DK625184A - Benzoxazinderivater - Google Patents
Benzoxazinderivater Download PDFInfo
- Publication number
- DK625184A DK625184A DK625184A DK625184A DK625184A DK 625184 A DK625184 A DK 625184A DK 625184 A DK625184 A DK 625184A DK 625184 A DK625184 A DK 625184A DK 625184 A DK625184 A DK 625184A
- Authority
- DK
- Denmark
- Prior art keywords
- benzoxazine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/18—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C265/00—Derivatives of isocyanic acid
- C07C265/16—Derivatives of isocyanic acid having isocyanate groups acylated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C273/00—Preparation of urea or its derivatives, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C273/18—Preparation of urea or its derivatives, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups of substituted ureas
- C07C273/1809—Preparation of urea or its derivatives, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups of substituted ureas with formation of the N-C(O)-N moiety
- C07C273/1818—Preparation of urea or its derivatives, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups of substituted ureas with formation of the N-C(O)-N moiety from -N=C=O and XNR'R"
- C07C273/1827—X being H
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
- C07K5/06043—Leu-amino acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- C07K5/06165—Dipeptides with the first amino acid being heterocyclic and Pro-amino acid; Derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
- C07K5/0823—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Pro-amino acid; Derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
- C07K5/101—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms, e.g. Val, Ile, Leu
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US56612983A | 1983-12-27 | 1983-12-27 | |
| US60860984A | 1984-05-09 | 1984-05-09 | |
| US06/673,996 US4657893A (en) | 1984-05-09 | 1984-11-26 | 4H-3,1-benzoxazin-4-ones and related compounds and use as enzyme inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK625184D0 DK625184D0 (da) | 1984-12-21 |
| DK625184A true DK625184A (da) | 1985-06-28 |
Family
ID=27415984
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK625184A DK625184A (da) | 1983-12-27 | 1984-12-21 | Benzoxazinderivater |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP0147211B1 (hu) |
| KR (1) | KR890000992B1 (hu) |
| CA (1) | CA1269800A (hu) |
| DE (1) | DE3483204D1 (hu) |
| DK (1) | DK625184A (hu) |
| ES (2) | ES8607260A1 (hu) |
| FI (1) | FI79842C (hu) |
| HU (1) | HU195648B (hu) |
| IL (1) | IL73943A (hu) |
| NO (1) | NO163184C (hu) |
| NZ (1) | NZ210669A (hu) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1309556C (en) * | 1987-06-09 | 1992-10-27 | Masayuki Kokubo | 4h-3,1-benzoxazin-4-one compounds and pharmaceutical composition thereoffor the inhibition of serine proteases |
| ES2067140T3 (es) * | 1990-09-10 | 1995-03-16 | Asahi Chemical Ind | Compuestos fenilester de acido benzoico y composiciones inhibidoras de la elastasa que contienen los mismos. |
| US5652237A (en) * | 1994-09-09 | 1997-07-29 | Warner-Lambert Company | 2-substituted-4H-3, 1-benzoxazin-4-ones and benzthiazin-4-ones as inhibitors of complement C1r protease for the treatment of inflammatory processes |
| US5985872A (en) * | 1995-05-24 | 1999-11-16 | G.D. Searle & Co. | 2-amino-benzoxazinones for the treatment of viral infections |
| GB9700597D0 (en) * | 1997-01-14 | 1997-03-05 | Sandoz Pharma Uk | Organic compounds |
| US6180625B1 (en) | 1998-03-24 | 2001-01-30 | Novo Nordisk A/S | Heterocyclic compounds regulating clotting |
| AU2826099A (en) * | 1998-03-24 | 1999-10-18 | Novo Nordisk A/S | Heterocyclic compounds regulating clotting |
| WO2000030646A1 (en) * | 1998-11-26 | 2000-06-02 | Novo Nordisk A/S | Heterocyclic compounds regulating clotting |
| GB9900416D0 (en) | 1999-01-08 | 1999-02-24 | Alizyme Therapeutics Ltd | Inhibitors |
| WO2000043371A2 (en) | 1999-01-22 | 2000-07-27 | Elan Pharmaceuticals, Inc. | Fused ring heteroaryl and heterocyclic compounds which inhibit leukocyte adhesion mediated by vla-4 |
| EP1144388B1 (en) | 1999-01-22 | 2010-01-13 | Elan Pharmaceuticals, Inc. | Acyl derivatives which treat vla-4 related disorders |
| US6436904B1 (en) | 1999-01-25 | 2002-08-20 | Elan Pharmaceuticals, Inc. | Compounds which inhibit leukocyte adhesion mediated by VLA-4 |
| TW200307671A (en) | 2002-05-24 | 2003-12-16 | Elan Pharm Inc | Heteroaryl compounds which inhibit leukocyte adhesion mediated by α 4 integrins |
| TWI281470B (en) | 2002-05-24 | 2007-05-21 | Elan Pharm Inc | Heterocyclic compounds which inhibit leukocyte adhesion mediated by alpha4 integrins |
| JP5081828B2 (ja) | 2005-09-29 | 2012-11-28 | エラン ファーマシューティカルズ，インコーポレイテッド | Ｖｌａ−４によって媒介される白血球粘着を阻害するカルバメート化合物 |
| NZ567270A (en) | 2005-09-29 | 2011-06-30 | Elan Pharm Inc | Pyrimidinyl amide compounds which inhibit leukocyte adhesion mediated by VLA-4 |
| KR20080100271A (ko) | 2006-02-27 | 2008-11-14 | 엘란 파마슈티칼스, 인크. | Ｖｌａ-4에 의해 매개되는 백혈구 부착을 억제하는 피리미디닐 술폰아미드 화합물 |
| JP2012525336A (ja) | 2009-04-27 | 2012-10-22 | エラン ファーマシューティカルズ，インコーポレイテッド | α−４インテグリンのピリジノンアンタゴニスト |
| EP3565543A4 (en) * | 2017-01-06 | 2020-10-14 | The Regents of The University of California | MU TYPE OPIOID RECEIVER MODULATORS |
| WO2019195634A1 (en) | 2018-04-04 | 2019-10-10 | Epiodyne, Inc. | Opioid receptor modulators and products and methods related thereto |
| TW202304869A (zh) | 2021-04-05 | 2023-02-01 | 美商艾碧奧戴股份有限公司 | 類鴉片受體調節劑 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3450700A (en) * | 1966-12-20 | 1969-06-17 | Upjohn Co | 2-tertiary amino-4h-3,1-benzoxazin-4-ones |
| DE2315303A1 (de) * | 1973-03-27 | 1974-10-17 | Bayer Ag | Verfahren zur herstellung von n-substituierten 2-amino-3,1-benzoxazin-4-onen |
-
1984
- 1984-12-20 NZ NZ210669A patent/NZ210669A/en unknown
- 1984-12-21 EP EP84309013A patent/EP0147211B1/en not_active Expired - Lifetime
- 1984-12-21 DE DE8484309013T patent/DE3483204D1/de not_active Expired - Fee Related
- 1984-12-21 NO NO845176A patent/NO163184C/no unknown
- 1984-12-21 CA CA000470962A patent/CA1269800A/en not_active Expired - Fee Related
- 1984-12-21 DK DK625184A patent/DK625184A/da not_active Application Discontinuation
- 1984-12-26 IL IL73943A patent/IL73943A/xx unknown
- 1984-12-26 KR KR1019840008352A patent/KR890000992B1/ko not_active IP Right Cessation
- 1984-12-26 ES ES539038A patent/ES8607260A1/es not_active Expired
- 1984-12-27 FI FI845116A patent/FI79842C/fi not_active IP Right Cessation
- 1984-12-27 HU HU844839A patent/HU195648B/hu not_active IP Right Cessation
-
1986
- 1986-01-14 ES ES550879A patent/ES8703437A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ES8607260A1 (es) | 1986-06-01 |
| FI845116L (fi) | 1985-06-28 |
| NO163184C (no) | 1990-04-18 |
| HUT36808A (en) | 1985-10-28 |
| IL73943A0 (en) | 1985-03-31 |
| IL73943A (en) | 1989-01-31 |
| FI845116A0 (fi) | 1984-12-27 |
| ES8703437A1 (es) | 1987-03-01 |
| FI79842B (fi) | 1989-11-30 |
| EP0147211B1 (en) | 1990-09-12 |
| NZ210669A (en) | 1988-05-30 |
| HU195648B (en) | 1988-06-28 |
| ES539038A0 (es) | 1986-06-01 |
| ES550879A0 (es) | 1987-03-01 |
| FI79842C (fi) | 1990-03-12 |
| DE3483204D1 (de) | 1990-10-18 |
| NO845176L (no) | 1985-06-28 |
| DK625184D0 (da) | 1984-12-21 |
| EP0147211A2 (en) | 1985-07-03 |
| EP0147211A3 (en) | 1985-08-14 |
| CA1269800A (en) | 1990-05-29 |
| KR850004472A (ko) | 1985-07-15 |
| KR890000992B1 (ko) | 1989-04-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |