DK570486A - Heterocyclisk substituerede 2(1h)-quinoloner, deres anvendelse til fremstilling af hjertestimulerende laegemidler, farmaceutiske praeparater indeholdende forbindelserne og mellemprodukter ved deres fremstilling - Google Patents

Heterocyclisk substituerede 2(1h)-quinoloner, deres anvendelse til fremstilling af hjertestimulerende laegemidler, farmaceutiske praeparater indeholdende forbindelserne og mellemprodukter ved deres fremstilling

Info

Publication number
DK570486A
DK570486A DK570486A DK570486A DK570486A DK 570486 A DK570486 A DK 570486A DK 570486 A DK570486 A DK 570486A DK 570486 A DK570486 A DK 570486A DK 570486 A DK570486 A DK 570486A
Authority
DK
Denmark
Prior art keywords
quinolons
medicines
intermediates
compounds
preparation
Prior art date
Application number
DK570486A
Other languages
Danish (da)
English (en)
Other versions
DK570486D0 (da
Inventor
Simon Fraser Campbell
David Anthony Roberts
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of DK570486D0 publication Critical patent/DK570486D0/da
Publication of DK570486A publication Critical patent/DK570486A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK570486A 1985-11-28 1986-11-27 Heterocyclisk substituerede 2(1h)-quinoloner, deres anvendelse til fremstilling af hjertestimulerende laegemidler, farmaceutiske praeparater indeholdende forbindelserne og mellemprodukter ved deres fremstilling DK570486A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858529362A GB8529362D0 (en) 1985-11-28 1985-11-28 Quinolone cardiac stimulants

Publications (2)

Publication Number Publication Date
DK570486D0 DK570486D0 (da) 1986-11-27
DK570486A true DK570486A (da) 1987-08-03

Family

ID=10588943

Family Applications (1)

Application Number Title Priority Date Filing Date
DK570486A DK570486A (da) 1985-11-28 1986-11-27 Heterocyclisk substituerede 2(1h)-quinoloner, deres anvendelse til fremstilling af hjertestimulerende laegemidler, farmaceutiske praeparater indeholdende forbindelserne og mellemprodukter ved deres fremstilling

Country Status (20)

Country Link
US (1) US4740513A (de)
EP (1) EP0226357A1 (de)
JP (1) JPS62138490A (de)
KR (1) KR890002795B1 (de)
CN (1) CN1004205B (de)
AU (1) AU569200B2 (de)
DD (2) DD270710A5 (de)
DK (1) DK570486A (de)
FI (1) FI864814A (de)
GB (1) GB8529362D0 (de)
HU (1) HU196989B (de)
IL (1) IL80799A0 (de)
NO (1) NO864782D0 (de)
NZ (1) NZ218428A (de)
PH (1) PH23868A (de)
PL (2) PL151696B1 (de)
PT (1) PT83810B (de)
SU (1) SU1470190A3 (de)
YU (1) YU44603B (de)
ZA (1) ZA868978B (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5358949A (en) * 1986-03-05 1994-10-25 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives and salts thereof and anti-arrhythmic agents containing the carbostyril derivatives
DK111387A (da) * 1986-03-05 1987-09-06 Otsuka Pharma Co Ltd Carbostyrilderivater og salte deraf, laegemiddel indeholdende saadanne derivater samt fremgangsmaade til fremstilling af derivaterne
GB8630702D0 (en) * 1986-12-23 1987-02-04 Wellcome Found Quinoline compound
US5166160A (en) * 1986-12-23 1992-11-24 Burroughs Wellcome Co. Quinoline compound
GB8709448D0 (en) * 1987-04-21 1987-05-28 Pfizer Ltd Heterobicyclic quinoline derivatives
US5064837A (en) * 1989-11-13 1991-11-12 Schering Corporation 3-substituted-1-aryl-2(h)-quinolones and their pharmaceutical compositions
DE19636994A1 (de) * 1996-09-12 1998-03-19 Basf Ag Verfahren zur Herstellung von (2'-Fluorphenyl)-3-halogenpyridinen
IL134662A0 (en) * 1997-09-24 2001-04-30 Orion Corp Bisethers of 1-oxa, aza and thianaphthalen-2- ones as phospholamban inhibitors
US6388080B1 (en) 2001-06-29 2002-05-14 Grayson Walker Stowell Polymorphic forms of 6-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
US6657061B2 (en) 2001-06-29 2003-12-02 Grayson Walker Stowell Polymorphic forms of 6-[4-1(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
US6531603B1 (en) 2001-06-29 2003-03-11 Grayson Walker Stowell Polymorphic forms of 6-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
US6660864B2 (en) 2001-06-29 2003-12-09 Grayson Walker Stowell Polymorphic forms of 6-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
US6573382B2 (en) 2001-06-29 2003-06-03 Grayson Walker Stowell Polymorphic forms of 6-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
US6596871B2 (en) 2001-06-29 2003-07-22 Grayson Walker Stowell Polymorphic forms of 6-[4-(1-cyclohexyl-1h-tetraol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
US8937184B2 (en) * 2005-02-16 2015-01-20 Abbvie B.V. 1H-imidazole derivatives as cannabinoid CB2 receptor modulators

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3993656A (en) * 1974-11-19 1976-11-23 Merck & Co., Inc. 1,8-Naphthyridine compounds
JPS5473783A (en) * 1977-11-15 1979-06-13 Otsuka Pharmaceut Co Ltd Pyridine derivative
DE2815956A1 (de) * 1978-04-13 1979-10-18 Bayer Ag Verfahren zur herstellung von in 2-stellung substituierten triazolen-1,2,3
JPS5535019A (en) * 1978-09-01 1980-03-11 Otsuka Pharmaceut Co Ltd Carbostyryl derivative
US4258185A (en) * 1978-10-17 1981-03-24 Yoshitomi Pharmaceutical Industries, Ltd. Pyridazinone compounds
JPS5576872A (en) * 1978-12-06 1980-06-10 Yoshitomi Pharmaceut Ind Ltd Imidazolidinone derivative
JPS5777676A (en) * 1980-10-31 1982-05-15 Otsuka Pharmaceut Co Ltd Carbostyril derivative
CA1164459A (en) * 1980-11-11 1984-03-27 Yung-Hsiung Yang Process for preparing (imidazo¬1,2-a|pyridine- 2-yl)-carbostyril or -3,4-dihydrocarbostyryl derivatives
EP0102046A1 (de) * 1982-08-26 1984-03-07 Schering Corporation Tricyclische Lactame, Verfahren zur Herstellung und diese enthaltende pharmazeutische Zubereitungen
CH655110A5 (de) * 1982-09-03 1986-03-27 Otsuka Pharma Co Ltd Carbostyrilderivate, verfahren zu deren herstellung und arzneimittel, welche diese enthalten.
PT79031B (en) * 1983-08-20 1986-08-22 Boots Co Plc Therapeutic agents
US4532250A (en) * 1983-11-23 1985-07-30 American Hospital Supply Corporation 5-Heteroarylimidazol-2-ones having cardiotonic activity
PT79699B (en) * 1983-12-22 1986-12-10 Pfizer Process for preparing quinolone inotropic agents
US4591591A (en) * 1984-03-08 1986-05-27 Eli Lilly And Company Pyridazinone derivatives as inotropic agents
US4721721A (en) * 1984-12-18 1988-01-26 Rorer Pharmaceutical Corporation 6-(4-thiazole) compounds, cardiotonic compositions including the same, and their uses

Also Published As

Publication number Publication date
YU44603B (en) 1990-10-31
FI864814A (fi) 1987-05-29
CN86108133A (zh) 1987-09-09
NO864782D0 (no) 1986-11-27
HU196989B (en) 1989-02-28
DD265403A5 (de) 1989-03-01
SU1470190A3 (ru) 1989-03-30
DK570486D0 (da) 1986-11-27
KR870004975A (ko) 1987-06-02
CN1004205B (zh) 1989-05-17
PL270983A1 (en) 1988-09-15
FI864814A0 (fi) 1986-11-26
GB8529362D0 (en) 1986-01-02
US4740513A (en) 1988-04-26
PT83810B (en) 1988-12-09
EP0226357A1 (de) 1987-06-24
IL80799A0 (en) 1987-02-27
YU202686A (en) 1987-12-31
KR890002795B1 (ko) 1989-07-31
PL262599A1 (en) 1988-07-07
PT83810A (en) 1986-12-01
NZ218428A (en) 1989-03-29
ZA868978B (en) 1988-07-27
DD270710A5 (de) 1989-08-09
AU569200B2 (en) 1988-01-21
PL151696B1 (en) 1990-09-28
PH23868A (en) 1989-11-23
HUT42082A (en) 1987-06-29
JPS62138490A (ja) 1987-06-22
AU6575486A (en) 1987-06-11

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