EA201100377A1 - Способ получения сульфонамидов - Google Patents

Способ получения сульфонамидов

Info

Publication number
EA201100377A1
EA201100377A1 EA201100377A EA201100377A EA201100377A1 EA 201100377 A1 EA201100377 A1 EA 201100377A1 EA 201100377 A EA201100377 A EA 201100377A EA 201100377 A EA201100377 A EA 201100377A EA 201100377 A1 EA201100377 A1 EA 201100377A1
Authority
EA
Eurasian Patent Office
Prior art keywords
formula
equivalents
base
sulphonamides
obtaining
Prior art date
Application number
EA201100377A
Other languages
English (en)
Inventor
Томас Шмидт
Йоахим Гебхардт
Зандра Лёр
Михаэль Кайль
Ян-Хендрик Веверс
Михаэль Ракк
Гуидо Майер
Аксель Плешке
Original Assignee
Басф Се
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE200510057681 external-priority patent/DE102005057681A1/de
Application filed by Басф Се filed Critical Басф Се
Publication of EA201100377A1 publication Critical patent/EA201100377A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C07C303/38—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reaction of ammonia or amines with sulfonic acids, or with esters, anhydrides, or halides thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C201/00—Preparation of esters of nitric or nitrous acid or of compounds containing nitro or nitroso groups bound to a carbon skeleton
    • C07C201/06—Preparation of nitro compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C201/00—Preparation of esters of nitric or nitrous acid or of compounds containing nitro or nitroso groups bound to a carbon skeleton
    • C07C201/06—Preparation of nitro compounds
    • C07C201/12—Preparation of nitro compounds by reactions not involving the formation of nitro groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C201/00—Preparation of esters of nitric or nitrous acid or of compounds containing nitro or nitroso groups bound to a carbon skeleton
    • C07C201/06—Preparation of nitro compounds
    • C07C201/16—Separation; Purification; Stabilisation; Use of additives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/13—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups
    • C07C205/20—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups having nitro groups and hydroxy groups bound to carbon atoms of six-membered aromatic rings
    • C07C205/21—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups having nitro groups and hydroxy groups bound to carbon atoms of six-membered aromatic rings having nitro groups and hydroxy groups bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C205/22—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups having nitro groups and hydroxy groups bound to carbon atoms of six-membered aromatic rings having nitro groups and hydroxy groups bound to carbon atoms of the same non-condensed six-membered aromatic ring having one nitro groups bound to the ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C07C303/40—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reactions not involving the formation of sulfonamide groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Способ получения сульфонамидов формулы Iгде заместители имеют значения, указанные в описании, реакцией хлоридов м-нитробензойной кислоты формулы II с аминосульфонами формулы III в присутствии В эквивалентов основания формулы IV, который отличается тем, что на стадии а) аминосульфоны формулы III реагируют с В1 эквивалентами основания формулы IV, а на стадии b) реакционную смесь, полученную на стадии а), подвергают взаимодействию с хлоридами м-нитробензойной кислоты формулы II и В2 эквивалентами основания формулы IV, где В, В1 и В2 имеют значения, указанные в описании.
EA201100377A 2005-12-01 2006-11-23 Способ получения сульфонамидов EA201100377A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE200510057681 DE102005057681A1 (de) 2005-12-01 2005-12-01 Verfahren zur Herstellung fluorierter m-Nitro-Benzoesäurechloride
EP06123569 2006-11-07

Publications (1)

Publication Number Publication Date
EA201100377A1 true EA201100377A1 (ru) 2011-08-30

Family

ID=37697933

Family Applications (2)

Application Number Title Priority Date Filing Date
EA200801432A EA200801432A1 (ru) 2005-12-01 2006-11-23 Способ получения сульфонамидов
EA201100377A EA201100377A1 (ru) 2005-12-01 2006-11-23 Способ получения сульфонамидов

Family Applications Before (1)

Application Number Title Priority Date Filing Date
EA200801432A EA200801432A1 (ru) 2005-12-01 2006-11-23 Способ получения сульфонамидов

Country Status (11)

Country Link
US (2) US8263806B2 (ru)
EP (1) EP1957443A2 (ru)
JP (1) JP5555426B2 (ru)
KR (3) KR101422433B1 (ru)
AR (1) AR057211A1 (ru)
AU (1) AU2006319263B2 (ru)
BR (1) BRPI0619760A2 (ru)
CA (3) CA2631113A1 (ru)
EA (2) EA200801432A1 (ru)
IL (3) IL191503A (ru)
WO (1) WO2007063028A2 (ru)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101422433B1 (ko) * 2005-12-01 2014-07-22 바스프 에스이 불소화 ｍ-니트로벤조일 클로라이드의 제조 방법
JP5465672B2 (ja) * 2007-10-12 2014-04-09 ビーエーエスエフ ソシエタス・ヨーロピア スルホン酸ジアミドの製法
IL271962B (en) 2017-07-28 2022-08-01 Basf Se Preparation of 3-aryl-5-trifluoromethyl-4,2,1-converted oxadiazoles
EP3587396A1 (en) * 2018-06-27 2020-01-01 Basf Se A method of isolating a n-(3-nitrobenzoyl)sulfamide
CN111499506B (zh) * 2020-03-23 2021-03-30 浙江本立科技股份有限公司 一种2,4-二氯-5-氟苯甲酰氯绿色生产工艺

Family Cites Families (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1240853B (de) 1962-12-06 1967-05-24 Smith Kline French Lab Verfahren zur Herstellung von Sulfurylamiden
US3198785A (en) * 1964-04-17 1965-08-03 Sandoz Ag Sulfamoyl azabicyclononanes and derivatives thereof
NL175521C (nl) * 1973-04-26 1984-11-16 Hoechst Ag Werkwijze voor het bereiden van carbonzuurchloriden.
DE2933148A1 (de) * 1979-08-16 1981-02-26 Bayer Ag Verfahren zur herstellung von aromatischen dicarbonsaeuredichloriden iv
DE3040295A1 (de) * 1980-10-25 1982-06-03 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von aromatischen carbonsaeurechloriden
JPS61155350A (ja) * 1984-12-28 1986-07-15 Ihara Nikkei Kagaku Kogyo Kk 脂肪酸クロライド及び芳香族酸クロライドの製造方法
EP0323487B1 (de) * 1987-06-19 1993-03-31 Ciba-Geigy Ag Heterocyclische verbindungen
EP0333791A1 (de) 1987-09-23 1989-09-27 Ciba-Geigy Ag Heterocyclische verbindungen
DE3812175A1 (de) * 1988-04-13 1989-10-26 Bayer Ag Verfahren zur herstellung von carbonsaeurehalogeniden
US5238908A (en) * 1989-08-31 1993-08-24 Rohm And Haas Company Herbicidal glutaramic acids and derivatives
JPH04117344A (ja) * 1990-09-05 1992-04-17 Res Assoc Util Of Light Oil 芳香族カルボン酸塩化物の製造方法
JPH09504508A (ja) * 1993-09-28 1997-05-06 チバ−ガイギー アクチエンゲゼルシャフト 殺虫剤及び殺ダニ剤としてのアクリル化スルホンアミド
CA2393515A1 (en) * 1999-12-07 2001-06-14 Basf Aktiengesellschaft Method for producing o-chloromethyl benzoic acid chlorides
DE19958758A1 (de) * 1999-12-07 2001-07-05 Basf Ag Verfahren zur Herstellung von o-Chlormethylbenzoesäurechloriden
JP2001187762A (ja) * 1999-12-28 2001-07-10 Nippon Light Metal Co Ltd 高純度芳香族酸クロライドの製造方法
JP2003519143A (ja) * 1999-12-28 2003-06-17 ファーマコピーア，インコーポレーティッド ピリミジン及びトリアジン系キナーゼ阻害剤
JP2004501084A (ja) * 2000-04-17 2004-01-15 ビーエーエスエフ　アクチェンゲゼルシャフト 除草活性を有する３−ヘテロ環置換ベンゾイソチアゾール及びベンゾイソオキサゾール化合物
US6251829B1 (en) * 2000-04-18 2001-06-26 Rohm And Haas Company Herbicidal benzoyloxy carboxylates and carboxamides
SI1226127T1 (sl) 2000-05-04 2009-10-31 Basf Se Substituirani fenilsulfamoil karboksamidi
ATE458724T1 (de) * 2001-06-26 2010-03-15 Bristol Myers Squibb Co N-heterocyclische inhibitoren der expression von tnf-alpha
WO2003007945A1 (en) * 2001-07-20 2003-01-30 Boehringer Ingelheim (Canada) Ltd. Viral polymerase inhibitors
DK1506169T3 (da) * 2002-05-16 2010-04-19 Basf Se Fremgangsmåde til fremstilling af sulfonsyrediamider
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BRPI0315932B1 (pt) * 2002-10-30 2019-08-13 Basf Ag processo para a preparação de iso(tio)cianatos de fenila, compostos, e, processo para a preparação do composto sendo amida do ácido aminobenzoilsulfâmico
WO2004106324A1 (en) 2003-05-27 2004-12-09 E.I. Dupont De Nemours And Company Azolecarboxamide herbicides
CA2574406C (en) 2004-07-22 2013-02-19 Basf Aktiengesellschaft Method for the production of 3-phenyl(thio)uracils and dithiouracils
ITMI20050275A1 (it) * 2005-02-22 2006-08-23 Miteni Spa Procedimento per la preparazione di derivati dell'acido benzoico attraverso un nuovo intermedio di sintesi
KR101422433B1 (ko) 2005-12-01 2014-07-22 바스프 에스이 불소화 ｍ-니트로벤조일 클로라이드의 제조 방법
JP5465672B2 (ja) 2007-10-12 2014-04-09 ビーエーエスエフ ソシエタス・ヨーロピア スルホン酸ジアミドの製法

Also Published As

Publication number Publication date
IL191503A (en) 2014-09-30
KR101422433B1 (ko) 2014-07-22
KR20130093695A (ko) 2013-08-22
KR20130093696A (ko) 2013-08-22
JP2009517440A (ja) 2009-04-30
WO2007063028A3 (de) 2007-08-23
US20120310010A1 (en) 2012-12-06
CA2821516A1 (en) 2007-06-07
AU2006319263B2 (en) 2012-06-28
US8263806B2 (en) 2012-09-11
AU2006319263A1 (en) 2007-06-07
KR101422434B1 (ko) 2014-07-22
EA200801432A1 (ru) 2008-12-30
EP1957443A2 (de) 2008-08-20
BRPI0619760A2 (pt) 2012-02-22
CA2821517A1 (en) 2007-06-07
IL215280A0 (en) 2011-10-31
AR057211A1 (es) 2007-11-21
WO2007063028A2 (de) 2007-06-07
IL215279A0 (en) 2011-10-31
JP5555426B2 (ja) 2014-07-23
CA2631113A1 (en) 2007-06-07
KR20080072093A (ko) 2008-08-05
US20100228054A1 (en) 2010-09-09
KR101430949B1 (ko) 2014-08-18

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