DK172766B1 - Derivater af det neutrale macrolid betegnet CP-63693 og farmaceutiske præparater indeholdende disse - Google Patents

Derivater af det neutrale macrolid betegnet CP-63693 og farmaceutiske præparater indeholdende disse Download PDF

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Publication number
DK172766B1
DK172766B1 DK198600288A DK28886A DK172766B1 DK 172766 B1 DK172766 B1 DK 172766B1 DK 198600288 A DK198600288 A DK 198600288A DK 28886 A DK28886 A DK 28886A DK 172766 B1 DK172766 B1 DK 172766B1
Authority
DK
Denmark
Prior art keywords
compounds
ethyl acetate
dimethylamino
reaction
mmol
Prior art date
Application number
DK198600288A
Other languages
Danish (da)
English (en)
Other versions
DK28886D0 (da
DK28886A (da
Inventor
Arthur Adam Nagel
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK28886D0 publication Critical patent/DK28886D0/da
Publication of DK28886A publication Critical patent/DK28886A/da
Application granted granted Critical
Publication of DK172766B1 publication Critical patent/DK172766B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK198600288A 1985-01-22 1986-01-21 Derivater af det neutrale macrolid betegnet CP-63693 og farmaceutiske præparater indeholdende disse DK172766B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69370285 1985-01-22
US06/693,702 US4585759A (en) 1985-01-22 1985-01-22 Antibacterial derivatives of a neutral macrolide

Publications (3)

Publication Number Publication Date
DK28886D0 DK28886D0 (da) 1986-01-21
DK28886A DK28886A (da) 1986-07-23
DK172766B1 true DK172766B1 (da) 1999-07-05

Family

ID=24785743

Family Applications (1)

Application Number Title Priority Date Filing Date
DK198600288A DK172766B1 (da) 1985-01-22 1986-01-21 Derivater af det neutrale macrolid betegnet CP-63693 og farmaceutiske præparater indeholdende disse

Country Status (8)

Country Link
US (1) US4585759A (de)
EP (1) EP0189281B1 (de)
JP (1) JPS61172893A (de)
AT (1) ATE36338T1 (de)
DE (1) DE3660493D1 (de)
DK (1) DK172766B1 (de)
GR (1) GR860148B (de)
IE (1) IE58451B1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AP9801420A0 (en) * 1998-01-02 1998-12-31 Pfizer Prod Inc Novel macrolides.
AP1060A (en) * 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
AU2003211113B2 (en) 2002-02-15 2007-08-09 Merckle Gmbh Antibiotic conjugates
AU2003215245A1 (en) 2002-02-15 2003-09-09 Sympore Gmbh Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
EP1483277A4 (de) 2002-02-15 2007-10-03 Merckle Gmbh Konjugate biologisch aktiver verbindungen, verfahren zu deren herstellung und anwendung, formulierung und pharmazeutische anwendungen davon
WO2011080739A2 (en) * 2009-12-29 2011-07-07 Yeda Research And Development Co. Ltd. Synergistic antibiotic combinations and derivatives
FR2995605B1 (fr) * 2012-09-18 2014-09-19 Sanofi Sa Derives de macrolides, leur preparation et leur application therapeutique.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3883507A (en) * 1971-01-25 1975-05-13 Schering Corp Novel esters of megalomicin A and processes for their preparation
FR2126108B1 (de) * 1971-02-25 1974-08-02 Rhone Poulenc Sa
JPS55151598A (en) * 1979-05-11 1980-11-26 Taisho Pharmaceut Co Ltd Erythromycin a derivative and its preparation

Also Published As

Publication number Publication date
GR860148B (en) 1986-05-21
JPS61172893A (ja) 1986-08-04
DE3660493D1 (en) 1988-09-15
ATE36338T1 (de) 1988-08-15
DK28886D0 (da) 1986-01-21
IE58451B1 (en) 1993-09-22
EP0189281B1 (de) 1988-08-10
IE860165L (en) 1986-07-22
DK28886A (da) 1986-07-23
EP0189281A2 (de) 1986-07-30
EP0189281A3 (en) 1986-10-22
US4585759A (en) 1986-04-29

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B1 Patent granted (law 1993)
PBP Patent lapsed

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