EP2138163A3 - Compositions de suppositoires contenant du ténofovir ou du ténofovir disoproxil - Google Patents
Compositions de suppositoires contenant du ténofovir ou du ténofovir disoproxil Download PDFInfo
- Publication number
- EP2138163A3 EP2138163A3 EP09173071A EP09173071A EP2138163A3 EP 2138163 A3 EP2138163 A3 EP 2138163A3 EP 09173071 A EP09173071 A EP 09173071A EP 09173071 A EP09173071 A EP 09173071A EP 2138163 A3 EP2138163 A3 EP 2138163A3
- Authority
- EP
- European Patent Office
- Prior art keywords
- tenofovir
- suppository formulations
- disoproxil
- formulations
- tenoforvir
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61F—FILTERS IMPLANTABLE INTO BLOOD VESSELS; PROSTHESES; DEVICES PROVIDING PATENCY TO, OR PREVENTING COLLAPSING OF, TUBULAR STRUCTURES OF THE BODY, e.g. STENTS; ORTHOPAEDIC, NURSING OR CONTRACEPTIVE DEVICES; FOMENTATION; TREATMENT OR PROTECTION OF EYES OR EARS; BANDAGES, DRESSINGS OR ABSORBENT PADS; FIRST-AID KITS
- A61F6/00—Contraceptive devices; Pessaries; Applicators therefor
- A61F6/02—Contraceptive devices; Pessaries; Applicators therefor for use by males
- A61F6/04—Condoms, sheaths or the like, e.g. combined with devices protecting against contagion
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/12—Aerosols; Foams
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Reproductive Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Dermatology (AREA)
- Biomedical Technology (AREA)
- Vascular Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Dispersion Chemistry (AREA)
- Gynecology & Obstetrics (AREA)
- Urology & Nephrology (AREA)
- AIDS & HIV (AREA)
- Endocrinology (AREA)
- Molecular Biology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US58683904P | 2004-07-09 | 2004-07-09 | |
EP05771562A EP1773296B1 (fr) | 2004-07-09 | 2005-07-01 | Gel pharmaceutique vaginal du tenofovir |
Related Parent Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP05771562.5 Division | 2005-07-01 | ||
EP05771562A Division EP1773296B1 (fr) | 2004-07-09 | 2005-07-01 | Gel pharmaceutique vaginal du tenofovir |
Publications (2)
Publication Number | Publication Date |
---|---|
EP2138163A2 EP2138163A2 (fr) | 2009-12-30 |
EP2138163A3 true EP2138163A3 (fr) | 2011-08-31 |
Family
ID=35839705
Family Applications (4)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP10182466A Withdrawn EP2283812A3 (fr) | 2004-07-09 | 2005-07-01 | Préparations antivirales topiques |
EP09173071A Withdrawn EP2138163A3 (fr) | 2004-07-09 | 2005-07-01 | Compositions de suppositoires contenant du ténofovir ou du ténofovir disoproxil |
EP05771562A Active EP1773296B1 (fr) | 2004-07-09 | 2005-07-01 | Gel pharmaceutique vaginal du tenofovir |
EP09173070A Withdrawn EP2138162A3 (fr) | 2004-07-09 | 2005-07-01 | Gel comprenant du ténofovir ou du ténofovir disoproxil |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP10182466A Withdrawn EP2283812A3 (fr) | 2004-07-09 | 2005-07-01 | Préparations antivirales topiques |
Family Applications After (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP05771562A Active EP1773296B1 (fr) | 2004-07-09 | 2005-07-01 | Gel pharmaceutique vaginal du tenofovir |
EP09173070A Withdrawn EP2138162A3 (fr) | 2004-07-09 | 2005-07-01 | Gel comprenant du ténofovir ou du ténofovir disoproxil |
Country Status (31)
Country | Link |
---|---|
US (5) | US20080035155A1 (fr) |
EP (4) | EP2283812A3 (fr) |
JP (2) | JP5121451B2 (fr) |
KR (1) | KR101225707B1 (fr) |
CN (1) | CN1984640B (fr) |
AP (1) | AP2666A (fr) |
AR (1) | AR050424A1 (fr) |
AT (1) | ATE447396T1 (fr) |
AU (1) | AU2005272032B2 (fr) |
BR (1) | BRPI0513196A (fr) |
CA (1) | CA2570877C (fr) |
CY (1) | CY1109757T1 (fr) |
DE (1) | DE602005017497D1 (fr) |
DK (1) | DK1773296T3 (fr) |
EA (2) | EA017763B1 (fr) |
ES (1) | ES2336017T3 (fr) |
HK (1) | HK1103026A1 (fr) |
HR (2) | HRP20070040A2 (fr) |
IL (2) | IL180172A (fr) |
IS (1) | IS8584A (fr) |
MX (1) | MX2007000122A (fr) |
NO (1) | NO20070762L (fr) |
NZ (1) | NZ552172A (fr) |
PL (2) | PL382306A1 (fr) |
PT (1) | PT1773296E (fr) |
RS (1) | RS51213B (fr) |
SI (1) | SI1773296T1 (fr) |
TW (1) | TW200612955A (fr) |
UA (1) | UA93354C2 (fr) |
WO (1) | WO2006017044A2 (fr) |
ZA (1) | ZA200700932B (fr) |
Families Citing this family (60)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8512718B2 (en) | 2000-07-03 | 2013-08-20 | Foamix Ltd. | Pharmaceutical composition for topical application |
IL152486A0 (en) | 2002-10-25 | 2003-05-29 | Meir Eini | Alcohol-free cosmetic and pharmaceutical foam carrier |
US8119150B2 (en) | 2002-10-25 | 2012-02-21 | Foamix Ltd. | Non-flammable insecticide composition and uses thereof |
US7704518B2 (en) * | 2003-08-04 | 2010-04-27 | Foamix, Ltd. | Foamable vehicle and pharmaceutical compositions thereof |
US20080138296A1 (en) | 2002-10-25 | 2008-06-12 | Foamix Ltd. | Foam prepared from nanoemulsions and uses |
CA2502986C (fr) | 2002-10-25 | 2011-08-23 | Foamix Ltd. | Mousse cosmetique et pharmaceutique |
US10117812B2 (en) | 2002-10-25 | 2018-11-06 | Foamix Pharmaceuticals Ltd. | Foamable composition combining a polar solvent and a hydrophobic carrier |
US9265725B2 (en) | 2002-10-25 | 2016-02-23 | Foamix Pharmaceuticals Ltd. | Dicarboxylic acid foamable vehicle and pharmaceutical compositions thereof |
US9211259B2 (en) | 2002-11-29 | 2015-12-15 | Foamix Pharmaceuticals Ltd. | Antibiotic kit and composition and uses thereof |
US7700076B2 (en) | 2002-10-25 | 2010-04-20 | Foamix, Ltd. | Penetrating pharmaceutical foam |
US8486376B2 (en) | 2002-10-25 | 2013-07-16 | Foamix Ltd. | Moisturizing foam containing lanolin |
US9668972B2 (en) | 2002-10-25 | 2017-06-06 | Foamix Pharmaceuticals Ltd. | Nonsteroidal immunomodulating kit and composition and uses thereof |
US20060018937A1 (en) * | 2002-10-25 | 2006-01-26 | Foamix Ltd. | Steroid kit and foamable composition and uses thereof |
US8119109B2 (en) * | 2002-10-25 | 2012-02-21 | Foamix Ltd. | Foamable compositions, kits and methods for hyperhidrosis |
US7820145B2 (en) * | 2003-08-04 | 2010-10-26 | Foamix Ltd. | Oleaginous pharmaceutical and cosmetic foam |
US8900554B2 (en) | 2002-10-25 | 2014-12-02 | Foamix Pharmaceuticals Ltd. | Foamable composition and uses thereof |
US20080317679A1 (en) * | 2002-10-25 | 2008-12-25 | Foamix Ltd. | Foamable compositions and kits comprising one or more of a channel agent, a cholinergic agent, a nitric oxide donor, and related agents and their uses |
US20060233721A1 (en) * | 2002-10-25 | 2006-10-19 | Foamix Ltd. | Foam containing unique oil globules |
US7575739B2 (en) | 2003-04-28 | 2009-08-18 | Foamix Ltd. | Foamable iodine composition |
US8486374B2 (en) | 2003-08-04 | 2013-07-16 | Foamix Ltd. | Hydrophilic, non-aqueous pharmaceutical carriers and compositions and uses |
US8795693B2 (en) | 2003-08-04 | 2014-08-05 | Foamix Ltd. | Compositions with modulating agents |
UA93354C2 (ru) * | 2004-07-09 | 2011-02-10 | Гилиад Сайенсиз, Инк. | Местный противовирусный препарат |
BRPI0612428A2 (pt) * | 2005-05-09 | 2010-11-09 | Foamix Ltd | composição farmacêutica higroscópica, veìculo farmacêutico espumoso e composição farmacêutica espumosa |
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CA2769677A1 (fr) | 2009-07-29 | 2011-02-03 | Foamix Ltd. | Compositions hydro-alcooliques moussantes a base d'agents non tensioactifs non polymeres, mousses legeres, et leurs utilisations |
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CA2776366C (fr) | 2009-10-02 | 2017-07-18 | Foamix Ltd. | Compositions moussantes sans eau et sans surfactant, mousses et gels friables, ainsi que leurs utilisations |
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EP2389929A1 (fr) * | 2010-05-30 | 2011-11-30 | Abdi Ibrahim Ilac Sanayi ve Ticaret Anonim Sirketi | Formulations pharmaceutiques de Ténofovir |
WO2011156416A1 (fr) * | 2010-06-11 | 2011-12-15 | Gilead Sciences, Inc. | Formulations antivirales topiques pour la prévention de la transmission du vhs-2 |
SG194725A1 (en) | 2011-05-02 | 2013-12-30 | Aptalis Pharmatech Inc | Rapid dissolve tablet compositions for vaginal administration |
EP2794624B1 (fr) | 2011-12-22 | 2019-05-15 | Geron Corporation | Analogues de guanine en tant que substrats de télomérase et affecteurs de la longueur de télomères |
EP2861215A4 (fr) * | 2012-06-13 | 2015-04-22 | Evofem Inc | Compositions et méthodes d'amélioration de l'efficacité de microbicides contraceptifs |
CN102786549B (zh) * | 2012-08-13 | 2013-07-03 | 洛阳聚慧投资股份有限公司 | 一组具有抑制hiv-1病毒复制活性的替诺福韦双酯化合物、制备方法及其药物用途 |
CN107312039B (zh) * | 2012-08-30 | 2019-06-25 | 江苏豪森药业集团有限公司 | 一种替诺福韦前药的制备方法 |
US20150246065A1 (en) * | 2012-09-14 | 2015-09-03 | Cipla Limited | Topical Pharmaceutical Composition |
EP2968127A4 (fr) * | 2013-03-15 | 2016-09-07 | Conrad | Préparations à faible taux de glycérol destinées au traitement et à la prévention du vih |
KR102407408B1 (ko) | 2013-12-19 | 2022-06-10 | 에보펨 인코포레이티드 | 알긴산계 항균성 화합물을 사용하는 염증 및 질병을 억제하기 위한 조성물 및 방법 |
KR20230130175A (ko) | 2014-12-26 | 2023-09-11 | 에모리 유니버시티 | N4-하이드록시시티딘, 이와 관련된 유도체 및 이의 항 바이러스적 용도 |
MX2017011630A (es) | 2016-09-08 | 2018-09-25 | Foamix Pharmaceuticals Ltd | Composiciones y metodos para tratar rosacea y acne. |
CN110225750A (zh) | 2016-10-04 | 2019-09-10 | 伊沃菲姆股份有限公司 | 细菌性阴道病的治疗和预防方法 |
AU2018378832B9 (en) | 2017-12-07 | 2021-05-27 | Emory University | N4-hydroxycytidine and derivatives and anti-viral uses related thereto |
CN108096206A (zh) * | 2018-02-01 | 2018-06-01 | 海南天煌制药有限公司 | 一种富马酸替诺福韦二吡呋酯片剂及其制备方法 |
US20210379089A1 (en) * | 2018-10-23 | 2021-12-09 | Eastern Virginia Medical School | Pharmaceutical compositions and methods of making on demand solid dosage formulations |
KR20230013013A (ko) * | 2019-09-20 | 2023-01-26 | 애보트 라피드 다이어그노스틱스 인터내셔널 언리미티드 컴퍼니 | 테노포비르 및 그의 유도체에 대해 지시된 항체 |
CN112891323B (zh) * | 2020-01-22 | 2023-08-18 | 首都医科大学附属北京地坛医院 | 一种抗hiv外用消毒剂及其制备方法 |
CN117338733B (zh) * | 2023-10-12 | 2024-05-28 | 杭州和泽坤元药业有限公司 | 一种富马酸替诺福韦二吡呋酯片及其制备工艺 |
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- 2005-07-01 US US11/631,876 patent/US20080035155A1/en not_active Abandoned
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