EA200801209A1 - Гетероароматические сульфонамидные пролекарства - Google Patents
Гетероароматические сульфонамидные пролекарстваInfo
- Publication number
- EA200801209A1 EA200801209A1 EA200801209A EA200801209A EA200801209A1 EA 200801209 A1 EA200801209 A1 EA 200801209A1 EA 200801209 A EA200801209 A EA 200801209A EA 200801209 A EA200801209 A EA 200801209A EA 200801209 A1 EA200801209 A1 EA 200801209A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- heteroaromatic
- procaraments
- sulphonamide
- compounds
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/64—Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
- A61K31/5685—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone having an oxo group in position 17, e.g. androsterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/59—Compounds containing 9, 10- seco- cyclopenta[a]hydrophenanthrene ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/02—Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Epidemiology (AREA)
- Gynecology & Obstetrics (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Pregnancy & Childbirth (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102005057421A DE102005057421A1 (de) | 2005-11-30 | 2005-11-30 | Heteroaromatische Sulfonamid-Prodrugs |
PCT/EP2006/011727 WO2007062875A1 (de) | 2005-11-30 | 2006-11-27 | Heteroaromatische sulfonamid-prodrugs |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200801209A1 true EA200801209A1 (ru) | 2008-12-30 |
Family
ID=37875507
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200801209A EA200801209A1 (ru) | 2005-11-30 | 2006-11-27 | Гетероароматические сульфонамидные пролекарства |
Country Status (14)
Country | Link |
---|---|
EP (1) | EP1959964A1 (xx) |
JP (1) | JP2009517425A (xx) |
KR (1) | KR20080074197A (xx) |
CN (1) | CN101321535A (xx) |
AU (1) | AU2006319381A1 (xx) |
BR (1) | BRPI0619214A2 (xx) |
CA (1) | CA2632279A1 (xx) |
DE (1) | DE102005057421A1 (xx) |
EA (1) | EA200801209A1 (xx) |
EC (1) | ECSP088488A (xx) |
IL (1) | IL191563A0 (xx) |
NO (1) | NO20082916L (xx) |
WO (1) | WO2007062875A1 (xx) |
ZA (1) | ZA200805660B (xx) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN101987104A (zh) * | 2009-08-05 | 2011-03-23 | 天津金耀集团有限公司 | 一种杂芳香基氨磺酰基羧酸酯碳酸酐酶抑制剂的眼用组合物 |
CN101987102A (zh) * | 2009-08-05 | 2011-03-23 | 天津金耀集团有限公司 | 一种糖皮质激素杂芳香基氨磺酰基羧酸酯的眼用抗炎组合物 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1593609A (en) * | 1978-01-31 | 1981-07-22 | Christiaens Sa A | Pyridine sulfonamides |
DE10027887A1 (de) * | 2000-05-31 | 2001-12-13 | Jenapharm Gmbh | Verbindungen mit einer Sulfonamidgruppe und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen |
US6355666B1 (en) * | 2000-06-23 | 2002-03-12 | Medinox, Inc. | Protected forms of pharmacologically active agents and uses therefor |
AR053845A1 (es) * | 2005-04-15 | 2007-05-23 | Tibotec Pharm Ltd | 5-tiazolilmetil[(1s,2r)-3-[[(2-amino-6-benzoxazolil)sulfonil)](2-metilpropil)amino]-2-hidroxi-1-(fenilmetil)propil]carbamato como mejorador de farmacos metabolizados por el citocromo p450 |
-
2005
- 2005-11-30 DE DE102005057421A patent/DE102005057421A1/de not_active Ceased
-
2006
- 2006-11-27 JP JP2008542679A patent/JP2009517425A/ja active Pending
- 2006-11-27 KR KR1020087015778A patent/KR20080074197A/ko not_active Application Discontinuation
- 2006-11-27 EA EA200801209A patent/EA200801209A1/ru unknown
- 2006-11-27 AU AU2006319381A patent/AU2006319381A1/en not_active Abandoned
- 2006-11-27 EP EP06829355A patent/EP1959964A1/de not_active Withdrawn
- 2006-11-27 CA CA002632279A patent/CA2632279A1/en not_active Abandoned
- 2006-11-27 WO PCT/EP2006/011727 patent/WO2007062875A1/de active Application Filing
- 2006-11-27 BR BRPI0619214-9A patent/BRPI0619214A2/pt not_active Application Discontinuation
- 2006-11-27 CN CNA2006800450153A patent/CN101321535A/zh active Pending
-
2008
- 2008-05-20 IL IL191563A patent/IL191563A0/en unknown
- 2008-05-30 EC EC2008008488A patent/ECSP088488A/es unknown
- 2008-06-27 NO NO20082916A patent/NO20082916L/no not_active Application Discontinuation
- 2008-06-27 ZA ZA200805660A patent/ZA200805660B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
NO20082916L (no) | 2008-06-27 |
BRPI0619214A2 (pt) | 2011-09-20 |
WO2007062875B1 (de) | 2007-08-09 |
ZA200805660B (en) | 2009-11-25 |
KR20080074197A (ko) | 2008-08-12 |
AU2006319381A1 (en) | 2007-06-07 |
CA2632279A1 (en) | 2007-06-07 |
IL191563A0 (en) | 2009-08-03 |
CN101321535A (zh) | 2008-12-10 |
ECSP088488A (es) | 2008-06-30 |
EP1959964A1 (de) | 2008-08-27 |
DE102005057421A1 (de) | 2007-05-31 |
WO2007062875A1 (de) | 2007-06-07 |
JP2009517425A (ja) | 2009-04-30 |
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