ES2062351T3 - Derivados de triazolo (4,5-c) piridina anticonvulsivos. - Google Patents

Derivados de triazolo (4,5-c) piridina anticonvulsivos.

Info

Publication number
ES2062351T3
ES2062351T3 ES90304271T ES90304271T ES2062351T3 ES 2062351 T3 ES2062351 T3 ES 2062351T3 ES 90304271 T ES90304271 T ES 90304271T ES 90304271 T ES90304271 T ES 90304271T ES 2062351 T3 ES2062351 T3 ES 2062351T3
Authority
ES
Spain
Prior art keywords
anticonvulsives
piridine
triazole derivatives
disclosed
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES90304271T
Other languages
English (en)
Inventor
James Leroy Kelley
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wellcome Foundation Ltd
Original Assignee
Wellcome Foundation Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Foundation Ltd filed Critical Wellcome Foundation Ltd
Application granted granted Critical
Publication of ES2062351T3 publication Critical patent/ES2062351T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

SE PRESENTAN UNA SERIE DE COMPUESTOS DE TRIAZOLOPIRIMIDINA Y COMPUESTOS FARMACEUTICOS QUE LA CONTIENEN. LOS COMPUESTOS PRESENTADOS SON UTILES EN EL TRATAMIENTO DE DESORDENES NERVIOSOS CENTRALES, TALES COMO LA EPILEPSIA EN LOS MAMIFEROS. TAMBIEN SE PRESENTAN METODOS PARA LA PREPARACION DE ESTAS TRIAZOLOPIRIMIDINAS.
ES90304271T 1989-04-21 1990-04-20 Derivados de triazolo (4,5-c) piridina anticonvulsivos. Expired - Lifetime ES2062351T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898909136A GB8909136D0 (en) 1989-04-21 1989-04-21 Anticonvulsant pyridines and analogues thereof

Publications (1)

Publication Number Publication Date
ES2062351T3 true ES2062351T3 (es) 1994-12-16

Family

ID=10655494

Family Applications (1)

Application Number Title Priority Date Filing Date
ES90304271T Expired - Lifetime ES2062351T3 (es) 1989-04-21 1990-04-20 Derivados de triazolo (4,5-c) piridina anticonvulsivos.

Country Status (21)

Country Link
EP (1) EP0399653B1 (es)
JP (1) JP2865367B2 (es)
KR (1) KR0183972B1 (es)
AT (1) ATE113046T1 (es)
CA (1) CA2015047A1 (es)
CY (1) CY2003B1 (es)
DD (1) DD293823A5 (es)
DE (1) DE69013396T2 (es)
DK (1) DK0399653T3 (es)
ES (1) ES2062351T3 (es)
FI (1) FI93448C (es)
GB (1) GB8909136D0 (es)
HK (1) HK78397A (es)
HU (2) HU206210B (es)
IE (1) IE67335B1 (es)
IL (1) IL94150A (es)
LV (1) LV5780B4 (es)
NZ (1) NZ233404A (es)
PH (1) PH27118A (es)
PT (1) PT93822B (es)
ZA (1) ZA903021B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002518391A (ja) 1998-06-16 2002-06-25 メルク シャープ エンド ドーム リミテッド Ｇａｂａ受容体のリガンドとしてのトリアゾロ−ピリジン誘導体

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3929812A (en) * 1974-05-20 1975-12-30 Squibb & Sons Inc Derivatives of 1H-triazolo {8 4,5-c{9 pyridine-7-carboxylic acids and esters
DE3873812D1 (de) * 1987-04-07 1992-09-24 Ciba Geigy Ag 3h-1,2,3-triazolo(4,5-d)pyrimidine.

Also Published As

Publication number Publication date
HU902502D0 (en) 1990-08-28
DE69013396D1 (de) 1994-11-24
IL94150A (en) 1994-02-27
FI901981A0 (fi) 1990-04-20
DK0399653T3 (da) 1994-11-14
HU206210B (en) 1992-09-28
IL94150A0 (en) 1991-01-31
FI93448B (fi) 1994-12-30
FI93448C (fi) 1995-04-10
ZA903021B (en) 1991-12-24
KR0183972B1 (ko) 1999-05-01
IE67335B1 (en) 1996-03-20
NZ233404A (en) 1992-08-26
GB8909136D0 (en) 1989-06-07
AU626409B2 (en) 1992-07-30
LV5780A4 (lv) 1996-12-20
PT93822A (pt) 1990-11-20
EP0399653B1 (en) 1994-10-19
CA2015047A1 (en) 1990-10-21
JPH02292286A (ja) 1990-12-03
CY2003B1 (en) 1998-04-30
PT93822B (pt) 1996-09-30
IE901409L (en) 1990-10-21
JP2865367B2 (ja) 1999-03-08
KR900016208A (ko) 1990-11-12
LV5780B4 (lv) 1997-04-20
ATE113046T1 (de) 1994-11-15
HK78397A (en) 1997-06-20
HU211137A9 (en) 1995-10-30
DD293823A5 (de) 1991-09-12
EP0399653A1 (en) 1990-11-28
HUT53905A (en) 1990-12-28
PH27118A (en) 1993-03-16
DE69013396T2 (de) 1995-05-04
AU5372290A (en) 1990-10-25

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