DK171132B1 - Monocycliske beta-lactam-forbindelser og fremgangsmåde til fremstilling deraf - Google Patents

Monocycliske beta-lactam-forbindelser og fremgangsmåde til fremstilling deraf Download PDF

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Publication number
DK171132B1
DK171132B1 DK114384A DK114384A DK171132B1 DK 171132 B1 DK171132 B1 DK 171132B1 DK 114384 A DK114384 A DK 114384A DK 114384 A DK114384 A DK 114384A DK 171132 B1 DK171132 B1 DK 171132B1
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DK
Denmark
Prior art keywords
group
amino
alkyl
formula
hydroxy
Prior art date
Application number
DK114384A
Other languages
Danish (da)
English (en)
Other versions
DK114384A (da
DK114384D0 (da
Inventor
Marvin Joseph Miller
Original Assignee
Univ Notre Dame Du Lac
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Notre Dame Du Lac filed Critical Univ Notre Dame Du Lac
Publication of DK114384D0 publication Critical patent/DK114384D0/da
Publication of DK114384A publication Critical patent/DK114384A/da
Application granted granted Critical
Publication of DK171132B1 publication Critical patent/DK171132B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK114384A 1983-03-28 1984-02-28 Monocycliske beta-lactam-forbindelser og fremgangsmåde til fremstilling deraf DK171132B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US47937583 1983-03-28
US06/479,375 US4565654A (en) 1983-03-28 1983-03-28 N-Acyloxy monocyclic β-lactams

Publications (3)

Publication Number Publication Date
DK114384D0 DK114384D0 (da) 1984-02-28
DK114384A DK114384A (da) 1984-09-29
DK171132B1 true DK171132B1 (da) 1996-06-24

Family

ID=23903742

Family Applications (2)

Application Number Title Priority Date Filing Date
DK114384A DK171132B1 (da) 1983-03-28 1984-02-28 Monocycliske beta-lactam-forbindelser og fremgangsmåde til fremstilling deraf
DK113695A DK171676B1 (da) 1983-03-28 1995-10-10 Fremgangsmåde til fremstilling af N-hydroxy-2-azetidinoner eller syreadditionssalte deraf

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK113695A DK171676B1 (da) 1983-03-28 1995-10-10 Fremgangsmåde til fremstilling af N-hydroxy-2-azetidinoner eller syreadditionssalte deraf

Country Status (12)

Country Link
US (1) US4565654A (el)
EP (1) EP0123442B1 (el)
JP (1) JPH0745464B2 (el)
KR (1) KR910004090B1 (el)
CA (1) CA1331755C (el)
DE (1) DE3472102D1 (el)
DK (2) DK171132B1 (el)
GB (1) GB2137203B (el)
GR (1) GR81468B (el)
HU (1) HU197303B (el)
IE (1) IE57040B1 (el)
IL (1) IL71300A (el)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4638061A (en) * 1985-01-28 1987-01-20 E. R. Squibb & Sons, Inc. [3S(Z)]-2-[[[1-(2-amino-4-thiazolyl)-2-[[2,2-dimethyl-4-oxo-1-(sulfooxy)-3-azetidinyl]amino]-2-oxoethylidene]-amino]oxy] acetic acid and intermediate
US4772694A (en) * 1986-07-24 1988-09-20 Eli Lilly And Company Chiral 3-(1,2,5-trisubstituted imidazolidinone) azetidinone antibiotic intermediates
US4751296A (en) * 1986-08-06 1988-06-14 University Of Notre Dame Du Lac Process for 4-halomethyl-azetidinones by cyclization of O-acylhydroxamates
JP2591233Y2 (ja) * 1991-06-25 1999-03-03 東プレ株式会社 バン型車における荷物扉の煽止装置
US5631365A (en) 1993-09-21 1997-05-20 Schering Corporation Hydroxy-substituted azetidinone compounds useful as hypocholesterolemic agents
US5925659A (en) * 1996-05-07 1999-07-20 Merck & Co., Inc. Antibacterial agents
US11400079B2 (en) 2017-10-05 2022-08-02 University Of Notre Dame Du Lac Antibacterial monobactams

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US337197A (en) * 1886-03-02 Ments
US4337197A (en) * 1980-10-31 1982-06-29 E. R. Squibb & Sons, Inc. O-sulfated β-lactam hydroxamic acids and intermediates
US4386034A (en) * 1981-02-02 1983-05-31 E. R. Squibb & Sons, Inc. Sulfamated amino acid amides
JPS58113174A (ja) * 1981-12-26 1983-07-05 Toyama Chem Co Ltd 新規なアゼチジン誘導体またはその塩類を含有する抗菌剤
EP0117053A1 (en) * 1983-02-10 1984-08-29 Ajinomoto Co., Inc. Azetidinone derivatives

Also Published As

Publication number Publication date
IL71300A0 (en) 1984-06-29
GR81468B (el) 1984-12-11
GB2137203A (en) 1984-10-03
IE57040B1 (en) 1992-03-25
GB8407768D0 (en) 1984-05-02
IL71300A (en) 1990-01-18
DK113695A (da) 1995-10-10
DK171676B1 (da) 1997-03-10
US4565654A (en) 1986-01-21
GB2137203B (en) 1987-01-14
KR910004090B1 (ko) 1991-06-22
JPS6045560A (ja) 1985-03-12
KR840008145A (ko) 1984-12-13
DE3472102D1 (en) 1988-07-21
DK114384A (da) 1984-09-29
EP0123442B1 (en) 1988-06-15
IE840742L (en) 1984-09-28
EP0123442A1 (en) 1984-10-31
CA1331755C (en) 1994-08-30
DK114384D0 (da) 1984-02-28
JPH0745464B2 (ja) 1995-05-17
HU197303B (en) 1989-03-28

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed