EA199800028A1 - Винилсульфоксиды и способы их синтеза - Google Patents

Винилсульфоксиды и способы их синтеза

Info

Publication number
EA199800028A1
EA199800028A1 EA199800028A EA199800028A EA199800028A1 EA 199800028 A1 EA199800028 A1 EA 199800028A1 EA 199800028 A EA199800028 A EA 199800028A EA 199800028 A EA199800028 A EA 199800028A EA 199800028 A1 EA199800028 A1 EA 199800028A1
Authority
EA
Eurasian Patent Office
Prior art keywords
synthesis
vinylsulphoxides
methods
new
diarylvinyl
Prior art date
Application number
EA199800028A
Other languages
English (en)
Other versions
EA000405B1 (ru
Inventor
Джеймс А. Айкинс
Рэндэл С. Миллер
Тони Й. Занг
Original Assignee
Эли Лилли Энд Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/483,130 external-priority patent/US6372945B1/en
Priority claimed from US08/478,706 external-priority patent/US5659087A/en
Application filed by Эли Лилли Энд Компани filed Critical Эли Лилли Энд Компани
Publication of EA199800028A1 publication Critical patent/EA199800028A1/ru
Publication of EA000405B1 publication Critical patent/EA000405B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/16—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C317/18—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton with sulfone or sulfoxide groups bound to acyclic carbon atoms of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)

Abstract

В настоящем изобретении предложены новые диарилвинилсульфоксиды и новый способ их синтеза.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA199800028A 1995-06-07 1996-06-04 Винилсульфоксиды и способ их синтеза EA000405B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/483,130 US6372945B1 (en) 1995-06-07 1995-06-07 Process for the synthesis of vinyl sulfoxides
US08/478,706 US5659087A (en) 1995-06-07 1995-06-07 Diarylvinyl sulfoxides
PCT/US1996/009163 WO1996040691A1 (en) 1995-06-07 1996-06-04 Vinyl sulfoxides and a process for their synthesis

Publications (2)

Publication Number Publication Date
EA199800028A1 true EA199800028A1 (ru) 1998-08-27
EA000405B1 EA000405B1 (ru) 1999-06-24

Family

ID=27045988

Family Applications (1)

Application Number Title Priority Date Filing Date
EA199800028A EA000405B1 (ru) 1995-06-07 1996-06-04 Винилсульфоксиды и способ их синтеза

Country Status (16)

Country Link
EP (1) EP0830361A4 (ru)
JP (1) JPH11507061A (ru)
KR (1) KR19990022362A (ru)
CN (2) CN1192741A (ru)
AU (1) AU697352B2 (ru)
BR (1) BR9608579A (ru)
CA (1) CA2220145A1 (ru)
CZ (1) CZ393097A3 (ru)
EA (1) EA000405B1 (ru)
HU (1) HUP9900922A3 (ru)
IL (1) IL122090A0 (ru)
NO (2) NO975578L (ru)
NZ (1) NZ310179A (ru)
PL (1) PL324035A1 (ru)
TR (3) TR199801495T2 (ru)
WO (1) WO1996040691A1 (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE60020954T2 (de) * 1999-04-02 2006-05-11 Temple University Of The Commonwealth System Of Higher Education (e)-styrylsulfone als krebsbestreitende mittel
AU2003266940B2 (en) 2002-09-30 2007-02-08 A/S Gea Farmaceutisk Fabrik Novel raloxifene acid addition salts and/or solvates thereof, improved method for purification of said raloxifene acid addition salts and/or solvates thereof and pharmaceutical compositions comprising these

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5512701A (en) * 1995-06-07 1996-04-30 Eli Lilly And Company Process for the synthesis of vinyl sulfenic acid derivatives
US5514826A (en) * 1995-06-07 1996-05-07 Eli Lilly And Company Vinyl sulfenic acid derivatives
IL122127A (en) * 1995-06-07 2001-05-20 Lilly Co Eli Derivatives of sulfonic vinyl acids, process for their preparation and use in the synthesis of benzo [b]

Also Published As

Publication number Publication date
HUP9900922A2 (hu) 1999-07-28
NO20005987D0 (no) 2000-11-27
NZ310179A (en) 1999-09-29
CA2220145A1 (en) 1996-12-19
HUP9900922A3 (en) 2000-06-28
CN1341596A (zh) 2002-03-27
TR199801495T2 (xx) 1998-09-21
WO1996040691A1 (en) 1996-12-19
PL324035A1 (en) 1998-05-11
TR199701510T1 (xx) 1998-03-21
CZ393097A3 (cs) 1998-06-17
AU6092096A (en) 1996-12-30
NO975578D0 (no) 1997-12-03
KR19990022362A (ko) 1999-03-25
EP0830361A1 (en) 1998-03-25
AU697352B2 (en) 1998-10-01
TR199801494T2 (xx) 1998-09-21
IL122090A0 (en) 1998-04-05
CN1192741A (zh) 1998-09-09
BR9608579A (pt) 1999-01-05
NO975578L (no) 1997-12-03
JPH11507061A (ja) 1999-06-22
EP0830361A4 (en) 1998-12-30
EA000405B1 (ru) 1999-06-24
NO5987A (no) 1997-12-03

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU