EG21037A - Process for the synthesis of benzathiophenes - Google Patents

Process for the synthesis of benzathiophenes

Info

Publication number
EG21037A
EG21037A EG96197A EG96197A EG21037A EG 21037 A EG21037 A EG 21037A EG 96197 A EG96197 A EG 96197A EG 96197 A EG96197 A EG 96197A EG 21037 A EG21037 A EG 21037A
Authority
EG
Egypt
Prior art keywords
benzathiophenes
synthesis
Prior art date
Application number
EG96197A
Other languages
English (en)
Inventor
Jeffrey Thomas Vicenzi
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of EG21037A publication Critical patent/EG21037A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
EG96197A 1996-09-25 1997-09-18 Process for the synthesis of benzathiophenes EG21037A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2669596P 1996-09-25 1996-09-25

Publications (1)

Publication Number Publication Date
EG21037A true EG21037A (en) 2000-09-30

Family

ID=21833302

Family Applications (1)

Application Number Title Priority Date Filing Date
EG96197A EG21037A (en) 1996-09-25 1997-09-18 Process for the synthesis of benzathiophenes

Country Status (31)

Country Link
US (1) US5977383A (de)
EP (1) EP0832889B1 (de)
JP (1) JP2001501208A (de)
KR (1) KR20000048539A (de)
CN (1) CN1088704C (de)
AR (1) AR013321A1 (de)
AT (1) ATE318805T1 (de)
AU (1) AU718919B2 (de)
BR (1) BR9712844A (de)
CA (1) CA2266617A1 (de)
CO (1) CO4900043A1 (de)
CZ (1) CZ92899A3 (de)
DE (1) DE69735339T2 (de)
EA (1) EA001914B1 (de)
EG (1) EG21037A (de)
ES (1) ES2257761T3 (de)
HU (1) HUP9904228A3 (de)
ID (1) ID21349A (de)
IL (1) IL129001A (de)
IN (1) IN183239B (de)
MY (1) MY118009A (de)
NO (1) NO991193L (de)
NZ (1) NZ334591A (de)
PE (1) PE2699A1 (de)
PL (1) PL332208A1 (de)
TR (1) TR199900672T2 (de)
TW (1) TW472053B (de)
UA (1) UA62938C2 (de)
WO (1) WO1998013363A1 (de)
YU (1) YU15399A (de)
ZA (1) ZA978372B (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002230409A1 (en) * 2000-11-27 2002-06-03 Eli Lilly And Company Process for preparing 3-aryl-benzo(b)thiophenes

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1138163A (en) * 1965-05-21 1968-12-27 Bristol Myers Co Benzothiophene derivatives having anti-fertility properties
US3394125A (en) * 1965-10-23 1968-07-23 Bristol Myers Co 2-phenyl-3-tertiary-aminoalkoxy phenyl-and corresponding tertiaryaminoalkyl thio benzfurans substituted in the benzo nucleus with an alkoxy or tertiaryamino alkoxy or alkylthio group
US4230862A (en) * 1975-10-28 1980-10-28 Eli Lilly And Company Antifertility compounds
US4133814A (en) * 1975-10-28 1979-01-09 Eli Lilly And Company 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents
AT364852B (de) * 1977-11-05 1981-11-25 Thomae Gmbh Dr K Verfahren zur herstellung von kondensierten isothiazol-3(2h)-on-1,1-dioxiden und von deren salzen
US4436748A (en) * 1980-10-20 1984-03-13 Hoechst-Roussel Pharmaceuticals Inc. Benzo[b]thiophenes
PH18628A (en) * 1981-04-03 1985-08-23 Lilly Co Eli "6-hydroxy-2-(4-hydroxyphenyl)-3 4-(2- piperidine or 3-methylpyrollidine -benzo b thiophene compounds
IL65378A (en) * 1981-04-03 1986-02-28 Lilly Co Eli Process for preparing 3-(4-aminoethoxybenzoyl)benzo-(b)thiophenes
US4418068A (en) * 1981-04-03 1983-11-29 Eli Lilly And Company Antiestrogenic and antiandrugenic benzothiophenes
IL65379A0 (en) * 1981-04-03 1982-05-31 Lilly Co Eli Process for preparing acylated benzothiophenes
US4358593A (en) * 1981-04-03 1982-11-09 Eli Lilly And Company Process for preparing 3-(4-aminoethoxybenzoyl)benzo[b]thiophenes
US4380635A (en) * 1981-04-03 1983-04-19 Eli Lilly And Company Synthesis of acylated benzothiophenes
US4544746A (en) * 1982-05-17 1985-10-01 Ciba-Geigy Corporation Process for preparing 2-anilinoacridone
JPH02501301A (ja) * 1987-09-25 1990-05-10 チバ‐ガイギー　アクチェンゲゼルシャフト ４‐（トリアルキルベンジル）‐ピペラジニル化合物のジアシル誘導体
US5395842A (en) * 1988-10-31 1995-03-07 Endorecherche Inc. Anti-estrogenic compounds and compositions
DE4117512A1 (de) * 1991-05-25 1992-11-26 Schering Ag 2-phenylbenzo(b)furane und -thiophene, verfahren zu deren herstellung und diese enthaltende pharmazeutische praeparate
JP3157882B2 (ja) * 1991-11-15 2001-04-16 帝国臓器製薬株式会社 新規なベンゾチオフエン誘導体
DE4204969A1 (de) * 1992-02-19 1993-08-26 Basf Ag Verfahren zur herstellung von benzo(b)thiophenen
US6756388B1 (en) * 1993-10-12 2004-06-29 Pfizer Inc. Benzothiophenes and related compounds as estrogen agonists
US5523416A (en) * 1994-07-22 1996-06-04 Eli Lilly And Company Process for preparing 3-(4-aminoethoxy-benzoyl) benzo (B)-thiophenes
US5606076A (en) * 1995-06-07 1997-02-25 Eli Lilly And Company Process for the synthesis of benzo[b]thiophenes
US5606075A (en) * 1995-06-07 1997-02-25 Eli Lilly And Company Process for the synthesis of benzo[b]thiophenes

Also Published As

Publication number Publication date
HUP9904228A3 (en) 2001-06-28
EA001914B1 (ru) 2001-10-22
HUP9904228A2 (hu) 2001-05-28
EP0832889B1 (de) 2006-03-01
AR013321A1 (es) 2000-12-27
IL129001A (en) 2003-06-24
JP2001501208A (ja) 2001-01-30
EP0832889A1 (de) 1998-04-01
NO991193D0 (no) 1999-03-11
DE69735339T2 (de) 2006-10-12
IN183239B (de) 1999-10-09
WO1998013363A1 (en) 1998-04-02
PL332208A1 (en) 1999-08-30
US5977383A (en) 1999-11-02
DE69735339D1 (de) 2006-04-27
CN1230957A (zh) 1999-10-06
EA199900330A1 (ru) 2000-06-26
BR9712844A (pt) 1999-11-16
YU15399A (sh) 2001-07-10
CO4900043A1 (es) 2000-03-27
NZ334591A (en) 2000-07-28
UA62938C2 (en) 2004-01-15
CN1088704C (zh) 2002-08-07
PE2699A1 (es) 1999-02-04
IL129001A0 (en) 2000-02-17
AU4356197A (en) 1998-04-17
TR199900672T2 (xx) 1999-06-21
AU718919B2 (en) 2000-04-20
ID21349A (id) 1999-05-27
KR20000048539A (ko) 2000-07-25
NO991193L (no) 1999-03-25
TW472053B (en) 2002-01-11
MY118009A (en) 2004-08-30
CA2266617A1 (en) 1998-04-02
ATE318805T1 (de) 2006-03-15
ZA978372B (en) 1999-03-17
CZ92899A3 (cs) 1999-09-15
ES2257761T3 (es) 2006-08-01

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