EA200701296A1 - 3,5-дизамещенные и 3,5,7-тризамещенные 3h-оксазоло- и 3h-тиазоло[4,5-d] пиримидин-2-оны и их пролекарства - Google Patents

3,5-дизамещенные и 3,5,7-тризамещенные 3h-оксазоло- и 3h-тиазоло[4,5-d] пиримидин-2-оны и их пролекарства

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Publication number
EA200701296A1
EA200701296A1 EA200701296A EA200701296A EA200701296A1 EA 200701296 A1 EA200701296 A1 EA 200701296A1 EA 200701296 A EA200701296 A EA 200701296A EA 200701296 A EA200701296 A EA 200701296A EA 200701296 A1 EA200701296 A1 EA 200701296A1
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EA
Eurasian Patent Office
Prior art keywords
oxazolo
thiazolo
pyrimidin
medicines
triple
Prior art date
Application number
EA200701296A
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English (en)
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EA013594B1 (ru
Inventor
Стефен И. Веббер
Грегори Дж. Хейли
Джозеф Р. Леннокс
Алан Синь Сян
Эрик Дж. Руден
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Анадис Фармасьютикалз, Инк.
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Application filed by Анадис Фармасьютикалз, Инк. filed Critical Анадис Фармасьютикалз, Инк.
Publication of EA200701296A1 publication Critical patent/EA200701296A1/ru
Publication of EA013594B1 publication Critical patent/EA013594B1/ru

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Abstract

Изобретение относится к соединениям 3,5-дизамещенных и 3,5,7-тризамещенных 3H-оксазоло- и 3H-тиазоло[4,5-d]пиримидин-2-онов и их пролекарствам, которые имеют иммуномодуляторную активность. Изобретение также относится к терапевтическому или профилактическому применению таких соединений и содержащих их фармацевтических композиций и к способам лечения описанных здесь болезней и расстройств посредством назначения эффективных количеств таких соединений и пролекарств.
EA200701296A 2004-12-17 2005-12-16 3,5-ДИЗАМЕЩЕННЫЕ И 3,5,7-ТРИЗАМЕЩЕННЫЕ 3H-ОКСАЗОЛО- И 3H-ТИАЗОЛО[4,5-d]ПИРИМИДИН-2-ОНЫ И ИХ ПРОЛЕКАРСТВА EA013594B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US63663404P 2004-12-17 2004-12-17
US63663304P 2004-12-17 2004-12-17
PCT/US2005/045589 WO2006066080A1 (en) 2004-12-17 2005-12-16 3, 5-DISUBSTITUTED AND 3,5,7-TRISUBSTITUTED-3H-OXAZOLO AND 3H-THIAZOLO [4,5-d]PYRIMIDIN-2-ONE COMPOUNDS AND PRODRUGS THEREOF

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EA200701296A1 true EA200701296A1 (ru) 2007-12-28
EA013594B1 EA013594B1 (ru) 2010-06-30

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EA200701296A EA013594B1 (ru) 2004-12-17 2005-12-16 3,5-ДИЗАМЕЩЕННЫЕ И 3,5,7-ТРИЗАМЕЩЕННЫЕ 3H-ОКСАЗОЛО- И 3H-ТИАЗОЛО[4,5-d]ПИРИМИДИН-2-ОНЫ И ИХ ПРОЛЕКАРСТВА

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US (4) US7560544B2 (ru)
EP (2) EP2561872B1 (ru)
JP (1) JP5303149B2 (ru)
KR (1) KR101320008B1 (ru)
CN (1) CN102504001B (ru)
AR (1) AR052995A1 (ru)
AU (1) AU2005316397B2 (ru)
BR (1) BRPI0518861B8 (ru)
CA (1) CA2589529C (ru)
DK (2) DK2561872T3 (ru)
EA (1) EA013594B1 (ru)
EG (1) EG25920A (ru)
ES (2) ES2459368T3 (ru)
GT (1) GT200500374A (ru)
HK (2) HK1108377A1 (ru)
IL (2) IL183512A (ru)
MX (1) MX2007007263A (ru)
MY (1) MY176938A (ru)
NO (1) NO20073615L (ru)
NZ (1) NZ555723A (ru)
PA (1) PA8657201A1 (ru)
PE (1) PE20060837A1 (ru)
PL (2) PL2561872T3 (ru)
PT (2) PT1824482E (ru)
SI (2) SI1824482T1 (ru)
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