EA201171195A1 - Конъюгаты, частицы, композиции "полимер-агент" и способы их применения - Google Patents

Конъюгаты, частицы, композиции "полимер-агент" и способы их применения

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Publication number
EA201171195A1
EA201171195A1 EA201171195A EA201171195A EA201171195A1 EA 201171195 A1 EA201171195 A1 EA 201171195A1 EA 201171195 A EA201171195 A EA 201171195A EA 201171195 A EA201171195 A EA 201171195A EA 201171195 A1 EA201171195 A1 EA 201171195A1
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EA
Eurasian Patent Office
Prior art keywords
particles
polymer
conjugates
methods
application
Prior art date
Application number
EA201171195A
Other languages
English (en)
Other versions
EA201171195A8 (ru
Inventor
Скотт Элиасоф
Томас С. Кроуфорд
Геети Гангел
Лоренс Алан Райтер
Пей-Сзе Нг
Original Assignee
Серулин Фарма Инк.
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Publication date
Application filed by Серулин Фарма Инк. filed Critical Серулин Фарма Инк.
Publication of EA201171195A1 publication Critical patent/EA201171195A1/ru
Publication of EA201171195A8 publication Critical patent/EA201171195A8/ru

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    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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    • A61K47/56Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
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  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

В данном изобретении описаны конъюгаты и частицы "полимер-агент", которые могут применяться, например, в лечении рака. Также в данном описании описаны смеси, композиции и лекарственные формы, содержащие частицы, способы применения частиц (например, для лечения расстройства), наборы, включающие конъюгаты и частицы "полимер-агент", способы получения конъюгатов и частиц "полимер-агент", способы хранения частиц и способы анализа частиц.
EA201171195A 2009-03-30 2010-03-26 Конъюгаты, частицы, композиции "полимер-агент" и способы их применения EA201171195A8 (ru)

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US20120282306A1 (en) 2012-11-08
EP2413901A4 (en) 2015-05-06
JP2012522055A (ja) 2012-09-20
US20130011445A1 (en) 2013-01-10
US20110268658A1 (en) 2011-11-03
CN102378626A (zh) 2012-03-14
US20110189092A1 (en) 2011-08-04
CN102378626B (zh) 2014-05-14
WO2010117668A1 (en) 2010-10-14
CA2756072A1 (en) 2010-10-14
IL215123A0 (en) 2011-12-29
EP2413901A1 (en) 2012-02-08
EA201171195A8 (ru) 2014-08-29
US20100247668A1 (en) 2010-09-30
US20140099263A1 (en) 2014-04-10
MX2011010390A (es) 2011-12-14
JP2015117250A (ja) 2015-06-25
AU2010234916A1 (en) 2011-10-13
US20140286873A1 (en) 2014-09-25
BRPI1014854A2 (pt) 2016-05-03

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