcare S.A. Asymmetric ureas and medical uses thereof
GB201321746D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
NO2699580T3 (xx) 2014-01-24 2018-02-24
EA037040B1 (ru) 2016-03-22 2021-01-29 Хелсинн Хелскеа Са Асимметричные бензолсульфонилмочевины и их применение в качестве модуляторов рецептора грелина
US20220072013A1 (en) * 2018-12-21 2022-03-10 Ca*Tx, Inc. Pharmaceutical Combinations for the Treatment of Cancer

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GB9624482D0 (en) 1995-12-18 1997-01-15 Zeneca Phaema S A Chemical compounds
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WO2006001751A1 (en) 2006-01-05
EP1761494A1 (en) 2007-03-14
MY139268A (en) 2009-09-30
AR049830A1 (es) 2006-09-06
AU2005257707B2 (en) 2009-03-26
UY28974A1 (es) 2006-01-31
US20070259914A1 (en) 2007-11-08
NO20070431L (no) 2007-03-26
MXPA06014413A (es) 2007-02-19
CA2571087A1 (en) 2006-01-05
EP1761494B1 (en) 2010-04-21
UA88303C2 (ru) 2009-10-12
JP2008503572A (ja) 2008-02-07
CN101006058A (zh) 2007-07-25
AU2005257707A1 (en) 2006-01-05
TW200610759A (en) 2006-04-01
ZA200610526B (en) 2008-08-27
JP5147393B2 (ja) 2013-02-20
DE602005020787D1 (de) 2010-06-02
SE0401657D0 (sv) 2004-06-24
BRPI0512420A (pt) 2008-03-04
RU2006146877A (ru) 2008-07-27

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