EA201200918A1 - Производные пирролидин карбоновой кислоты как агонисты сопряженного с g-белком рецептора 43 (gpr43), фармацевтическая композиция и методы их использования при лечении метаболических нарушений - Google Patents

Производные пирролидин карбоновой кислоты как агонисты сопряженного с g-белком рецептора 43 (gpr43), фармацевтическая композиция и методы их использования при лечении метаболических нарушений

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EA201200918A1
EA201200918A1 EA201200918A EA201200918A EA201200918A1 EA 201200918 A1 EA201200918 A1 EA 201200918A1 EA 201200918 A EA201200918 A EA 201200918A EA 201200918 A EA201200918 A EA 201200918A EA 201200918 A1 EA201200918 A1 EA 201200918A1
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Eurasian Patent Office
Prior art keywords
treatment
metabolicche
gpr43
agonists
methods
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EA201200918A
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English (en)
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EA023861B3 (ru
EA023861B1 (ru
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Хамид Ховейда
Дидье Шилс
Людивин Зут
Жюльен Парк
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Эроскрин С.А.
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Publication of EA201200918A1 publication Critical patent/EA201200918A1/ru
Publication of EA023861B1 publication Critical patent/EA023861B1/ru
Publication of EA023861B3 publication Critical patent/EA023861B3/ru

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Abstract

Данное изобретение касается новых соединений формулы I, а также их использования в лечении и/или предотвращении метаболических заболеваний.
EA201200918A 2009-12-18 2010-12-17 Производные пирролидин карбоновой кислоты как агонисты сопряженного с g-белком рецептора 43 (gpr43), фармацевтическая композиция и методы их использования при лечении метаболических нарушений EA023861B3 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP09306270 2009-12-18
US37337010P 2010-08-13 2010-08-13
US37601310P 2010-08-23 2010-08-23
PCT/EP2010/070040 WO2011073376A1 (en) 2009-12-18 2010-12-17 Pyrrolidine or thiazolidine carboxylic acid derivatives, pharmaceutical composition and methods for use in treating metabolic disordersas as agonists of g- protein coupled receptor 43 (gpr43)

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EA201200918A1 true EA201200918A1 (ru) 2012-12-28
EA023861B1 EA023861B1 (ru) 2016-07-29
EA023861B3 EA023861B3 (ru) 2016-09-30

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KR (1) KR101827529B1 (ru)
CN (1) CN102812003B (ru)
AU (1) AU2010332765C1 (ru)
BR (1) BR112012018374B1 (ru)
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