UY28974A1 - Derivados heterocíclicos de piperidina, composiciones que los contienen y procedimiento de preparación - Google Patents

Derivados heterocíclicos de piperidina, composiciones que los contienen y procedimiento de preparación

Info

Publication number
UY28974A1
UY28974A1 UY28974A UY28974A UY28974A1 UY 28974 A1 UY28974 A1 UY 28974A1 UY 28974 A UY28974 A UY 28974A UY 28974 A UY28974 A UY 28974A UY 28974 A1 UY28974 A1 UY 28974A1
Authority
UY
Uruguay
Prior art keywords
compositions
hiperocyclic
piperidine
derivatives
contain
Prior art date
Application number
UY28974A
Other languages
English (en)
Inventor
Howard Tucker
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32733687&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY28974(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY28974A1 publication Critical patent/UY28974A1/es

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
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  • Physical Education & Sports Medicine (AREA)
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  • Oncology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Molecular Biology (AREA)
  • Ophthalmology & Optometry (AREA)
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Abstract

Compuestos de fórmula (I): composiciones que los contienen, procedimientos para su preparación y su uso en terapia médica (por ejemplo modulando la actividad del receptor CCR5 en un animal de sangre caliente).
UY28974A 2004-06-24 2005-06-21 Derivados heterocíclicos de piperidina, composiciones que los contienen y procedimiento de preparación UY28974A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0401657A SE0401657D0 (sv) 2004-06-24 2004-06-24 Chemical compounds

Publications (1)

Publication Number Publication Date
UY28974A1 true UY28974A1 (es) 2006-01-31

Family

ID=32733687

Family Applications (1)

Application Number Title Priority Date Filing Date
UY28974A UY28974A1 (es) 2004-06-24 2005-06-21 Derivados heterocíclicos de piperidina, composiciones que los contienen y procedimiento de preparación

Country Status (22)

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US (1) US20070259914A1 (es)
EP (1) EP1761494B1 (es)
JP (1) JP5147393B2 (es)
CN (1) CN101006058A (es)
AR (1) AR049830A1 (es)
AT (1) ATE465148T1 (es)
AU (1) AU2005257707B2 (es)
BR (1) BRPI0512420A (es)
CA (1) CA2571087A1 (es)
DE (1) DE602005020787D1 (es)
ES (1) ES2342181T3 (es)
IL (1) IL179729A0 (es)
MX (1) MXPA06014413A (es)
MY (1) MY139268A (es)
NO (1) NO20070431L (es)
RU (1) RU2381216C2 (es)
SE (1) SE0401657D0 (es)
TW (1) TW200610759A (es)
UA (1) UA88303C2 (es)
UY (1) UY28974A1 (es)
WO (1) WO2006001751A1 (es)
ZA (1) ZA200610526B (es)

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TW200610761A (en) * 2004-04-23 2006-04-01 Astrazeneca Ab Chemical compounds
ATE472549T1 (de) 2006-09-18 2010-07-15 Hoffmann La Roche Octahydropyrroloä3,4-cüpyrrolderivate und ihre verwendung als antivirale mittel
EP2173715A2 (en) * 2007-07-13 2010-04-14 Euroscreen S.A. Use of piperidine derivatives as agonists of chemokine receptor activity
WO2009151910A2 (en) * 2008-05-25 2009-12-17 Wyeth Combination product of receptor tyrosine kinase inhibitor and fatty acid synthase inhibitor for treating cancer
WO2012113103A1 (en) 2011-02-25 2012-08-30 Helsinn Healthcare S.A. Asymmetric ureas and medical uses thereof
GB201321746D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
NO2699580T3 (es) 2014-01-24 2018-02-24
SI3390355T1 (sl) 2016-03-22 2023-07-31 Helsinn Healthcare S. A. Benzensulfonil-asimetrične sečnine in njihove medicinske uporabe
JP2022516252A (ja) * 2018-12-21 2022-02-25 シーエー*ティーエックス, インコーポレイテッド がんを処置するための薬学的組合せ

Family Cites Families (15)

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EP0880508B1 (en) 1996-02-13 2003-04-16 AstraZeneca AB Quinazoline derivatives as vegf inhibitors
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NO20070431L (no) 2007-03-26
IL179729A0 (en) 2007-05-15
DE602005020787D1 (de) 2010-06-02
MXPA06014413A (es) 2007-02-19
SE0401657D0 (sv) 2004-06-24
BRPI0512420A (pt) 2008-03-04
RU2381216C2 (ru) 2010-02-10
AU2005257707B2 (en) 2009-03-26
US20070259914A1 (en) 2007-11-08
CA2571087A1 (en) 2006-01-05
ES2342181T3 (es) 2010-07-02
RU2006146877A (ru) 2008-07-27
JP2008503572A (ja) 2008-02-07
AR049830A1 (es) 2006-09-06
UA88303C2 (ru) 2009-10-12
TW200610759A (en) 2006-04-01
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EP1761494B1 (en) 2010-04-21
EP1761494A1 (en) 2007-03-14
MY139268A (en) 2009-09-30
ATE465148T1 (de) 2010-05-15
JP5147393B2 (ja) 2013-02-20

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