EA004512B1 - Циклокарбаматные производные в качестве модуляторов рецептора прогестерона - Google Patents
Циклокарбаматные производные в качестве модуляторов рецептора прогестерона Download PDFInfo
- Publication number
- EA004512B1 EA004512B1 EA200101176A EA200101176A EA004512B1 EA 004512 B1 EA004512 B1 EA 004512B1 EA 200101176 A EA200101176 A EA 200101176A EA 200101176 A EA200101176 A EA 200101176A EA 004512 B1 EA004512 B1 EA 004512B1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- substituted
- alkyl
- oxazin
- alkoxy
- dimethyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/18—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US18301299P | 1999-05-04 | 1999-05-04 | |
| US09/552,633 US6509334B1 (en) | 1999-05-04 | 2000-04-19 | Cyclocarbamate derivatives as progesterone receptor modulators |
| PCT/US2000/011822 WO2000066571A1 (en) | 1999-05-04 | 2000-05-01 | Cyclocarbamate derivatives as progesterone receptor modulators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA200101176A1 EA200101176A1 (ru) | 2002-04-25 |
| EA004512B1 true EA004512B1 (ru) | 2004-04-29 |
Family
ID=26878647
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA200101176A EA004512B1 (ru) | 1999-05-04 | 2000-05-01 | Циклокарбаматные производные в качестве модуляторов рецептора прогестерона |
Country Status (19)
| Country | Link |
|---|---|
| EP (1) | EP1173426A1 (tr) |
| JP (1) | JP2002543193A (tr) |
| KR (1) | KR20010114250A (tr) |
| CN (1) | CN1145618C (tr) |
| AU (1) | AU766428B2 (tr) |
| BG (1) | BG106079A (tr) |
| BR (1) | BR0010213A (tr) |
| CA (1) | CA2371726A1 (tr) |
| CZ (1) | CZ20013951A3 (tr) |
| EA (1) | EA004512B1 (tr) |
| HU (1) | HUP0201609A3 (tr) |
| IL (1) | IL146280A0 (tr) |
| MX (1) | MXPA01011286A (tr) |
| NO (1) | NO321361B1 (tr) |
| NZ (1) | NZ515355A (tr) |
| PL (1) | PL351127A1 (tr) |
| SG (1) | SG114650A1 (tr) |
| SK (1) | SK15912001A3 (tr) |
| TR (1) | TR200103286T2 (tr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL1756095T3 (pl) * | 2004-04-27 | 2008-10-31 | Wyeth Corp | Cyjanopirole zawierające cykliczne karbaminianowe i tiokarbaminianowe biaryle oraz sposoby ich wytwarzania |
| JPWO2006077821A1 (ja) * | 2005-01-19 | 2008-06-19 | 大日本住友製薬株式会社 | アルドステロン受容体調節剤としての芳香族スルホン化合物 |
| CA2701406C (en) | 2007-10-05 | 2016-01-26 | Banyu Pharmaceutical Co., Ltd. | Benzoxazinone derivative |
| CN111925353B (zh) * | 2020-08-31 | 2022-04-08 | 苏州大学附属第二医院 | 一种2-噻吩甲腈的制备方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0510235A1 (en) * | 1991-04-26 | 1992-10-28 | Dong-A Pharm. Co., Ltd. | Novel benzoxazine or benzothiazine derivatives and process for the preparation of the same |
| WO1995020389A1 (en) * | 1994-01-28 | 1995-08-03 | Merck & Co., Inc. | Benzoxazinones as inhibitors of hiv reverse transcriptase |
| EP1382597A3 (en) * | 1994-12-22 | 2004-04-07 | Ligand Pharmaceuticals, Inc. | Steroid receptor modulator compounds and methods |
| EP0929533B1 (en) * | 1996-10-02 | 2003-09-03 | Bristol-Myers Squibb Pharma Company | 4,4-disubstituted-1,4-dihydro-2h-3,1-benzoxazin-2-ones useful as hiv reverse transcriptase inhibitors and intermediates and processes for making the same |
-
2000
- 2000-05-01 EP EP00928689A patent/EP1173426A1/en not_active Withdrawn
- 2000-05-01 CZ CZ20013951A patent/CZ20013951A3/cs unknown
- 2000-05-01 MX MXPA01011286A patent/MXPA01011286A/es unknown
- 2000-05-01 EA EA200101176A patent/EA004512B1/ru not_active IP Right Cessation
- 2000-05-01 NZ NZ515355A patent/NZ515355A/xx unknown
- 2000-05-01 CA CA002371726A patent/CA2371726A1/en not_active Abandoned
- 2000-05-01 SK SK1591-2001A patent/SK15912001A3/sk unknown
- 2000-05-01 KR KR1020017013970A patent/KR20010114250A/ko not_active Application Discontinuation
- 2000-05-01 AU AU46886/00A patent/AU766428B2/en not_active Ceased
- 2000-05-01 JP JP2000615601A patent/JP2002543193A/ja active Pending
- 2000-05-01 SG SG200400080A patent/SG114650A1/en unknown
- 2000-05-01 BR BR0010213-0A patent/BR0010213A/pt not_active Application Discontinuation
- 2000-05-01 HU HU0201609A patent/HUP0201609A3/hu unknown
- 2000-05-01 CN CNB008071004A patent/CN1145618C/zh not_active Expired - Fee Related
- 2000-05-01 PL PL00351127A patent/PL351127A1/xx not_active Application Discontinuation
- 2000-05-01 TR TR2001/03286T patent/TR200103286T2/tr unknown
- 2000-05-01 IL IL14628000A patent/IL146280A0/xx unknown
-
2001
- 2001-11-02 BG BG106079A patent/BG106079A/xx unknown
- 2001-11-02 NO NO20015378A patent/NO321361B1/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CN1145618C (zh) | 2004-04-14 |
| AU766428B2 (en) | 2003-10-16 |
| AU4688600A (en) | 2000-11-17 |
| NZ515355A (en) | 2004-02-27 |
| JP2002543193A (ja) | 2002-12-17 |
| EA200101176A1 (ru) | 2002-04-25 |
| MXPA01011286A (es) | 2003-07-14 |
| KR20010114250A (ko) | 2001-12-31 |
| CN1349517A (zh) | 2002-05-15 |
| EP1173426A1 (en) | 2002-01-23 |
| CA2371726A1 (en) | 2000-11-09 |
| TR200103286T2 (tr) | 2002-07-22 |
| NO20015378D0 (no) | 2001-11-02 |
| SG114650A1 (en) | 2005-09-28 |
| BG106079A (en) | 2002-05-31 |
| PL351127A1 (en) | 2003-03-24 |
| BR0010213A (pt) | 2002-02-19 |
| SK15912001A3 (sk) | 2002-06-04 |
| CZ20013951A3 (cs) | 2002-05-15 |
| IL146280A0 (en) | 2002-07-25 |
| NO321361B1 (no) | 2006-05-02 |
| HUP0201609A2 (en) | 2002-08-28 |
| NO20015378L (no) | 2002-01-03 |
| HUP0201609A3 (en) | 2002-12-28 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US6509334B1 (en) | Cyclocarbamate derivatives as progesterone receptor modulators | |
| US6436929B1 (en) | Cyclothiocarbamate derivatives as progesterone receptor modulators | |
| US6444668B1 (en) | Combination regimens using progesterone receptor modulators | |
| CA2371712C (en) | Cyclothiocarbamate derivatives as progesterone receptor modulators | |
| EP1173210B1 (en) | Contraceptive compositions containing antiprogestinic and progestinic | |
| EA004512B1 (ru) | Циклокарбаматные производные в качестве модуляторов рецептора прогестерона |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PD4A | Registration of transfer of a eurasian patent in accordance with the succession in title | ||
| MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM |
|
| MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): RU |