EA200000521A1 - СПОСОБЫ ПОЛУЧЕНИЯ ПИРРОЛО[3,2-b]ПИРИДИНОВ И ПРОМЕЖУТОЧНЫЕ ПРОДУКТЫ - Google Patents

СПОСОБЫ ПОЛУЧЕНИЯ ПИРРОЛО[3,2-b]ПИРИДИНОВ И ПРОМЕЖУТОЧНЫЕ ПРОДУКТЫ

Info

Publication number
EA200000521A1
EA200000521A1 EA200000521A EA200000521A EA200000521A1 EA 200000521 A1 EA200000521 A1 EA 200000521A1 EA 200000521 A EA200000521 A EA 200000521A EA 200000521 A EA200000521 A EA 200000521A EA 200000521 A1 EA200000521 A1 EA 200000521A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pyridine
methods
intermediate products
pyrrolo
producing
Prior art date
Application number
EA200000521A
Other languages
English (en)
Inventor
Винсент Манкузо
Фредди Андре Напора
Уко Эффионг Удодонг
Дэниэл Эдвард II Веррал
Original Assignee
Эли Лилли Энд Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Эли Лилли Энд Компани filed Critical Эли Лилли Энд Компани
Publication of EA200000521A1 publication Critical patent/EA200000521A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Данное изобретение предоставляет способы и промежуточные продукты формулы (I), в которой X и R имеют значения, определенные в описании, для получения 5-амино-3-(1-метилпиперидин-4-ил) пирроло [3,2-b]пиридина.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200000521A 1997-11-14 1998-10-19 СПОСОБЫ ПОЛУЧЕНИЯ ПИРРОЛО[3,2-b]ПИРИДИНОВ И ПРОМЕЖУТОЧНЫЕ ПРОДУКТЫ EA200000521A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6585397P 1997-11-14 1997-11-14
PCT/US1998/022046 WO1999025708A1 (en) 1997-11-14 1998-10-19 PYRROLO[3,2-b]PYRIDINE PROCESSES AND INTERMEDIATES

Publications (1)

Publication Number Publication Date
EA200000521A1 true EA200000521A1 (ru) 2000-10-30

Family

ID=22065573

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200000521A EA200000521A1 (ru) 1997-11-14 1998-10-19 СПОСОБЫ ПОЛУЧЕНИЯ ПИРРОЛО[3,2-b]ПИРИДИНОВ И ПРОМЕЖУТОЧНЫЕ ПРОДУКТЫ

Country Status (25)

Country Link
US (1) US6150525A (ru)
EP (1) EP0916669B1 (ru)
JP (1) JP2001523677A (ru)
KR (1) KR20010024610A (ru)
CN (1) CN1278814A (ru)
AR (1) AR013761A1 (ru)
AT (1) ATE236903T1 (ru)
AU (1) AU9808898A (ru)
BR (1) BR9814158A (ru)
CA (1) CA2309860A1 (ru)
DE (1) DE69813149T2 (ru)
DK (1) DK0916669T3 (ru)
EA (1) EA200000521A1 (ru)
ES (1) ES2196503T3 (ru)
HR (1) HRP20000296A2 (ru)
HU (1) HUP0100429A3 (ru)
ID (1) ID26628A (ru)
IL (1) IL135582A0 (ru)
NO (1) NO20002407L (ru)
NZ (1) NZ503616A (ru)
PL (1) PL340421A1 (ru)
PT (1) PT916669E (ru)
TR (1) TR200001329T2 (ru)
WO (1) WO1999025708A1 (ru)
ZA (1) ZA989389B (ru)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1990007926A1 (en) * 1989-01-20 1990-07-26 Pfizer Inc. 3-(1,2,5,6-tetrahydropyridyl)-pyrrolopyridines
US5521196A (en) * 1994-10-05 1996-05-28 Eli Lilly And Company 5-HT1F agonists for the treatment of migraine
US5521197A (en) * 1994-12-01 1996-05-28 Eli Lilly And Company 3-<1-alkylenearyl>-4-<1,2,3,6-tetrahydropyridinyl>-and 3-<1-alkylenearyl>-4-piperidinyl-1h-indoles: new 5-HT1F agonists
JPH11502816A (ja) * 1995-03-20 1999-03-09 イーライ・リリー・アンド・カンパニー ５−置換−３−（１，２，３，６−テトラヒドロピリジン−４−イル）−および３−（ピペリジン−４−イル）−１ｈ−インドール類：新規５−ｈｔ▲下１ｆ▼アゴニスト
ZA979961B (en) * 1996-11-15 1999-05-05 Lilly Co Eli 5-HT1F agonists

Also Published As

Publication number Publication date
DE69813149T2 (de) 2004-05-06
AU9808898A (en) 1999-06-07
BR9814158A (pt) 2000-09-26
WO1999025708A1 (en) 1999-05-27
NO20002407D0 (no) 2000-05-09
IL135582A0 (en) 2001-05-20
NO20002407L (no) 2000-07-12
DK0916669T3 (da) 2003-04-28
HUP0100429A3 (en) 2001-12-28
EP0916669A2 (en) 1999-05-19
AR013761A1 (es) 2001-01-10
JP2001523677A (ja) 2001-11-27
US6150525A (en) 2000-11-21
CN1278814A (zh) 2001-01-03
ES2196503T3 (es) 2003-12-16
EP0916669A3 (en) 2001-05-23
CA2309860A1 (en) 1999-05-27
DE69813149D1 (de) 2003-05-15
HRP20000296A2 (en) 2000-08-31
PL340421A1 (en) 2001-02-12
KR20010024610A (ko) 2001-03-26
ZA989389B (en) 2000-04-14
TR200001329T2 (tr) 2001-01-22
HUP0100429A2 (hu) 2001-08-28
EP0916669B1 (en) 2003-04-09
NZ503616A (en) 2001-06-29
ATE236903T1 (de) 2003-04-15
ID26628A (id) 2001-01-25
PT916669E (pt) 2003-07-31

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