EA201791910A1 - Инъецируемые препараты длительного действия, содержащие изоксазолиновое действующее вещество, способы и применение - Google Patents
Инъецируемые препараты длительного действия, содержащие изоксазолиновое действующее вещество, способы и применениеInfo
- Publication number
- EA201791910A1 EA201791910A1 EA201791910A EA201791910A EA201791910A1 EA 201791910 A1 EA201791910 A1 EA 201791910A1 EA 201791910 A EA201791910 A EA 201791910A EA 201791910 A EA201791910 A EA 201791910A EA 201791910 A1 EA201791910 A1 EA 201791910A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- long
- isoxasoline
- applications
- methods
- injectable preparations
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
- A01P7/00—Arthropodicides
- A01P7/04—Insecticides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/69—Boron compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Настоящее изобретение касается инъецируемых препаратов длительного действия для борьбы с паразитами у животных, содержащих по меньшей мере одно изоксазолиновое действующее вещество, полоксамер и сорастворитель. В настоящем изобретении описаны также улучшенные способы удаления, борьбы или предотвращения появления паразитарных инфекций и заражений у животного, включающие введение инъецируемых препаратов длительного действия по настоящему изобретению животному, нуждающемуся в этом.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201562121350P | 2015-02-26 | 2015-02-26 | |
PCT/US2016/019688 WO2016138339A1 (en) | 2015-02-26 | 2016-02-26 | Long-acting injectable formulations comprising an isoxazoline active agent, methods and uses thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
EA201791910A1 true EA201791910A1 (ru) | 2017-12-29 |
EA035993B1 EA035993B1 (ru) | 2020-09-10 |
Family
ID=56015068
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201992772A EA201992772A1 (ru) | 2015-02-26 | 2016-02-26 | Инъецируемые препараты длительного действия, содержащие изоксазолиновое действующее вещество, способы и применение |
EA201791910A EA035993B1 (ru) | 2015-02-26 | 2016-02-26 | Инъецируемые препараты длительного действия, содержащие изоксазолиновое действующее вещество, способы и применение |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201992772A EA201992772A1 (ru) | 2015-02-26 | 2016-02-26 | Инъецируемые препараты длительного действия, содержащие изоксазолиновое действующее вещество, способы и применение |
Country Status (15)
Country | Link |
---|---|
US (2) | US10561641B2 (ru) |
EP (1) | EP3261617A1 (ru) |
JP (2) | JP6789232B2 (ru) |
KR (1) | KR102560198B1 (ru) |
CN (1) | CN107427496B (ru) |
AR (1) | AR103803A1 (ru) |
AU (3) | AU2016222532B2 (ru) |
CA (1) | CA2977376C (ru) |
CL (1) | CL2017002164A1 (ru) |
CO (1) | CO2017008584A2 (ru) |
EA (2) | EA201992772A1 (ru) |
MX (2) | MX2017010740A (ru) |
NZ (1) | NZ734948A (ru) |
UY (1) | UY36570A (ru) |
WO (1) | WO2016138339A1 (ru) |
Families Citing this family (12)
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UY36570A (es) * | 2015-02-26 | 2016-10-31 | Merial Inc | Formulaciones inyectables de acción prolongada que comprenden un agente activo isoxazolina, métodos y usos de las mismas |
UY37137A (es) * | 2016-02-24 | 2017-09-29 | Merial Inc | Compuestos antiparasitarios de isoxazolina, formulaciones inyectables de acción prolongada que los comprenden, métodos y usos de los mismos |
WO2018039508A1 (en) | 2016-08-25 | 2018-03-01 | Merial, Inc. | Method for reducing unwanted effects in parasiticidal treatments |
WO2018187623A1 (en) | 2017-04-05 | 2018-10-11 | Merial, Inc. | Crystalline forms of (s)-afoxolaner |
BR112020008848A2 (pt) | 2017-11-07 | 2020-10-20 | Intervet International B.V. | processo de preparação de partículas de isoxazolina de tamanho grande |
CA3081646C (en) * | 2017-11-07 | 2024-03-19 | Intervet International B.V. | Injectable isoxazoline pharmaceutical compositions and uses thereof |
NZ766141A (en) | 2017-12-15 | 2024-01-26 | Tarsus Pharmaceuticals Inc | Isoxazoline parasiticide formulations and methods for treating blepharitis |
TWI812673B (zh) * | 2018-02-12 | 2023-08-21 | 美商富曼西公司 | 用於防治無脊椎害蟲之萘異噁唑啉化合物 |
WO2020225143A1 (en) | 2019-05-03 | 2020-11-12 | Intervet International B.V. | Injectable pharmaceutical compositions and uses thereof |
EP4075981A1 (en) * | 2019-12-16 | 2022-10-26 | Intervet International B.V. | Composition for lice control |
DK4153133T3 (da) | 2020-05-20 | 2024-02-05 | Intervet Int Bv | Injicerbare farmaceutiske sammensætninger og anvendelser deraf |
CN116570556B (zh) * | 2023-05-17 | 2023-11-07 | 郑州福源动物药业有限公司 | 一种用于治疗畜禽大肠埃希菌和巴氏杆菌感染的复方磺胺氯达嗪钠溶液及其制备方法 |
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AR103803A1 (es) | 2017-06-07 |
AU2016222532B2 (en) | 2018-07-12 |
MX2017010740A (es) | 2017-12-04 |
CL2017002164A1 (es) | 2018-04-27 |
US10561641B2 (en) | 2020-02-18 |
NZ734948A (en) | 2018-07-27 |
US20160256442A1 (en) | 2016-09-08 |
EA035993B1 (ru) | 2020-09-10 |
JP2018509405A (ja) | 2018-04-05 |
KR20170131464A (ko) | 2017-11-29 |
BR112017018442A2 (pt) | 2018-04-17 |
JP6789232B2 (ja) | 2020-11-25 |
CN107427496B (zh) | 2021-05-14 |
CA2977376A1 (en) | 2016-09-01 |
KR102560198B1 (ko) | 2023-07-26 |
AU2016222532A1 (en) | 2017-09-21 |
EP3261617A1 (en) | 2018-01-03 |
US20200022959A1 (en) | 2020-01-23 |
AU2018205137B2 (en) | 2019-08-08 |
CN107427496A (zh) | 2017-12-01 |
JP7089564B2 (ja) | 2022-06-22 |
AU2018205137A1 (en) | 2018-08-02 |
EA201992772A1 (ru) | 2020-06-26 |
MX2020009010A (es) | 2020-10-12 |
UY36570A (es) | 2016-10-31 |
JP2021008485A (ja) | 2021-01-28 |
CO2017008584A2 (es) | 2017-11-10 |
US11484528B2 (en) | 2022-11-01 |
WO2016138339A1 (en) | 2016-09-01 |
AU2019261769A1 (en) | 2019-12-05 |
CA2977376C (en) | 2024-03-05 |
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