ECSP088179A - Compuestos de carbamato para usarse en el tratamiento de desordenes neurodegenerativos - Google Patents
Compuestos de carbamato para usarse en el tratamiento de desordenes neurodegenerativosInfo
- Publication number
- ECSP088179A ECSP088179A EC2008008179A ECSP088179A ECSP088179A EC SP088179 A ECSP088179 A EC SP088179A EC 2008008179 A EC2008008179 A EC 2008008179A EC SP088179 A ECSP088179 A EC SP088179A EC SP088179 A ECSP088179 A EC SP088179A
- Authority
- EC
- Ecuador
- Prior art keywords
- formula
- group
- phenyl
- alkyl
- treatment
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/325—Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Diabetes (AREA)
- Psychology (AREA)
- Emergency Medicine (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Endocrinology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Esta invención se dirige a métodos para proveer neuroprotección que comprenden administrar a un sujeto que necesita de la misma una cantidad terapéuticamente efectiva de un compuesto seleccionado a partir del grupo que consiste de la fórmula (I) y de la fórmula (II), o una sal o éster farmacéuticamente aceptable del mismo,:Fórmula (I) Fórmula (II)en donde el fenilo está sustituido en X con uno a cinco átomos de halógeno seleccionados a partir del grupo que consiste de flúor, cloro, bromo y yodo; y, R1, R2, R3, R4, R5 y R6 son independientemente seleccionados a partir del grupo que consiste de hidrógeno y alquilo de C1-C4; en donde alquilo de C1-C4 está opcionalmente sustituido con fenilo (en donde fenilo está opcionalmente sustituido con sustituyentes independientemente seleccionados a partir del grupo que consiste de halógeno, alquilo de C1-C4, alcoxi de C1-C4, amino, nitro y ciano).
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US69840305P | 2005-07-12 | 2005-07-12 |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP088179A true ECSP088179A (es) | 2008-03-26 |
Family
ID=37637734
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EC2008008179A ECSP088179A (es) | 2005-07-12 | 2008-02-12 | Compuestos de carbamato para usarse en el tratamiento de desordenes neurodegenerativos |
Country Status (18)
Country | Link |
---|---|
US (2) | US20070021500A1 (es) |
EP (1) | EP1917009A2 (es) |
JP (1) | JP2009501224A (es) |
KR (1) | KR20080031951A (es) |
CN (1) | CN101287459A (es) |
AR (1) | AR054551A1 (es) |
AU (1) | AU2006269381A1 (es) |
BR (1) | BRPI0613006A2 (es) |
CA (1) | CA2615129A1 (es) |
CR (1) | CR9721A (es) |
EA (1) | EA200800294A1 (es) |
EC (1) | ECSP088179A (es) |
IL (1) | IL188729A0 (es) |
NI (1) | NI200800008A (es) |
NO (1) | NO20080738L (es) |
TW (1) | TW200800158A (es) |
WO (1) | WO2007008562A2 (es) |
ZA (1) | ZA200801401B (es) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7962215B2 (en) | 2004-07-23 | 2011-06-14 | Synapse Biomedical, Inc. | Ventilatory assist system and methods to improve respiratory function |
CN101272776B (zh) * | 2005-07-26 | 2012-10-03 | 詹森药业有限公司 | 氨基甲酸酯在制备治疗物质滥用相关疾病药物中的用途 |
US9050005B2 (en) | 2005-08-25 | 2015-06-09 | Synapse Biomedical, Inc. | Method and apparatus for transgastric neurostimulation |
US20080097153A1 (en) * | 2006-08-24 | 2008-04-24 | Ignagni Anthony R | Method and apparatus for grasping an abdominal wall |
KR20090076958A (ko) * | 2006-10-06 | 2009-07-13 | 얀센 파마슈티카 엔.브이. | 신규 (s)-(+)-2-(2-클로로페닐)-2-하이드록시-에틸 카바메이트 결정 |
US9079016B2 (en) * | 2007-02-05 | 2015-07-14 | Synapse Biomedical, Inc. | Removable intramuscular electrode |
WO2008144578A1 (en) * | 2007-05-17 | 2008-11-27 | Synapse Biomedical, Inc. | Devices and methods for assessing motor point electromyogram as a biomarker |
US8428726B2 (en) | 2007-10-30 | 2013-04-23 | Synapse Biomedical, Inc. | Device and method of neuromodulation to effect a functionally restorative adaption of the neuromuscular system |
US8478412B2 (en) * | 2007-10-30 | 2013-07-02 | Synapse Biomedical, Inc. | Method of improving sleep disordered breathing |
WO2011071995A2 (en) | 2009-12-08 | 2011-06-16 | Case Western Reserve University | Compounds and methods of treating ocular disorders |
US8609849B1 (en) | 2010-11-30 | 2013-12-17 | Fox Chase Chemical Diversity Center, Inc. | Hydroxylated sulfamides exhibiting neuroprotective action and their method of use |
KR101418061B1 (ko) * | 2012-09-28 | 2014-07-10 | 한국과학기술연구원 | 성상교세포의 글루타메이트 방출 기작 |
KR101758543B1 (ko) * | 2013-03-12 | 2017-07-14 | (주)바이오팜솔루션즈 | 페닐카바메이트 화합물 및 이를 포함하는 신경가스에 의한 질환의 예방 또는 치료용 조성물 |
US8652527B1 (en) | 2013-03-13 | 2014-02-18 | Upsher-Smith Laboratories, Inc | Extended-release topiramate capsules |
US9101545B2 (en) | 2013-03-15 | 2015-08-11 | Upsher-Smith Laboratories, Inc. | Extended-release topiramate capsules |
CA3016253C (en) * | 2016-02-29 | 2020-12-29 | Bio-Pharm Solutions Co., Ltd. | Sulfamate derivative compounds, processes for preparing them and their uses |
US11471683B2 (en) | 2019-01-29 | 2022-10-18 | Synapse Biomedical, Inc. | Systems and methods for treating sleep apnea using neuromodulation |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5698588A (en) * | 1996-01-16 | 1997-12-16 | Yukong Limited | Halogen substituted carbamate compounds from 2-phenyl-1,2-ethanediol |
US6306909B1 (en) * | 1997-03-12 | 2001-10-23 | Queen's University At Kingston | Anti-epileptogenic agents |
SK286621B6 (sk) * | 1999-08-20 | 2009-02-05 | Ortho-Mcneil Pharmaceutical, Inc. | Farmaceutický prostriedok obsahujúci kombináciu tramadolového materiálu a antikonvulzívneho činidla, táto kombinácia a jej použitie na výrobu liečiva |
CN1235579C (zh) * | 2001-02-27 | 2006-01-11 | 奥索-麦克尼尔药品公司 | 用于预防或治疗神经变性疾病的氨基甲酸酯化合物 |
US20060194873A1 (en) * | 2004-09-16 | 2006-08-31 | Choi Yong M | Methods of treating epileptogenesis and epilepsy |
PE20070325A1 (es) * | 2005-06-29 | 2007-05-12 | Alza Corp | Formas de dosificacion oral que comprenden compuestos derivados de carbamato |
-
2006
- 2006-07-06 US US11/481,601 patent/US20070021500A1/en not_active Abandoned
- 2006-07-07 CN CNA2006800331046A patent/CN101287459A/zh active Pending
- 2006-07-07 EP EP06786448A patent/EP1917009A2/en not_active Withdrawn
- 2006-07-07 WO PCT/US2006/026291 patent/WO2007008562A2/en active Application Filing
- 2006-07-07 EA EA200800294A patent/EA200800294A1/ru unknown
- 2006-07-07 JP JP2008521436A patent/JP2009501224A/ja not_active Withdrawn
- 2006-07-07 KR KR1020087003268A patent/KR20080031951A/ko not_active Application Discontinuation
- 2006-07-07 BR BRPI0613006-2A patent/BRPI0613006A2/pt not_active IP Right Cessation
- 2006-07-07 AU AU2006269381A patent/AU2006269381A1/en not_active Abandoned
- 2006-07-07 CA CA002615129A patent/CA2615129A1/en not_active Abandoned
- 2006-07-11 AR ARP060102977A patent/AR054551A1/es not_active Application Discontinuation
- 2006-07-11 TW TW095125161A patent/TW200800158A/zh unknown
-
2008
- 2008-01-10 IL IL188729A patent/IL188729A0/en unknown
- 2008-01-11 NI NI200800008A patent/NI200800008A/es unknown
- 2008-02-11 CR CR9721A patent/CR9721A/es unknown
- 2008-02-11 ZA ZA200801401A patent/ZA200801401B/xx unknown
- 2008-02-11 NO NO20080738A patent/NO20080738L/no not_active Application Discontinuation
- 2008-02-12 EC EC2008008179A patent/ECSP088179A/es unknown
-
2009
- 2009-01-30 US US12/362,970 patent/US20090137652A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
IL188729A0 (en) | 2008-11-03 |
TW200800158A (en) | 2008-01-01 |
CR9721A (es) | 2008-11-24 |
US20090137652A1 (en) | 2009-05-28 |
KR20080031951A (ko) | 2008-04-11 |
CA2615129A1 (en) | 2007-01-18 |
EP1917009A2 (en) | 2008-05-07 |
US20070021500A1 (en) | 2007-01-25 |
WO2007008562A2 (en) | 2007-01-18 |
CN101287459A (zh) | 2008-10-15 |
WO2007008562A3 (en) | 2007-08-16 |
JP2009501224A (ja) | 2009-01-15 |
NI200800008A (es) | 2010-11-25 |
AU2006269381A1 (en) | 2007-01-18 |
BRPI0613006A2 (pt) | 2010-12-14 |
AR054551A1 (es) | 2007-06-27 |
EA200800294A1 (ru) | 2008-06-30 |
NO20080738L (no) | 2008-04-10 |
ZA200801401B (en) | 2009-08-26 |
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