EA022988B9 - Соединения фенилкетонкарбоксилата и их фармацевтическое применение - Google Patents

Соединения фенилкетонкарбоксилата и их фармацевтическое применение

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Publication number
EA022988B9
EA022988B9 EA201370104A EA201370104A EA022988B9 EA 022988 B9 EA022988 B9 EA 022988B9 EA 201370104 A EA201370104 A EA 201370104A EA 201370104 A EA201370104 A EA 201370104A EA 022988 B9 EA022988 B9 EA 022988B9
Authority
EA
Eurasian Patent Office
Prior art keywords
compounds
diseases
phenylketonkarboxylate
pharmaceutical applications
kidney diseases
Prior art date
Application number
EA201370104A
Other languages
English (en)
Russian (ru)
Other versions
EA022988B1 (ru
EA201370104A1 (ru
Inventor
Було Закари
Кристофер Пенне
Шон Эбботт
Лин Ганьон
Брижит Груа
Пьер Лорин
Жан-Франсуа Бьенвэню
Original Assignee
Прометик Биосайнсиз Инк.
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45992998&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA022988(B9) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Прометик Биосайнсиз Инк. filed Critical Прометик Биосайнсиз Инк.
Publication of EA201370104A1 publication Critical patent/EA201370104A1/ru
Publication of EA022988B1 publication Critical patent/EA022988B1/ru
Publication of EA022988B9 publication Critical patent/EA022988B9/ru

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    • C07C59/40—Unsaturated compounds
    • C07C59/76—Unsaturated compounds containing keto groups
    • C07C59/90—Unsaturated compounds containing keto groups containing singly bound oxygen-containing groups
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • A61K31/222—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin with compounds having aromatic groups, e.g. dipivefrine, ibopamine
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    • C07C217/82—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings of the same non-condensed six-membered aromatic ring
    • C07C217/84—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings of the same non-condensed six-membered aromatic ring the oxygen atom of at least one of the etherified hydroxy groups being further bound to an acyclic carbon atom
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EA201370104A 2010-10-27 2011-10-26 Соединения фенилкетонкарбоксилата и их фармацевтическое применение EA022988B9 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40706810P 2010-10-27 2010-10-27
PCT/CA2011/001176 WO2012055014A1 (en) 2010-10-27 2011-10-26 Phenylketone carboxylate compounds and pharmaceutical uses thereof

Publications (3)

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