EA200800464A1 - Фармацевтическая композиция, содержащая периндоприл или его соли - Google Patents

Фармацевтическая композиция, содержащая периндоприл или его соли

Info

Publication number
EA200800464A1
EA200800464A1 EA200800464A EA200800464A EA200800464A1 EA 200800464 A1 EA200800464 A1 EA 200800464A1 EA 200800464 A EA200800464 A EA 200800464A EA 200800464 A EA200800464 A EA 200800464A EA 200800464 A1 EA200800464 A1 EA 200800464A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pharmaceutical composition
salt
composition containing
perindopril
containing perindopril
Prior art date
Application number
EA200800464A
Other languages
English (en)
Inventor
Петер Свете
Original Assignee
Лек Фармасьютиклз Д. Д.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Лек Фармасьютиклз Д. Д. filed Critical Лек Фармасьютиклз Д. Д.
Publication of EA200800464A1 publication Critical patent/EA200800464A1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Medicinal Preparation (AREA)
  • Hospice & Palliative Care (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)

Abstract

Настоящее изобретение относится к стабильной фармацевтической композиции ингибитора АКФ периндоприла или его солей, характеризующихся определенным распределением частиц по размеру.
EA200800464A 2005-08-30 2006-08-28 Фармацевтическая композиция, содержащая периндоприл или его соли EA200800464A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SI200500244 2005-08-30
PCT/EP2006/008400 WO2007025695A1 (en) 2005-08-30 2006-08-28 Pharmaceutical composition comprising perindopril or its salts

Publications (1)

Publication Number Publication Date
EA200800464A1 true EA200800464A1 (ru) 2008-08-29

Family

ID=37564304

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200800464A EA200800464A1 (ru) 2005-08-30 2006-08-28 Фармацевтическая композиция, содержащая периндоприл или его соли

Country Status (9)

Country Link
US (1) US20090136578A1 (ru)
EP (1) EP1937216A1 (ru)
JP (1) JP2009506085A (ru)
CN (1) CN101252915A (ru)
AU (1) AU2006286810A1 (ru)
BR (1) BRPI0615607A2 (ru)
CA (1) CA2619911A1 (ru)
EA (1) EA200800464A1 (ru)
WO (1) WO2007025695A1 (ru)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI22543A (sl) 2007-06-27 2008-12-31 Krka, Tovarna Zdravil, D.D., Novo Mesto Nove soli perindoprila
CN101766598A (zh) * 2008-12-31 2010-07-07 东英(江苏)药业有限公司 含有培哚普利的药物组合物
RU2558099C2 (ru) * 2012-12-11 2015-07-27 Общество с ограниченной ответственностью "Трейдсервис" Комбинированное лекарственное средство для лечения артериальной гипертензии у больных сахарным диабетом
WO2016178591A2 (en) 2015-05-05 2016-11-10 Gene Predit, Sa Genetic markers and treatment of male obesity
CN106620644B (zh) * 2016-12-13 2021-05-25 杭州新诺华医药有限公司 一种稳定的培哚普利吲达帕胺片及制备工艺
CN111419810B (zh) * 2020-04-29 2022-02-11 南京长澳医药科技有限公司 一种高稳定性培哚普利叔丁胺片剂及其制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2771010B1 (fr) * 1997-11-19 2003-08-15 Adir Utilisation d'une combinaison d'un inhibiteur de l'enzyme de conversion de l'angiotensine et d'un diuretique pour le traitement des desordres microcirculatoires
FR2818550B1 (fr) * 2000-12-26 2003-02-07 Servier Lab Composition pharmaceutique solide thermoformable pour la liberation controle de perindopril
US7101573B2 (en) * 2001-09-28 2006-09-05 Mcneil-Pcc, Inc. Simethicone solid oral dosage form
FR2841140B1 (fr) * 2002-06-24 2004-10-01 Servier Lab Microcapsules pour la liberation retardee et controlee du perindopril
BR0318561A (pt) * 2003-10-21 2006-10-10 Lupin Ltd processo seletivo para a preparação de erbumino perindopril cristalino
GB2394660A (en) * 2003-12-17 2004-05-05 Niche Generics Ltd Stabilisation of pharmaceutical compositions comprising ACE inhibitor by absence of acidic excipients having large specific surface area, eg silicon dioxide
EA011712B1 (ru) * 2004-03-29 2009-04-28 Ле Лаборатуар Сервье Способ производства твёрдой фармацевтической композиции
SK50252005A3 (sk) * 2005-03-22 2006-10-05 Vúlm, A.S. Farmaceutický prípravok obsahujúci perindopril erbumín, spôsob jeho prípravy a stabilizácie

Also Published As

Publication number Publication date
WO2007025695A1 (en) 2007-03-08
EP1937216A1 (en) 2008-07-02
JP2009506085A (ja) 2009-02-12
BRPI0615607A2 (pt) 2011-05-24
CN101252915A (zh) 2008-08-27
CA2619911A1 (en) 2007-03-08
AU2006286810A1 (en) 2007-03-08
US20090136578A1 (en) 2009-05-28

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