EE200200529A - Tsüklilised ß-aminohappe derivaadid kui maatriksmetalloproteaaside ja TNF-a inhibiitorid - Google Patents

Tsüklilised ß-aminohappe derivaadid kui maatriksmetalloproteaaside ja TNF-a inhibiitorid

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Publication number
EE200200529A
EE200200529A EEP200200529A EEP200200529A EE200200529A EE 200200529 A EE200200529 A EE 200200529A EE P200200529 A EEP200200529 A EE P200200529A EE P200200529 A EEP200200529 A EE P200200529A EE 200200529 A EE200200529 A EE 200200529A
Authority
EE
Estonia
Prior art keywords
tnf
inhibitors
cyclic
amino acid
acid derivatives
Prior art date
Application number
EEP200200529A
Other languages
English (en)
Estonian (et)
Inventor
Duan Jingwu
Chen Linhua
R. Ott Gregory
Decicco Carl
Lu Zhonghui
P. Maduskuie Thomas Jr.
E. Voss Matthew
Xue Chu-Biao
Original Assignee
Bristol-Myers Squibb Pharma Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Pharma Company filed Critical Bristol-Myers Squibb Pharma Company
Publication of EE200200529A publication Critical patent/EE200200529A/xx

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    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • C07C259/08—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids having carbon atoms of hydroxamic groups bound to carbon atoms of rings other than six-membered aromatic rings
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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EEP200200529A 2000-03-17 2001-03-15 Tsüklilised ß-aminohappe derivaadid kui maatriksmetalloproteaaside ja TNF-a inhibiitorid EE200200529A (et)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US19018200P 2000-03-17 2000-03-17
US23337300P 2000-09-18 2000-09-18
US25553900P 2000-12-14 2000-12-14
PCT/US2001/008334 WO2001070673A2 (en) 2000-03-17 2001-03-15 CYCLIC β-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-$g(a)

Publications (1)

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EE200200529A true EE200200529A (et) 2004-02-16

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EEP200200529A EE200200529A (et) 2000-03-17 2001-03-15 Tsüklilised ß-aminohappe derivaadid kui maatriksmetalloproteaaside ja TNF-a inhibiitorid

Country Status (20)

Country Link
US (2) US6743807B2 (xx)
EP (1) EP1263755A2 (xx)
JP (1) JP2003528072A (xx)
KR (1) KR20030009391A (xx)
CN (1) CN1481377A (xx)
AR (1) AR035710A1 (xx)
AU (1) AU2001250849A1 (xx)
BR (1) BR0109467A (xx)
CA (1) CA2401870A1 (xx)
CZ (1) CZ20023033A3 (xx)
EE (1) EE200200529A (xx)
HK (1) HK1049165A1 (xx)
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WO2001070673A2 (en) 2001-09-27
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IL151552A0 (en) 2003-04-10
BR0109467A (pt) 2003-06-03
US20040162426A1 (en) 2004-08-19
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PL360678A1 (en) 2004-09-20
US6984648B2 (en) 2006-01-10
HK1049165A1 (zh) 2003-05-02
CA2401870A1 (en) 2001-09-27
CN1481377A (zh) 2004-03-10
NO20024402D0 (no) 2002-09-13
WO2001070673A3 (en) 2002-03-14
AR035710A1 (es) 2004-07-07
EP1263755A2 (en) 2002-12-11
HUP0300850A2 (hu) 2003-07-28
US20020016336A1 (en) 2002-02-07
MXPA02009020A (es) 2003-02-12
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US6743807B2 (en) 2004-06-01
CZ20023033A3 (cs) 2003-01-15
KR20030009391A (ko) 2003-01-29

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