ATE458724T1 - N-heterocyclische inhibitoren der expression von tnf-alpha - Google Patents
N-heterocyclische inhibitoren der expression von tnf-alphaInfo
- Publication number
- ATE458724T1 ATE458724T1 AT02739978T AT02739978T ATE458724T1 AT E458724 T1 ATE458724 T1 AT E458724T1 AT 02739978 T AT02739978 T AT 02739978T AT 02739978 T AT02739978 T AT 02739978T AT E458724 T1 ATE458724 T1 AT E458724T1
- Authority
- AT
- Austria
- Prior art keywords
- tnf
- alpha expression
- compounds
- heterocyclic inhibitors
- disclosed
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 108091000080 Phosphotransferase Proteins 0.000 abstract 1
- 108060008682 Tumor Necrosis Factor Proteins 0.000 abstract 1
- 102100040247 Tumor necrosis factor Human genes 0.000 abstract 1
- 230000016396 cytokine production Effects 0.000 abstract 1
- 230000005764 inhibitory process Effects 0.000 abstract 1
- 102000002574 p38 Mitogen-Activated Protein Kinases Human genes 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 102000020233 phosphotransferase Human genes 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/891,750 US6906067B2 (en) | 1999-12-28 | 2001-06-26 | N-heterocyclic inhibitors of TNF-α expression |
| PCT/US2002/020212 WO2003002542A1 (en) | 2000-12-22 | 2002-06-25 | N-heterocyclic inhibitors of tnf-alpha expression |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE458724T1 true ATE458724T1 (de) | 2010-03-15 |
Family
ID=31947149
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT02739978T ATE458724T1 (de) | 2001-06-26 | 2002-06-25 | N-heterocyclische inhibitoren der expression von tnf-alpha |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP1409463B1 (de) |
| JP (1) | JP2004535446A (de) |
| AT (1) | ATE458724T1 (de) |
| CA (1) | CA2451125A1 (de) |
| DE (1) | DE60235470D1 (de) |
| ES (1) | ES2339226T3 (de) |
| HU (1) | HUP0401712A3 (de) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1910385B1 (de) * | 2005-08-04 | 2013-07-24 | Sirtris Pharmaceuticals, Inc. | Benzothiazole und thiazolopyridine als sirtuinmodulatoren |
| EA200801432A1 (ru) * | 2005-12-01 | 2008-12-30 | Басф Се | Способ получения сульфонамидов |
| JP2009545598A (ja) * | 2006-08-01 | 2009-12-24 | プリーシス・ファーマシューティカルズ・インコーポレイテッド | Ｐ３８キナーゼ阻害剤 |
| CN101821233B (zh) | 2007-10-12 | 2016-06-29 | 巴斯夫欧洲公司 | 生产磺酸二酰胺的方法 |
| AU2009289378A1 (en) * | 2008-09-02 | 2010-03-11 | Boehringer Ingelheim International Gmbh | Novel benzamides, production thereof, and use thereof as medicaments |
| AU2011336764B2 (en) * | 2010-11-29 | 2017-02-23 | Galleon Pharmaceuticals, Inc. | Novel compounds as respiratory stimulants for treatment of breathing control disorders or diseases |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO311614B1 (no) * | 1996-10-01 | 2001-12-17 | Janssen Pharmaceutica Nv | Substituerte diamino-1,3,5-triazinderivater |
| WO1999001442A1 (en) * | 1997-07-02 | 1999-01-14 | Zeneca Limited | Triazine derivatives and their use as antibacterial agents |
| CA2394727A1 (en) * | 1999-12-28 | 2001-07-05 | Pharmacopeia, Inc. | Pyrimidine and triazine kinase inhibitors |
-
2002
- 2002-06-25 CA CA002451125A patent/CA2451125A1/en not_active Abandoned
- 2002-06-25 JP JP2003508923A patent/JP2004535446A/ja active Pending
- 2002-06-25 EP EP02739978A patent/EP1409463B1/de not_active Expired - Lifetime
- 2002-06-25 HU HU0401712A patent/HUP0401712A3/hu unknown
- 2002-06-25 AT AT02739978T patent/ATE458724T1/de not_active IP Right Cessation
- 2002-06-25 ES ES02739978T patent/ES2339226T3/es not_active Expired - Lifetime
- 2002-06-25 DE DE60235470T patent/DE60235470D1/de not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| EP1409463B1 (de) | 2010-02-24 |
| EP1409463A1 (de) | 2004-04-21 |
| DE60235470D1 (de) | 2010-04-08 |
| ES2339226T3 (es) | 2010-05-18 |
| HUP0401712A2 (hu) | 2004-12-28 |
| EP1409463A4 (de) | 2004-11-17 |
| JP2004535446A (ja) | 2004-11-25 |
| HUP0401712A3 (en) | 2009-06-29 |
| CA2451125A1 (en) | 2003-01-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |