EA201171371A1 - Полиненасыщенные жирные кислоты для лечения заболеваний, связанных с сердечно-сосудистыми, метаболическими и воспалительными заболеваниями - Google Patents

Полиненасыщенные жирные кислоты для лечения заболеваний, связанных с сердечно-сосудистыми, метаболическими и воспалительными заболеваниями

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EA201171371A1
EA201171371A1 EA201171371A EA201171371A EA201171371A1 EA 201171371 A1 EA201171371 A1 EA 201171371A1 EA 201171371 A EA201171371 A EA 201171371A EA 201171371 A EA201171371 A EA 201171371A EA 201171371 A1 EA201171371 A1 EA 201171371A1
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treatment
cardiovascular
metabolic
diseases
polynesative
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EA201171371A
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EA021177B1 (ru
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Рагнар Ховланд
Анне Кристин Хольмеиде
Торе Скъерет
Мортен Брендванг
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Пронова Биофарма Норге Ас
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Application filed by Пронова Биофарма Норге Ас filed Critical Пронова Биофарма Норге Ас
Publication of EA201171371A1 publication Critical patent/EA201171371A1/ru
Publication of EA021177B1 publication Critical patent/EA021177B1/ru

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Abstract

Настоящее изобретение относится к липидным соединениям общей формулы (I) R-O-C(R)(R)-X (I), где Rпредставляет собой С-Салкильную группу, С-Салкенильную группу, содержащую 1-6 двойных связей или С-Салкинильную группу, содержащую 1-6 тройных связей; Rи Rодинаковы или отличаются друг от друга и их можно выбрать из различных заместителей; и Х представляет собой карбоновую кислоту или ее производные, такие как эфир карбоновой кислоты, ангидрид карбоновой кислоты, фосфолипид, или триглицерид, или карбоксамид; или к их фармацевтически приемлемым солям, сольватам, сольватам таких солей или к их пролекарствам. Настоящее изобретение относится также к фармацевтическим композициям и липидным композициям, включающим по меньшей мере одно соединение настоящего изобретения, и к таким соединениям для использования в качестве лекарственных препаратов или для использования при лечении, в частности при лечении заболеваний, связанных с сердечно-сосудистыми, метаболическими и воспалительными заболеваниями.
EA201171371A 2009-05-08 2010-05-07 Полиненасыщенные жирные кислоты для лечения заболеваний, связанных с сердечно-сосудистыми, метаболическими и воспалительными заболеваниями EA021177B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17650309P 2009-05-08 2009-05-08
PCT/IB2010/001251 WO2010128401A1 (en) 2009-05-08 2010-05-07 Polyunsaturated fatty acids for the treatment of diseases related to cardiovascular, metabolic and inflammatory disease areas

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EA201171371A1 true EA201171371A1 (ru) 2012-05-30
EA021177B1 EA021177B1 (ru) 2015-04-30

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US (2) US8735436B2 (ru)
EP (1) EP2427415B1 (ru)
JP (2) JP5843755B2 (ru)
KR (1) KR101783817B1 (ru)
CN (1) CN102459142B (ru)
AR (2) AR078507A1 (ru)
AU (1) AU2010244136B2 (ru)
BR (1) BRPI1015120B8 (ru)
CA (1) CA2760877C (ru)
CL (1) CL2011002745A1 (ru)
CO (1) CO6430454A2 (ru)
DK (1) DK2427415T3 (ru)
EA (1) EA021177B1 (ru)
ES (1) ES2726765T3 (ru)
HR (1) HRP20190732T1 (ru)
IL (1) IL216171A (ru)
MA (1) MA33341B1 (ru)
MX (2) MX2011011614A (ru)
MY (1) MY165292A (ru)
NZ (2) NZ596386A (ru)
PH (1) PH12015500930A1 (ru)
PL (1) PL2427415T3 (ru)
PT (1) PT2427415T (ru)
SG (1) SG175401A1 (ru)
TR (1) TR201905768T4 (ru)
TW (1) TWI558395B (ru)
UA (1) UA109528C2 (ru)
WO (1) WO2010128401A1 (ru)
ZA (2) ZA201108163B (ru)

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UA109528C2 (uk) 2015-09-10
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WO2010128401A9 (en) 2011-12-08
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TWI558395B (zh) 2016-11-21
ZA201108163B (en) 2018-11-28
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US20140221439A1 (en) 2014-08-07
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CA2760877A1 (en) 2010-11-11
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