DK3030549T3 - Pyridazinonforbindelser og anvendelser deraf - Google Patents

Pyridazinonforbindelser og anvendelser deraf Download PDF

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DK3030549T3
DK3030549T3 DK14843298.2T DK14843298T DK3030549T3 DK 3030549 T3 DK3030549 T3 DK 3030549T3 DK 14843298 T DK14843298 T DK 14843298T DK 3030549 T3 DK3030549 T3 DK 3030549T3
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pyridazinon
compounds
pyridazinon compounds
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DK14843298.2T
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Danish (da)
English (en)
Inventor
Leonid Beigelman
Robert Than Hendricks
Antitsa Dimitrova Stoycheva
Jerome Deval
Sarah Katherine Stevens
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Janssen Biopharma Inc
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • A61K31/24—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group having an amino or nitro group
    • A61K31/245—Amino benzoic acid types, e.g. procaine, novocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
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    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/504—Pyridazines; Hydrogenated pyridazines forming part of bridged ring systems
    • A—HUMAN NECESSITIES
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/529—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim forming part of bridged ring systems
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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PH12016500492A1 (en) 2016-05-16
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AU2014318837A1 (en) 2016-03-24
EP3030549A1 (en) 2016-06-15
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MX370085B (es) 2019-11-29
HRP20190822T1 (hr) 2019-08-23
KR102286860B1 (ko) 2021-08-05
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KR20160052683A (ko) 2016-05-12
LT3030549T (lt) 2019-06-25
IL244434A0 (en) 2016-04-21
EP3030549A4 (en) 2017-03-15
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CA2922943A1 (en) 2015-03-19
JP2016530315A (ja) 2016-09-29
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CN105722831A (zh) 2016-06-29
US10364226B2 (en) 2019-07-30
PH12016500492B1 (en) 2016-05-16
EA034868B1 (ru) 2020-03-31
US20160221963A1 (en) 2016-08-04
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EP3030549B1 (en) 2019-02-20
IL244434B (en) 2020-09-30
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SI3030549T1 (sl) 2019-08-30
AU2014318837B2 (en) 2019-05-30

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