ES2282497T3 - 2-amino-cicloalcancarboxamidas sustiruidas y su empleo como inhibidores de cistein proteasa. - Google Patents

2-amino-cicloalcancarboxamidas sustiruidas y su empleo como inhibidores de cistein proteasa. Download PDF

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Publication number
ES2282497T3
ES2282497T3 ES02787799T ES02787799T ES2282497T3 ES 2282497 T3 ES2282497 T3 ES 2282497T3 ES 02787799 T ES02787799 T ES 02787799T ES 02787799 T ES02787799 T ES 02787799T ES 2282497 T3 ES2282497 T3 ES 2282497T3
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indole
methyl
amino
cyclohexyl
carbonyl
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Spanish (es)
Inventor
Tobias Gabriel
Nancy Elisabeth Krauss
Taraneh Mirzadegan
Wylie Solang Palmer
David Bernard Smith
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F Hoffmann La Roche AG
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F Hoffmann La Roche AG
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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ES02787799T 2001-12-04 2002-11-25 2-amino-cicloalcancarboxamidas sustiruidas y su empleo como inhibidores de cistein proteasa. Expired - Lifetime ES2282497T3 (es)

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US33675001P 2001-12-04 2001-12-04
US336750P 2001-12-04

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US7005445B2 (en) * 2001-10-22 2006-02-28 The Research Foundation Of State University Of New York Protein kinase and phosphatase inhibitors and methods for designing them
GB0128996D0 (en) 2001-12-04 2002-01-23 Novartis Ag Organic compounds
DE60305446T4 (de) * 2002-01-07 2009-07-09 Eisai R&D Management Co., Ltd. Desazapurine und deren verwendung
SE0203712D0 (sv) 2002-12-13 2002-12-13 Astrazeneca Ab Novel compounds
GB0403038D0 (en) 2004-02-11 2004-03-17 Novartis Ag Organic compounds
US20090226552A1 (en) * 2004-07-22 2009-09-10 Colorado State University Research Foundation Agents and methods for diagnosing osteoarthritis
AU2006261954A1 (en) * 2005-06-28 2007-01-04 Merck & Co., Inc. Non-nucleoside reverse transcriptase inhibitors
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KR20050044660A (ko) 2005-05-12
US20030212097A1 (en) 2003-11-13
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DE60219068T2 (de) 2007-12-13
IL161992A0 (en) 2005-11-20
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EP1453801A1 (en) 2004-09-08
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