ES2189354T3 - Procedimiento para la preparacion de furoato mometasona. - Google Patents

Procedimiento para la preparacion de furoato mometasona.

Info

Publication number
ES2189354T3
ES2189354T3 ES99308380T ES99308380T ES2189354T3 ES 2189354 T3 ES2189354 T3 ES 2189354T3 ES 99308380 T ES99308380 T ES 99308380T ES 99308380 T ES99308380 T ES 99308380T ES 2189354 T3 ES2189354 T3 ES 2189354T3
Authority
ES
Spain
Prior art keywords
preparation
procedure
mometasone furoate
mometasone
furoate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES99308380T
Other languages
English (en)
Inventor
William Heggie
Joao Bandarra
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hovione Inter AG
Original Assignee
Hovione Inter AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hovione Inter AG filed Critical Hovione Inter AG
Application granted granted Critical
Publication of ES2189354T3 publication Critical patent/ES2189354T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/44—Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Un procedimiento para la preparación de furoato de mometasona, que comprende hacer reaccionar mometasona con cloruro de 2-furoílo en presencia de una amina terciaria en un disolvente inerte.
ES99308380T 1999-08-02 1999-10-25 Procedimiento para la preparacion de furoato mometasona. Expired - Lifetime ES2189354T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PT102343A PT102343B (pt) 1999-08-02 1999-08-02 Processo para a preparacao de furoato mometasona

Publications (1)

Publication Number Publication Date
ES2189354T3 true ES2189354T3 (es) 2003-07-01

Family

ID=20085881

Family Applications (1)

Application Number Title Priority Date Filing Date
ES99308380T Expired - Lifetime ES2189354T3 (es) 1999-08-02 1999-10-25 Procedimiento para la preparacion de furoato mometasona.

Country Status (22)

Country Link
US (1) US6177560B1 (es)
EP (1) EP1074558B1 (es)
JP (1) JP3746174B2 (es)
KR (1) KR100640066B1 (es)
CN (1) CN1149222C (es)
AT (1) ATE229970T1 (es)
AU (1) AU765592B2 (es)
CA (1) CA2295455C (es)
DE (1) DE69904585T2 (es)
DK (1) DK1074558T3 (es)
ES (1) ES2189354T3 (es)
HR (1) HRP990341B1 (es)
HU (1) HU227494B1 (es)
IL (1) IL133752A (es)
NO (1) NO321154B1 (es)
NZ (1) NZ500555A (es)
PL (1) PL191103B1 (es)
PT (1) PT102343B (es)
RU (1) RU2208616C2 (es)
SI (1) SI1074558T1 (es)
UA (1) UA60333C2 (es)
ZA (1) ZA996758B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070099883A1 (en) * 2005-10-07 2007-05-03 Cheryl Lynn Calis Anhydrous mometasone furoate formulation
EP1790754A1 (de) * 2005-11-24 2007-05-30 Siemens Aktiengesellschaft Schichtsystem mit Gadolinium-Mischkristall-Pyrochlorphase
US8021742B2 (en) * 2006-12-15 2011-09-20 Siemens Energy, Inc. Impact resistant thermal barrier coating system
US8815258B2 (en) 2009-05-29 2014-08-26 Pearl Therapeutics, Inc. Compositions, methods and systems for respiratory delivery of two or more active agents
US9463161B2 (en) 2009-05-29 2016-10-11 Pearl Therapeutics, Inc. Compositions for pulmonary delivery of long-acting muscarinic antagonists and associated methods and systems
PT105139B (pt) * 2010-06-01 2013-01-29 Hovione Farmaciencia S A Método para a monofluorometilação de substratos orgânicos para preparação de compostos orgânicos biologicamente activos
JP6454323B2 (ja) 2013-03-15 2019-01-16 パール セラピューティクス，インコーポレイテッド 粒子状結晶性材料のコンディショニングのための方法及びシステム
SG11201509543YA (en) 2013-05-22 2015-12-30 Pearl Therapeutics Inc Compositions, methods & systems for respiratory delivery of three or more active agents
CN105481933B (zh) * 2015-12-25 2017-09-19 山东京卫制药有限公司 一种合成糠酸莫米松的方法
CN105566437B (zh) * 2015-12-30 2018-07-20 山东京卫制药有限公司 一种8dm衍生物及利用其合成糠酸莫米松的方法
CN107266518B (zh) * 2016-04-08 2021-03-30 天津金耀集团有限公司 一种糠酸莫米松晶型及其制备方法
DK4197528T3 (da) 2021-07-09 2024-05-06 Astrazeneca Pharmaceuticals Lp Sammensætninger, fremgangsmåder og systemer til indgivelse af medicin med aerosol
WO2023119093A1 (en) 2021-12-20 2023-06-29 Astrazeneca Ab Compositions, methods and systems for aerosol drug delivery

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3260474D1 (en) * 1981-02-02 1984-09-06 Schering Corp Aromatic heterocyclic esters of steroids, their preparation and pharmaceutical compositions containing them
DK0923599T3 (da) * 1996-06-28 2002-04-22 Schering Corp Fremgangsmåde til fremstilling af 17-estere af 9alfa, 21-dihalogenpregnan-11beta, 17alfa-diol-20-oner
US5886200A (en) * 1996-07-01 1999-03-23 Schering Corporation Process for the preparation of 17-esters of 9 α, 21-dihalo-pregnane-11 β, 17 α-diol-20-ones

Also Published As

Publication number Publication date
HU227494B1 (en) 2011-07-28
AU765592B2 (en) 2003-09-25
CN1149222C (zh) 2004-05-12
PT102343B (pt) 2003-11-28
EP1074558A1 (en) 2001-02-07
IL133752A0 (en) 2001-04-30
KR20010020094A (ko) 2001-03-15
HU9903747D0 (en) 1999-12-28
JP3746174B2 (ja) 2006-02-15
DK1074558T3 (da) 2003-04-07
HUP9903747A2 (hu) 2001-05-28
NO321154B1 (no) 2006-03-27
NO995225L (no) 2001-02-05
PT102343A (pt) 2001-02-28
UA60333C2 (uk) 2003-10-15
NZ500555A (en) 2000-11-24
KR100640066B1 (ko) 2006-10-31
JP2001048897A (ja) 2001-02-20
DE69904585D1 (de) 2003-01-30
US6177560B1 (en) 2001-01-23
CA2295455A1 (en) 2001-02-02
NO995225D0 (no) 1999-10-26
HRP990341B1 (en) 2003-10-31
ZA996758B (en) 2000-08-30
CA2295455C (en) 2008-03-25
DE69904585T2 (de) 2003-05-15
SI1074558T1 (en) 2003-04-30
IL133752A (en) 2004-02-19
EP1074558B1 (en) 2002-12-18
HUP9903747A3 (en) 2001-07-30
CN1282744A (zh) 2001-02-07
HRP990341A2 (en) 2001-04-30
PL336452A1 (en) 2001-02-12
PL191103B1 (pl) 2006-03-31
AU5602499A (en) 2001-02-08
ATE229970T1 (de) 2003-01-15
RU2208616C2 (ru) 2003-07-20

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