EA032294B1 - Способ получения полиморфной формы производного n-(ариламино)сульфонамида, фармацевтическая композиция, содержащая указанное производное, и способ лечения с помощью указанного производного - Google Patents
Способ получения полиморфной формы производного n-(ариламино)сульфонамида, фармацевтическая композиция, содержащая указанное производное, и способ лечения с помощью указанного производного Download PDFInfo
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- EA032294B1 EA032294B1 EA201400552A EA201400552A EA032294B1 EA 032294 B1 EA032294 B1 EA 032294B1 EA 201400552 A EA201400552 A EA 201400552A EA 201400552 A EA201400552 A EA 201400552A EA 032294 B1 EA032294 B1 EA 032294B1
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- additional embodiments
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- cancer
- iodophenylamino
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| Application Number | Priority Date | Filing Date | Title |
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| US11/830,733 US8101799B2 (en) | 2005-07-21 | 2007-07-30 | Derivatives of N-(arylamino) sulfonamides as inhibitors of MEK |
| US3446408P | 2008-03-06 | 2008-03-06 | |
| US3446608P | 2008-03-06 | 2008-03-06 | |
| US4488608P | 2008-04-14 | 2008-04-14 |
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| EA201400552A1 EA201400552A1 (ru) | 2014-09-30 |
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| EA201400552A EA032294B1 (ru) | 2007-07-30 | 2008-07-28 | Способ получения полиморфной формы производного n-(ариламино)сульфонамида, фармацевтическая композиция, содержащая указанное производное, и способ лечения с помощью указанного производного |
| EA201000268A EA020624B1 (ru) | 2007-07-30 | 2008-07-28 | Кристаллическая полиморфная форма n-(-)-(3,4-дифтор-2-(2-фтор-4-йодфениламино)-6-метоксифенил)-l-(2,3-дигидроксипропил)циклопропан-1-сульфонамида и ее применение в качестве ингибитора mek |
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| EA201000268A EA020624B1 (ru) | 2007-07-30 | 2008-07-28 | Кристаллическая полиморфная форма n-(-)-(3,4-дифтор-2-(2-фтор-4-йодфениламино)-6-метоксифенил)-l-(2,3-дигидроксипропил)циклопропан-1-сульфонамида и ее применение в качестве ингибитора mek |
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| BR122021020474B1 (pt) * | 2008-09-09 | 2022-06-07 | F. Hoffmann-La Roche Ag | Polimorfos de acil sulfonamidas, seu uso, seu processo de preparação e composição farmacêutica que os compreende |
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| PE20120105A1 (es) | 2009-03-11 | 2012-02-22 | Ardea Biosciences Inc | Combinaciones farmaceuticas que comprenden refametinib |
| UY32486A (es) * | 2009-03-11 | 2010-10-29 | Ardea Biosciences Inc | Tratamiento del cáncer de páncreas |
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