EP1443901A4 - Systeme de liberation prolongee de medicaments solubles - Google Patents

Systeme de liberation prolongee de medicaments solubles

Info

Publication number
EP1443901A4
EP1443901A4 EP02782303A EP02782303A EP1443901A4 EP 1443901 A4 EP1443901 A4 EP 1443901A4 EP 02782303 A EP02782303 A EP 02782303A EP 02782303 A EP02782303 A EP 02782303A EP 1443901 A4 EP1443901 A4 EP 1443901A4
Authority
EP
European Patent Office
Prior art keywords
extended release
release system
soluble drug
drug extended
soluble
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
EP02782303A
Other languages
German (de)
English (en)
Other versions
EP1443901A2 (fr
Inventor
Victoria Rogers
Philippe J M Dor
Joseph A Fix
Hiroyuki Kojima
Kazuhiro Sako
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astellas Pharma Inc
Original Assignee
Yamanouchi Pharmaceutical Co Ltd
Yamanouchi Pharma Technologies Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamanouchi Pharmaceutical Co Ltd, Yamanouchi Pharma Technologies Inc filed Critical Yamanouchi Pharmaceutical Co Ltd
Publication of EP1443901A2 publication Critical patent/EP1443901A2/fr
Publication of EP1443901A4 publication Critical patent/EP1443901A4/fr
Ceased legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
EP02782303A 2001-11-13 2002-11-12 Systeme de liberation prolongee de medicaments solubles Ceased EP1443901A4 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US7877 1987-01-28
US787701A 2001-11-13 2001-11-13
PCT/US2002/036681 WO2003041656A2 (fr) 2001-11-13 2002-11-12 Systeme de liberation prolongee de medicaments solubles

Publications (2)

Publication Number Publication Date
EP1443901A2 EP1443901A2 (fr) 2004-08-11
EP1443901A4 true EP1443901A4 (fr) 2010-06-16

Family

ID=21728577

Family Applications (1)

Application Number Title Priority Date Filing Date
EP02782303A Ceased EP1443901A4 (fr) 2001-11-13 2002-11-12 Systeme de liberation prolongee de medicaments solubles

Country Status (10)

Country Link
EP (1) EP1443901A4 (fr)
JP (2) JP4882200B2 (fr)
KR (2) KR101016619B1 (fr)
CN (1) CN100534531C (fr)
AU (1) AU2002348279C1 (fr)
CA (1) CA2466657C (fr)
MX (1) MXPA04004544A (fr)
PL (1) PL374280A1 (fr)
RU (1) RU2322263C2 (fr)
WO (1) WO2003041656A2 (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050042289A1 (en) * 2003-04-29 2005-02-24 Yamanouchi Pharma Technologies, Inc. Tablets and methods for modified release of hydrophylic and other active agents
JP4822092B2 (ja) * 2003-09-01 2011-11-24 大正製薬株式会社 Ｗ／ｏ／ｗ型複合エマルション
CA2536040A1 (fr) * 2003-11-04 2005-05-26 Shire Laboratories Inc. Liberation prolongee de molecules actives d'un point de vue pharmacologique positivement chargees a partir d'une matrice contenant des polymeres avec des atomes d'oxygene polarises
US8197846B2 (en) 2003-11-10 2012-06-12 Astellas Pharma Inc. Sustained release pharmaceutical composition
KR100638041B1 (ko) * 2003-12-24 2006-10-23 주식회사 삼양사 수용성 약물의 경구투여용 나노입자 조성물 및 그의제조방법
US20120034276A1 (en) * 2009-03-25 2012-02-09 Aska Pharmaceutical Co., Ltd. Solid preparation
KR101319420B1 (ko) * 2011-03-18 2013-10-17 한남대학교 산학협력단 서방형 방출이 가능한 수용성 양이온 약물 전달 시스템
WO2012140674A1 (fr) * 2011-04-11 2012-10-18 Council Of Scientific & Industrial Research Dissociation de nano-containers induite en surface
CN102977413B (zh) * 2011-09-07 2015-05-13 江南大学 聚合物复合制备胶束的一种新方法
CN103083222B (zh) * 2011-10-28 2015-08-19 江南大学 一锅法制备三组分聚合物胶束
JP6041823B2 (ja) 2013-03-16 2016-12-14 ファイザー・インク トファシチニブの経口持続放出剤形
KR20220022829A (ko) * 2020-08-19 2022-02-28 주식회사 모든바이오 글리시리진 및 수용성 약물을 포함하는 나노 입자, 이를 포함하는 약제학적 조성물 및 이들의 제조 방법

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1263392A (en) * 1968-05-21 1972-02-09 American Home Prod Sustained release drug composition
WO1997006787A2 (fr) * 1995-08-17 1997-02-27 Dyer, Alison, Margaret Produits a liberation controlee
WO2000015198A1 (fr) * 1998-09-14 2000-03-23 Ranbaxy Laboratories Limited Systeme d'apport medicamenteux regule administre oralement pour une regulation spatiale et temporelle
EP0661045B1 (fr) * 1992-09-18 2002-07-03 Yamanouchi Pharmaceutical Co. Ltd. Preparation d'hydrogel a liberation prolongee

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6410466A (en) * 1987-07-01 1989-01-13 Brother Ind Ltd Data recording and reproducing method for magnetic disk
US5219563A (en) * 1988-05-11 1993-06-15 Glaxo Group Limited Drug adsorbates
US5788959A (en) * 1995-04-24 1998-08-04 University Of Maryland, Baltimore County Drug delivery device and method for employing the same
IT1297461B1 (it) * 1997-10-29 1999-12-17 Ciocca Maurizio Preparazione di compresse a rilascio controllato a base di complessi tra carragenano e farmaci basici solubili
US6287599B1 (en) * 2000-12-20 2001-09-11 Shire Laboratories, Inc. Sustained release pharmaceutical dosage forms with minimized pH dependent dissolution profiles
AR034517A1 (es) * 2001-06-21 2004-02-25 Astrazeneca Ab Formulacion farmaceutica

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1263392A (en) * 1968-05-21 1972-02-09 American Home Prod Sustained release drug composition
EP0661045B1 (fr) * 1992-09-18 2002-07-03 Yamanouchi Pharmaceutical Co. Ltd. Preparation d'hydrogel a liberation prolongee
WO1997006787A2 (fr) * 1995-08-17 1997-02-27 Dyer, Alison, Margaret Produits a liberation controlee
WO2000015198A1 (fr) * 1998-09-14 2000-03-23 Ranbaxy Laboratories Limited Systeme d'apport medicamenteux regule administre oralement pour une regulation spatiale et temporelle

Non-Patent Citations (4)

* Cited by examiner, † Cited by third party
Title
ATTWOOD D ET AL: "AGGREGATION OF ANTI DEPRESSANT DRUGS IN AQUEOUS SOLUTION", JOURNAL OF PHARMACY AND PHARMACOLOGY, LONDON; GB, vol. 30, no. 3, 1 January 1978 (1978-01-01), pages 176 - 180, XP008122056, ISSN: 0022-3573 *
KRISTMUNDSDOTTIR T ET AL: "CHITOSAN MATRIX TABLETS: THE INFLUENCE OF EXCIPIENTS ON DRUG RELEASE", DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY, NEW YORK, NY, US LNKD- DOI:10.3109/03639049509069249, vol. 21, no. 13, 1 January 1995 (1995-01-01), pages 1591 - 1598, XP009026687, ISSN: 0363-9045 *
MAGGI L ET AL: "Dissolution behaviour of hydrophilic matrix tablets containing two different polyethylene oxides (PEOs) for the controlled release of a water-soluble drug. Dimensionality study", BIOMATERIALS, ELSEVIER SCIENCE PUBLISHERS BV., BARKING, GB, vol. 23, no. 4, 15 February 2002 (2002-02-15), pages 1113 - 1119, XP004348129, ISSN: 0142-9612, DOI: 10.1016/S0142-9612(01)00223-X *
TOLIAT T ET AL: "Controlled release (CR) tablet formulation of diltiazem HCL using different polymers as retardant substances", PHARMACEUTICAL RESEARCH (NEW YORK), vol. 14, no. 11 SUPPL., November 1997 (1997-11-01), & ANNUAL MEETING OF THE AMERICAN ASSOCIATION OF PHARMACEUTICAL SCIENTISTS; BOSTON, MASSACHUSETTS, USA; NOVEMBER 2-6, 1997, pages S598, XP008121997, ISSN: 0724-8741 *

Also Published As

Publication number Publication date
CN1612726A (zh) 2005-05-04
KR20050044424A (ko) 2005-05-12
MXPA04004544A (es) 2005-03-31
KR101016619B1 (ko) 2011-02-23
JP4894958B2 (ja) 2012-03-14
AU2002348279C1 (en) 2008-09-04
JP2011068700A (ja) 2011-04-07
JP4882200B2 (ja) 2012-02-22
CA2466657C (fr) 2011-02-01
JP2005508995A (ja) 2005-04-07
KR101132969B1 (ko) 2012-04-09
EP1443901A2 (fr) 2004-08-11
RU2004117848A (ru) 2005-05-27
CA2466657A1 (fr) 2003-05-22
AU2002348279B2 (en) 2008-01-24
KR20100123779A (ko) 2010-11-24
RU2322263C2 (ru) 2008-04-20
CN100534531C (zh) 2009-09-02
PL374280A1 (en) 2005-10-03
WO2003041656A2 (fr) 2003-05-22
WO2003041656A3 (fr) 2003-10-23

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Legal Events

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