EA200100148A1 - Лекарственные средства, содержащие производные полигидроксиалкилпиразина, новые производные полигидроксиалкилпиразина и их получение - Google Patents

Лекарственные средства, содержащие производные полигидроксиалкилпиразина, новые производные полигидроксиалкилпиразина и их получение

Info

Publication number
EA200100148A1
EA200100148A1 EA200100148A EA200100148A EA200100148A1 EA 200100148 A1 EA200100148 A1 EA 200100148A1 EA 200100148 A EA200100148 A EA 200100148A EA 200100148 A EA200100148 A EA 200100148A EA 200100148 A1 EA200100148 A1 EA 200100148A1
Authority
EA
Eurasian Patent Office
Prior art keywords
derivatives
denotes
polyhydroxialkylpyrazine
polyhydroxialkylpirazine
new
Prior art date
Application number
EA200100148A
Other languages
English (en)
Other versions
EA003642B1 (ru
Inventor
Жорж Башиард
Жан-Кристоф Карри
Мишель Эвер
Брюно Филош
Серж Миньяни
Original Assignee
Авентис Фарма С.А.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Авентис Фарма С.А. filed Critical Авентис Фарма С.А.
Publication of EA200100148A1 publication Critical patent/EA200100148A1/ru
Publication of EA003642B1 publication Critical patent/EA003642B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/12—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)

Abstract

Изобретение относится к лекарственным средствам, содержащим в качестве активного начала, по меньшей мере одно, соединение формулыв которой Rобозначает цепь -(CHOH)-CHи либо Rобозначает цепь -CH-(CHOH)-CH, а Rобозначает атом водорода, либо Rобозначает атом водорода, а Rобозначает цепь -CH-(CHOH)-CH, или один из его стереоизомеров или одну из его солей с фармацевтически приемлемой минеральной или органической кислотой.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200100148A 1998-07-16 1999-07-13 Лекарственные средства, содержащие производные полигидроксиалкилпиразина, новые производные полигидроксиалкилпиразина и их получение EA003642B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9809088A FR2781155B1 (fr) 1998-07-16 1998-07-16 Medicaments contenant des derives de polyhydroxyalkylpyrazine, les nouveaux derives de polyhydroxyalkylpyrazine et leur preparation
PCT/FR1999/001719 WO2000004002A1 (fr) 1998-07-16 1999-07-13 Derives de polyhydroxyalkylpyrazine et leur preparation et medicaments les contenant

Publications (2)

Publication Number Publication Date
EA200100148A1 true EA200100148A1 (ru) 2001-06-25
EA003642B1 EA003642B1 (ru) 2003-08-28

Family

ID=9528674

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200100148A EA003642B1 (ru) 1998-07-16 1999-07-13 Лекарственные средства, содержащие производные полигидроксиалкилпиразина, новые производные полигидроксиалкилпиразина и их получение

Country Status (22)

Country Link
US (1) US6407110B2 (ru)
EP (1) EP1097145B1 (ru)
JP (1) JP4590099B2 (ru)
KR (1) KR20010071858A (ru)
CN (1) CN1309649A (ru)
AT (1) ATE241604T1 (ru)
AU (1) AU769948B2 (ru)
BR (1) BR9912094A (ru)
CA (1) CA2337350C (ru)
DE (1) DE69908367T2 (ru)
DK (1) DK1097145T3 (ru)
EA (1) EA003642B1 (ru)
ES (1) ES2201729T3 (ru)
FR (1) FR2781155B1 (ru)
HU (1) HUP0103302A3 (ru)
IL (1) IL140751A0 (ru)
NO (1) NO20010244D0 (ru)
NZ (1) NZ509237A (ru)
PL (1) PL345549A1 (ru)
PT (1) PT1097145E (ru)
WO (1) WO2000004002A1 (ru)
ZA (1) ZA200100375B (ru)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6948288B1 (en) * 2000-10-19 2005-09-27 Smith Gary E Roof tile support

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5390401A (en) * 1977-01-13 1978-08-09 Japan Tobacco & Salt Public Improving of smoking taste of cigarette
FR2744365B1 (fr) * 1996-02-06 1998-02-27 Inst Malgache Rech Appl Melanges isolables a partir de graines d'eugenia jambolana lamarck, leur preparation et l'utilisation de ces melanges et certains de leurs constituants comme medicaments

Also Published As

Publication number Publication date
AU4628399A (en) 2000-02-07
FR2781155B1 (fr) 2001-10-26
ZA200100375B (en) 2002-07-12
FR2781155A1 (fr) 2000-01-21
EP1097145A1 (fr) 2001-05-09
CA2337350A1 (fr) 2000-01-27
PT1097145E (pt) 2003-10-31
IL140751A0 (en) 2002-02-10
NO20010244L (no) 2001-01-15
NZ509237A (en) 2003-10-31
BR9912094A (pt) 2001-05-02
ATE241604T1 (de) 2003-06-15
CN1309649A (zh) 2001-08-22
CA2337350C (fr) 2009-06-09
EP1097145B1 (fr) 2003-05-28
DE69908367T2 (de) 2004-03-25
WO2000004002A1 (fr) 2000-01-27
NO20010244D0 (no) 2001-01-15
HUP0103302A2 (hu) 2002-03-28
AU769948B2 (en) 2004-02-12
JP4590099B2 (ja) 2010-12-01
US20010018439A1 (en) 2001-08-30
US6407110B2 (en) 2002-06-18
EA003642B1 (ru) 2003-08-28
PL345549A1 (en) 2001-12-17
JP2002520403A (ja) 2002-07-09
DE69908367D1 (de) 2003-07-03
ES2201729T3 (es) 2004-03-16
KR20010071858A (ko) 2001-07-31
DK1097145T3 (da) 2003-09-15
HUP0103302A3 (en) 2002-05-28

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU