ES2127845T3 - Procedimiento para la preparacion de 5-cloroimidazol-4-carbaldehidos sustituidos en posicion 2. - Google Patents

Procedimiento para la preparacion de 5-cloroimidazol-4-carbaldehidos sustituidos en posicion 2.

Info

Publication number
ES2127845T3
ES2127845T3 ES94103714T ES94103714T ES2127845T3 ES 2127845 T3 ES2127845 T3 ES 2127845T3 ES 94103714 T ES94103714 T ES 94103714T ES 94103714 T ES94103714 T ES 94103714T ES 2127845 T3 ES2127845 T3 ES 2127845T3
Authority
ES
Spain
Prior art keywords
preparation
carbaldehydes
chloroimidazole
substituted
optionally
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES94103714T
Other languages
English (en)
Inventor
Gareth Dr Griffiths
Rene Dr Imwinkelried
Jacques Dr Gosteli
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Lonza AG
Original Assignee
Lonza AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza AG filed Critical Lonza AG
Application granted granted Critical
Publication of ES2127845T3 publication Critical patent/ES2127845T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/68—Halogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Steroid Compounds (AREA)

Abstract

LOS 5 FORMULA GENERAL SON PRODUCTOS INTERMEDIOS PARA LA ELABORACION DE PRODUCTOS FARMACEUTICOS REDUCTORES DE LA PRESION ARTERIAL O DE COMPUESTOS CON ACTIVIDAD HERBICIDA. SE DESCRIBE UN PROCESO PARA LA ELABORACION DE ESTOS PRODUCTOS INTERMEDIOS ASI COMO UN NUEVO PROCESO PARA LA TRANSFORMACION POSTERIOR DE LOS 5 IMIDAZOLES EVENTUALMENTE 2 I, DONDE R1 SIGNIFICA HIDROGENO AL 5 CLORIMIDAZOL HIDOS EVENTUALMENTE 2
ES94103714T 1993-03-12 1994-03-10 Procedimiento para la preparacion de 5-cloroimidazol-4-carbaldehidos sustituidos en posicion 2. Expired - Lifetime ES2127845T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH74893 1993-03-12

Publications (1)

Publication Number Publication Date
ES2127845T3 true ES2127845T3 (es) 1999-05-01

Family

ID=4194282

Family Applications (2)

Application Number Title Priority Date Filing Date
ES94103636T Expired - Lifetime ES2108894T3 (es) 1993-03-12 1994-03-09 Procedimiento para la preparacion de 5-cloroimidazoles eventualmente sustituidos en posicion 2.
ES94103714T Expired - Lifetime ES2127845T3 (es) 1993-03-12 1994-03-10 Procedimiento para la preparacion de 5-cloroimidazol-4-carbaldehidos sustituidos en posicion 2.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES94103636T Expired - Lifetime ES2108894T3 (es) 1993-03-12 1994-03-09 Procedimiento para la preparacion de 5-cloroimidazoles eventualmente sustituidos en posicion 2.

Country Status (9)

Country Link
EP (2) EP0614890B1 (es)
JP (1) JP3716434B2 (es)
KR (1) KR100362353B1 (es)
AT (2) ATE157655T1 (es)
CA (2) CA2117209C (es)
DE (2) DE59403903D1 (es)
DK (2) DK0614890T3 (es)
ES (2) ES2108894T3 (es)
HU (2) HU219708B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2175420C (en) * 1995-05-17 2007-04-10 Gareth Griffiths Process for the preparation of optionally 2-substituted 5-chloroimidazole-4-carbaldehydes
JP4103149B2 (ja) * 1996-01-05 2008-06-18 ロンザ リミテッド ２−置換５−クロロイミダゾール−４−カルブアルデヒドの製造方法
KR101035559B1 (ko) * 2009-06-02 2011-05-19 한국화학연구원 클로로이미다졸 유도체 또는 이의 약학적으로 허용가능한 염을 유효성분으로 포함하는 골다공증 또는 비만의 예방 또는 치료용 약학적 조성물

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3409606A (en) * 1965-12-30 1968-11-05 American Cyanamid Co Halogenated chloroimidazole compounds
IL53783A (en) * 1977-02-03 1982-08-31 American Cyanamid Co Imidazo(1,5-d)-as-triazine-4 (3h)-(thi)one derivatives,their preparation and pharmaceutical compositions containing them
JPS5671074A (en) * 1979-11-12 1981-06-13 Takeda Chem Ind Ltd 1,2-disubstituted-4-halogenoimidazole-5-acetic acid derivative
DE3145927A1 (de) * 1981-11-20 1983-06-01 Basf Ag, 6700 Ludwigshafen 4(5)-methyl-5(4)-chlorimidazol und verfahren zu seiner herstellung
DE3330192A1 (de) * 1983-08-20 1985-03-07 Basf Ag, 6700 Ludwigshafen 4-alkylimidazol-derivate, ihre herstellung und verwendung
JPS62238383A (ja) * 1986-04-07 1987-10-19 Chiyoda Kagaku Kenkyusho:Kk 防食剤
CA1334092C (en) * 1986-07-11 1995-01-24 David John Carini Angiotensin ii receptor blocking imidazoles
JPH02262562A (ja) * 1988-10-20 1990-10-25 Ishihara Sangyo Kaisha Ltd イミダゾール系化合物
PT95899A (pt) * 1989-11-17 1991-09-13 Glaxo Group Ltd Processo para a preparacao de derivados indole
JPH0426678A (ja) * 1990-05-18 1992-01-29 Nippon Synthetic Chem Ind Co Ltd:The イミダゾール―４―クロロ―５―カルバルデヒド誘導体の製造法
US5126342A (en) * 1990-10-01 1992-06-30 Merck & Co., Inc. Imidazole angiotensin ii antagonists incorporating acidic functional groups
EP0505098A1 (en) * 1991-03-19 1992-09-23 Merck & Co. Inc. Imidazole derivatives bearing acidic functional groups as angiotensin II antagonists
RU2103262C1 (ru) * 1992-07-16 1998-01-27 Лонца АГ Гампель/Валлис Способ получения 2-замещенных 5-хлоримидазол-4-карбальдегидов

Also Published As

Publication number Publication date
ATE157655T1 (de) 1997-09-15
DK0614890T3 (da) 1997-10-13
HU9701565D0 (en) 1997-11-28
EP0614891A2 (de) 1994-09-14
DK0614891T3 (da) 1999-08-30
HU219708B (hu) 2001-06-28
JP3716434B2 (ja) 2005-11-16
DE59407547D1 (de) 1999-02-11
HUT66633A (en) 1994-12-28
CA2117209C (en) 2005-05-31
EP0614891B1 (de) 1998-12-30
CA2473422A1 (en) 1994-09-13
EP0614890A3 (de) 1995-01-11
KR100362353B1 (ko) 2003-03-19
CA2117209A1 (en) 1994-09-13
ES2108894T3 (es) 1998-01-01
ATE175199T1 (de) 1999-01-15
EP0614890B1 (de) 1997-09-03
HU9400736D0 (en) 1994-06-28
EP0614891A3 (de) 1995-05-03
JPH072789A (ja) 1995-01-06
EP0614890A2 (de) 1994-09-14
CA2473422C (en) 2007-05-22
HU213387B (en) 1997-05-28
DE59403903D1 (de) 1997-10-09

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