IL178032A0 - An improved process for the preparation of n-([1,2,4-]triazolopyrimidin-2-yl)aryl sulfonamides - Google Patents

An improved process for the preparation of n-([1,2,4-]triazolopyrimidin-2-yl)aryl sulfonamides

Info

Publication number
IL178032A0
IL178032A0 IL178032A IL17803206A IL178032A0 IL 178032 A0 IL178032 A0 IL 178032A0 IL 178032 A IL178032 A IL 178032A IL 17803206 A IL17803206 A IL 17803206A IL 178032 A0 IL178032 A0 IL 178032A0
Authority
IL
Israel
Prior art keywords
triazolopyrimidin
preparation
improved process
aryl sulfonamides
sulfonamides
Prior art date
Application number
IL178032A
Other versions
IL178032A (en
Original Assignee
Dow Agrosciences Llc
Hamilton Christopher Thomas
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc, Hamilton Christopher Thomas filed Critical Dow Agrosciences Llc
Publication of IL178032A0 publication Critical patent/IL178032A0/en
Publication of IL178032A publication Critical patent/IL178032A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

The N-arylsulfilimine-catalyzed coupling of aromatic sulfonyl chlorides with N-([1,2,4]triazolopyrimidin-2-yl)amines to form N-([1,2,4]triazolo-pyrimidin-2-yl)aryl sulfonamides is improved by the selection of 3-picoline or 3,5-lutidine as the base.
IL178032A 2004-03-26 2006-09-12 Process for the preparation of n-([1,2,4]triazolopyrimidin-2-yl)aryl sulfonamides IL178032A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US55702204P 2004-03-26 2004-03-26
PCT/US2005/009964 WO2005097793A1 (en) 2004-03-26 2005-03-24 An improved process for the preparation of n-([1,2,4]triazolopyrimidin-2-yl)aryl sulfonamides

Publications (2)

Publication Number Publication Date
IL178032A0 true IL178032A0 (en) 2006-12-31
IL178032A IL178032A (en) 2013-11-28

Family

ID=34963841

Family Applications (1)

Application Number Title Priority Date Filing Date
IL178032A IL178032A (en) 2004-03-26 2006-09-12 Process for the preparation of n-([1,2,4]triazolopyrimidin-2-yl)aryl sulfonamides

Country Status (16)

Country Link
US (1) US7339058B2 (en)
EP (1) EP1735309B1 (en)
JP (1) JP4929155B2 (en)
KR (1) KR101111014B1 (en)
CN (1) CN100509812C (en)
AT (1) ATE451370T1 (en)
AU (1) AU2005230862B2 (en)
BR (1) BRPI0509273B8 (en)
CA (1) CA2558245C (en)
DE (1) DE602005018182D1 (en)
DK (1) DK1735309T3 (en)
IL (1) IL178032A (en)
MX (1) MXPA06010913A (en)
TW (1) TWI337183B (en)
WO (1) WO2005097793A1 (en)
ZA (1) ZA200606604B (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103044431A (en) * 2012-10-22 2013-04-17 中国药科大学 Novel preparation method of penoxsulam
CN103319489B (en) * 2013-07-12 2015-04-08 黑龙江大学 Triazolopyrimidine sulfonamide compound, and synthetic method and application thereof
CN104341326A (en) * 2013-08-08 2015-02-11 天津诺维康生物技术有限公司 Preparation method for 2-substituted 6-(trifluoromethyl)benzenesulphonyl chloride
BR112017019116B1 (en) * 2015-03-10 2022-02-01 Oriental (Luzhou) Agrochemicals. Co., Ltd Method for preparing high purity sulfonamide compound and sulfonamide compound intermediate
CN105294515B (en) * 2015-11-13 2017-10-10 天津现代职业技术学院 The preparation method of 2 (2 ', 2 ' difluoroethoxy) 6 trifluoromethyl benzene sulfonyl chloride
CN105399746B (en) * 2015-12-28 2017-11-07 黑龙江凯奥科技开发有限公司 Triazolopyrimidine sulfonamide compound, the composition containing the compound and its application
GB2555635B (en) * 2016-11-07 2022-04-13 Rotam Agrochem Int Co Ltd A novel form of penoxsulam, a process for its preparation and use of the same
CN108892671B (en) * 2018-08-20 2021-04-20 常州沃腾化工科技有限公司 Preparation method of pyroxsulam
CN108707109A (en) * 2018-08-29 2018-10-26 常州沃腾化工科技有限公司 A kind of preparation method of 2- methoxyl groups -4- trifluoromethyl pyridine -3- sulfonic acid chlorides
ES2939695T3 (en) 2018-12-27 2023-04-26 Corteva Agriscience Llc Preparation of intermediates of a sulfonamide herbicide process
WO2020139734A1 (en) 2018-12-27 2020-07-02 Dow Agrosciences Llc Preparation of sulfonamide herbicide process intermediates
CN110698363B (en) * 2019-01-28 2022-02-01 杭州师范大学 Synthetic method of 2- (2, 2-difluoroethoxy) -6- (trifluoromethyl) benzenesulfonyl chloride
CN110563735B (en) * 2019-09-27 2022-03-29 江苏好收成韦恩农化股份有限公司 Method for preparing florasulam

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5177206A (en) 1991-10-08 1993-01-05 Dowelanco Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides
HU229886B1 (en) * 1996-09-24 2014-11-28 Dow Agrosciences Llc Benzenesulfonyl cloride derivates suitable for the preparation of herbicidal n-(triazoloazinyl) benzenesulfonamid e compounds
AR015104A1 (en) * 1996-11-13 2001-04-18 Dowelanco SUBSTITUTED N-ARILSULFYLIMINE COMPOUNDS, USED AS CATALYSTS IN THE PREPARATION OF N-ARYLARILSULFONAMIDE COMPOUNDS; PROCESS TO PREPARE SUCH COMPOUNDS AND ITS USE TO CATALIZE SUCH PREPARATION.
HU227229B1 (en) 2000-11-03 2010-11-29 Dow Agrosciences Llc Herbicidal n-(5,7-dimethoxy[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)arylsulfonamide derivatives, their preparation and use as herbicides
CN1221552C (en) 2000-11-03 2005-10-05 美国陶氏益农公司 N-([1,2,4] triazoloazinyl) thiophene sulfonamide compounds as herbicides

Also Published As

Publication number Publication date
CN100509812C (en) 2009-07-08
JP2007530587A (en) 2007-11-01
EP1735309A1 (en) 2006-12-27
CN1930164A (en) 2007-03-14
CA2558245A1 (en) 2005-10-20
US7339058B2 (en) 2008-03-04
KR20070014135A (en) 2007-01-31
BRPI0509273A (en) 2007-09-04
ZA200606604B (en) 2008-01-30
AU2005230862B2 (en) 2010-12-23
TW200536842A (en) 2005-11-16
ATE451370T1 (en) 2009-12-15
MXPA06010913A (en) 2006-12-15
KR101111014B1 (en) 2012-02-13
IL178032A (en) 2013-11-28
WO2005097793A1 (en) 2005-10-20
DK1735309T3 (en) 2010-04-06
TWI337183B (en) 2011-02-11
US20050215570A1 (en) 2005-09-29
CA2558245C (en) 2012-01-03
EP1735309B1 (en) 2009-12-09
DE602005018182D1 (en) 2010-01-21
BRPI0509273B1 (en) 2015-12-22
JP4929155B2 (en) 2012-05-09
BRPI0509273B8 (en) 2022-06-28
AU2005230862A1 (en) 2005-10-20

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