EA011169B1 - Система подкожной доставки, способ ее получения и ее применение для лечения холинергических дефицитных расстройств - Google Patents
Система подкожной доставки, способ ее получения и ее применение для лечения холинергических дефицитных расстройств Download PDFInfo
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- EA011169B1 EA011169B1 EA200501433A EA200501433A EA011169B1 EA 011169 B1 EA011169 B1 EA 011169B1 EA 200501433 A EA200501433 A EA 200501433A EA 200501433 A EA200501433 A EA 200501433A EA 011169 B1 EA011169 B1 EA 011169B1
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Classifications
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- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
- A61K9/204—Polyesters, e.g. poly(lactide-co-glycolide)
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- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
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- A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Psychiatry (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Toxicology (AREA)
- Dermatology (AREA)
- Hospice & Palliative Care (AREA)
- Addiction (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Thermotherapy And Cooling Therapy Devices (AREA)
- Percussion Or Vibration Massage (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IB0300942 | 2003-03-14 | ||
| IB0304945 | 2003-11-05 | ||
| PCT/IB2004/000734 WO2004080436A1 (en) | 2003-03-14 | 2004-03-15 | Subcutaneous delivery system, process for the preparation of the same and use of the same for the treatment of cholinergic deficient disorders |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA200501433A1 EA200501433A1 (ru) | 2006-02-24 |
| EA011169B1 true EA011169B1 (ru) | 2009-02-27 |
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| EA200501433A EA011169B1 (ru) | 2003-03-14 | 2004-03-15 | Система подкожной доставки, способ ее получения и ее применение для лечения холинергических дефицитных расстройств |
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| EP (2) | EP1603532B1 (enExample) |
| JP (1) | JP2006520378A (enExample) |
| KR (1) | KR20060023111A (enExample) |
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| BR (1) | BRPI0407818A (enExample) |
| CA (1) | CA2518883A1 (enExample) |
| CY (1) | CY1108482T1 (enExample) |
| DE (1) | DE602004015744D1 (enExample) |
| DK (1) | DK1603532T3 (enExample) |
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| ES (1) | ES2312981T3 (enExample) |
| IL (1) | IL170759A (enExample) |
| IS (1) | IS8067A (enExample) |
| MX (1) | MXPA05009626A (enExample) |
| NO (1) | NO20054258L (enExample) |
| NZ (1) | NZ542459A (enExample) |
| PL (1) | PL1603532T3 (enExample) |
| PT (1) | PT1603532E (enExample) |
| SI (1) | SI1603532T1 (enExample) |
| UA (1) | UA82226C2 (enExample) |
| WO (1) | WO2004080436A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2432556T3 (es) | 2004-08-04 | 2013-12-04 | Evonik Corporation | Métodos para fabricar dispositivos de suministro y sus dispositivos |
| US8124601B2 (en) * | 2007-11-21 | 2012-02-28 | Bristol-Myers Squibb Company | Compounds for the treatment of Hepatitis C |
| EP2222281B1 (en) | 2007-12-20 | 2018-12-05 | Evonik Corporation | Process for preparing microparticles having a low residual solvent volume |
| US8956636B2 (en) * | 2008-04-18 | 2015-02-17 | Warsaw Orthopedic, Inc. | Methods and compositions for treating postoperative pain comprosing ketorolac |
| WO2011132157A1 (en) | 2010-04-22 | 2011-10-27 | Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. | Oral sustained release formulation of huperzine a |
| WO2013173096A2 (en) * | 2012-05-18 | 2013-11-21 | Insero Health Inc. | Conjugates of huperzine and analogs thereof |
| KR101811797B1 (ko) * | 2013-04-03 | 2017-12-22 | 동국제약 주식회사 | 도네페질을 포함하는 비경구투여용 약제학적 조성물 |
| JP7111375B2 (ja) * | 2017-10-19 | 2022-08-02 | 株式会社佐藤園 | 学習記憶能力増強組成物 |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0806416A1 (en) * | 1994-12-28 | 1997-11-12 | Tsumura & Co. | Huperzine a derivatives, their preparation and their use |
| WO2003004024A1 (en) * | 2001-07-03 | 2003-01-16 | Shandong Luye Pharmaceutical Co., Ltd. | Injectable sustained-release microspheres of huperzine a compounds |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5106979A (en) * | 1989-02-21 | 1992-04-21 | University Of Pittsburgh | Method for the synthesis of huperzine A and analogs thereof and compounds useful therein |
| FR2756493B1 (fr) * | 1996-12-02 | 2001-04-13 | Delab | Dispositif d'administration locale de formulations solides ou semi-solides |
| US6352715B1 (en) | 1998-02-19 | 2002-03-05 | Sagittarius Life Science Corp | Transdermal rate-controlled delivery of Huperzine A for treatment of alzheimer's disease |
| US6565874B1 (en) * | 1998-10-28 | 2003-05-20 | Atrix Laboratories | Polymeric delivery formulations of leuprolide with improved efficacy |
| CN1279065A (zh) | 1999-07-06 | 2001-01-10 | 青岛科达生物工程有限公司 | 一种治疗记忆障碍和老年痴呆的药物组合物 |
| CN1383824A (zh) | 2002-05-21 | 2002-12-11 | 浙江省医学科学院 | 石杉碱鼻腔给药制剂 |
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2004
- 2004-03-15 ES ES04720662T patent/ES2312981T3/es not_active Expired - Lifetime
- 2004-03-15 SI SI200430920T patent/SI1603532T1/sl unknown
- 2004-03-15 JP JP2006506340A patent/JP2006520378A/ja active Pending
- 2004-03-15 EA EA200501433A patent/EA011169B1/ru not_active IP Right Cessation
- 2004-03-15 KR KR1020057016999A patent/KR20060023111A/ko not_active Ceased
- 2004-03-15 BR BRPI0407818-7A patent/BRPI0407818A/pt not_active IP Right Cessation
- 2004-03-15 EP EP04720662A patent/EP1603532B1/en not_active Expired - Lifetime
- 2004-03-15 UA UAA200509681A patent/UA82226C2/uk unknown
- 2004-03-15 AU AU2004218896A patent/AU2004218896B2/en not_active Ceased
- 2004-03-15 DE DE602004015744T patent/DE602004015744D1/de not_active Expired - Lifetime
- 2004-03-15 DK DK04720662T patent/DK1603532T3/da active
- 2004-03-15 EP EP08159962A patent/EP1977735A1/en not_active Withdrawn
- 2004-03-15 WO PCT/IB2004/000734 patent/WO2004080436A1/en not_active Ceased
- 2004-03-15 PT PT04720662T patent/PT1603532E/pt unknown
- 2004-03-15 CA CA002518883A patent/CA2518883A1/en not_active Abandoned
- 2004-03-15 US US10/549,167 patent/US20070059369A1/en not_active Abandoned
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- 2004-03-15 NZ NZ542459A patent/NZ542459A/en unknown
- 2004-03-15 AT AT04720662T patent/ATE404170T1/de not_active IP Right Cessation
- 2004-03-15 PL PL04720662T patent/PL1603532T3/pl unknown
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2005
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- 2005-09-15 NO NO20054258A patent/NO20054258L/no not_active Application Discontinuation
- 2005-10-11 IS IS8067A patent/IS8067A/is unknown
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2008
- 2008-11-06 CY CY20081101257T patent/CY1108482T1/el unknown
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0806416A1 (en) * | 1994-12-28 | 1997-11-12 | Tsumura & Co. | Huperzine a derivatives, their preparation and their use |
| WO2003004024A1 (en) * | 2001-07-03 | 2003-01-16 | Shandong Luye Pharmaceutical Co., Ltd. | Injectable sustained-release microspheres of huperzine a compounds |
Non-Patent Citations (3)
| Title |
|---|
| DATABASE CHEMABS 'Online! CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; LIU, WANHUI ET AL.: "Injectable release-sustained microsphere of huperzine A, its derivative, or its salt and its preparation", XP002289907, retrieved from STN, Database accession no. 140:327054, abstract & CN 1393220 CN (GREEN LEAF PHARMACEUTICAL CO., LTD., SHANDONG, PEOP. REP. CHINA) 3 July 2001 (2001-07-03) * |
| DATABASE CHEMABS 'Online! CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; LIU, WANHUI ET AL.: "Injectable sustained-release microspheres of huperzine A compounds", XP002289908, retrieved from STN, Database accession no. 138:112410, abstract & WO 03/004024 A1 (SHANDONG LUYE PHARMACEUTICAL CO., LTD., PEOP. REP. CHINA) 16 January 2003 (2003-01-16) * |
| LALLEMENT G. ET AL.: '"New prospect for pretreatment of organophosphate intoxication: Huperzine. A. Experimental data.!" MEDECINE ET ARMEES, vol. 30, no. 3, 2002, pages 219-224, XP008033273, ISSN: 0300-4937 * |
Also Published As
| Publication number | Publication date |
|---|---|
| IL170759A (en) | 2010-06-16 |
| EP1977735A1 (en) | 2008-10-08 |
| EP1603532A1 (en) | 2005-12-14 |
| DK1603532T3 (da) | 2008-12-08 |
| AU2004218896A1 (en) | 2004-09-23 |
| HK1089085A1 (zh) | 2006-11-24 |
| ES2312981T3 (es) | 2009-03-01 |
| NZ542459A (en) | 2008-12-24 |
| AU2004218896B2 (en) | 2010-04-01 |
| SI1603532T1 (sl) | 2009-02-28 |
| DE602004015744D1 (de) | 2008-09-25 |
| IS8067A (is) | 2005-10-11 |
| CA2518883A1 (en) | 2004-09-23 |
| US20070059369A1 (en) | 2007-03-15 |
| EA200501433A1 (ru) | 2006-02-24 |
| PL1603532T3 (pl) | 2009-02-27 |
| CY1108482T1 (el) | 2014-04-09 |
| NO20054258D0 (no) | 2005-09-15 |
| WO2004080436A1 (en) | 2004-09-23 |
| MXPA05009626A (es) | 2005-10-18 |
| NO20054258L (no) | 2005-11-24 |
| EP1603532B1 (en) | 2008-08-13 |
| PT1603532E (pt) | 2008-11-20 |
| ATE404170T1 (de) | 2008-08-15 |
| JP2006520378A (ja) | 2006-09-07 |
| BRPI0407818A (pt) | 2006-02-14 |
| KR20060023111A (ko) | 2006-03-13 |
| UA82226C2 (uk) | 2008-03-25 |
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