EA019865B1 - Лекарственная форма, содержащая 1{6-[(3-циклобутил-2,3,4,5-тетрагидро-1н-3-бензазепин-7-ил)окси]-3-пиридинил}-2-пирролидинон или его соль и стабилизатор, который уменьшает его деградацию - Google Patents
Лекарственная форма, содержащая 1{6-[(3-циклобутил-2,3,4,5-тетрагидро-1н-3-бензазепин-7-ил)окси]-3-пиридинил}-2-пирролидинон или его соль и стабилизатор, который уменьшает его деградацию Download PDFInfo
- Publication number
- EA019865B1 EA019865B1 EA200970817A EA200970817A EA019865B1 EA 019865 B1 EA019865 B1 EA 019865B1 EA 200970817 A EA200970817 A EA 200970817A EA 200970817 A EA200970817 A EA 200970817A EA 019865 B1 EA019865 B1 EA 019865B1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- dosage form
- cyclobutyl
- tetrahydro
- pyridinyl
- oxy
- Prior art date
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Landscapes
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| PCT/EP2008/052430 WO2008104590A2 (en) | 2007-03-01 | 2008-02-28 | Novel dosage form |
Publications (2)
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| EA200970817A1 EA200970817A1 (ru) | 2010-06-30 |
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| US9108948B2 (en) | 2006-06-23 | 2015-08-18 | Abbvie Inc. | Cyclopropyl amine derivatives |
| CN103382174A (zh) | 2006-06-23 | 2013-11-06 | 雅培制药有限公司 | 作为组胺h3受体调节物的环丙胺衍生物 |
| EP2328587A1 (en) * | 2008-08-29 | 2011-06-08 | Glaxo Group Limited | Dosage form comprising 1-isopropyl-4-{ [4-(tetrahydro-2h-pyran- 4-yloxy)phenyl]carbonyl}hexahydro-1h-1,4-diazepine or a salt thereof |
| US9186353B2 (en) * | 2009-04-27 | 2015-11-17 | Abbvie Inc. | Treatment of osteoarthritis pain |
| WO2011051423A1 (en) | 2009-11-02 | 2011-05-05 | Glaxo Group Limited | Treatment or prophylaxis of dementia, neurodegenerative disorders, schizophrenia, adhd, somnolence or epilepsy |
| US8853390B2 (en) | 2010-09-16 | 2014-10-07 | Abbvie Inc. | Processes for preparing 1,2-substituted cyclopropyl derivatives |
| US20130244943A1 (en) | 2011-09-06 | 2013-09-19 | Allergan, Inc. | Hyaluronic acid-collagen matrices for dermal filling and volumizing applications |
| EP3233087B1 (en) | 2014-12-16 | 2019-10-02 | Axovant Sciences GmbH | Geminal substituted quinuclidine amide compounds as agonists of alpha-7 nicotinic acetylcholine receptors |
| AU2016274694A1 (en) | 2015-06-10 | 2018-01-18 | Axovant Sciences Gmbh | Aminobenzisoxazole compounds as agonists of A7-nicotinic acetylcholine receptors |
| JP2018523707A (ja) | 2015-08-12 | 2018-08-23 | アクソバント サイエンシズ ゲーエムベーハー | α７−ニコチン性アセチルコリン受容体のアゴニストとしてのジェミナル置換アミノベンゾイソオキサゾール化合物 |
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| WO2004056369A1 (en) * | 2002-12-20 | 2004-07-08 | Glaxo Group Limited | Benzo ‘ d!azepine derivatives for the treatment of neurological disorders |
| WO2005042491A1 (en) * | 2003-10-22 | 2005-05-12 | Arena Pharmaceuticals, Inc. | Benzazepine derivatives and methods of prophylaxis or treatment of 5ht2c receptor associated diseases |
| WO2005123723A1 (en) * | 2004-06-18 | 2005-12-29 | Glaxo Group Limited | 3-cycloalkylbenzazepines as histamine h3 antagonists |
| WO2006018260A1 (en) * | 2004-08-16 | 2006-02-23 | Glaxo Group Limited | Tetrahydrobenzazepines as antagonists and/or reverse agonists of the histamine h 3 receptor |
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| AU7719894A (en) * | 1993-09-03 | 1995-03-22 | Smithkline Beecham Corporation | Stabilized tablet formulation |
| IL143299A0 (en) * | 1998-12-01 | 2002-04-21 | Novo Nordisk As | Pharmaceutical composition comprising 5-[[4- [3-methyl-4-oxo-3, 4-dihydro-2-quinazolinyl] methoxy] phenyl-methyl] thiadiazolidine-2, 4-dione and the process for its preparation |
| US20040037869A1 (en) * | 2002-08-16 | 2004-02-26 | Douglas Cleverly | Non-animal product containing veterinary formulations |
| CA2529320C (en) * | 2003-06-17 | 2013-03-05 | Arena Pharmaceuticals, Inc. | Benzazepine derivatives useful for the treatment of 5ht2c receptor associated diseases |
| US20070021391A1 (en) * | 2003-06-30 | 2007-01-25 | Takayuki Doi | Preventive/remedy for urinary disturbance |
| US20060002986A1 (en) * | 2004-06-09 | 2006-01-05 | Smithkline Beecham Corporation | Pharmaceutical product |
| JP2006022039A (ja) * | 2004-07-08 | 2006-01-26 | Towa Yakuhin Kk | 高い安定性を有するシンバスタチン固形製剤 |
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2008
- 2008-02-27 CL CL200800596A patent/CL2008000596A1/es unknown
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2004056369A1 (en) * | 2002-12-20 | 2004-07-08 | Glaxo Group Limited | Benzo ‘ d!azepine derivatives for the treatment of neurological disorders |
| WO2005042491A1 (en) * | 2003-10-22 | 2005-05-12 | Arena Pharmaceuticals, Inc. | Benzazepine derivatives and methods of prophylaxis or treatment of 5ht2c receptor associated diseases |
| WO2005123723A1 (en) * | 2004-06-18 | 2005-12-29 | Glaxo Group Limited | 3-cycloalkylbenzazepines as histamine h3 antagonists |
| WO2006018260A1 (en) * | 2004-08-16 | 2006-02-23 | Glaxo Group Limited | Tetrahydrobenzazepines as antagonists and/or reverse agonists of the histamine h 3 receptor |
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| MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
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