DK170021B1 - Fremgangsmåde og mellemprodukter til fremstilling af cis,endo-2-azabicycloalkan-3-carboxylsyrederivater - Google Patents

Fremgangsmåde og mellemprodukter til fremstilling af cis,endo-2-azabicycloalkan-3-carboxylsyrederivater Download PDF

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Publication number
DK170021B1
DK170021B1 DK389585A DK389585A DK170021B1 DK 170021 B1 DK170021 B1 DK 170021B1 DK 389585 A DK389585 A DK 389585A DK 389585 A DK389585 A DK 389585A DK 170021 B1 DK170021 B1 DK 170021B1
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DK
Denmark
Prior art keywords
formula
cis
alkoxy
carboxylic acid
endo
Prior art date
Application number
DK389585A
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Danish (da)
English (en)
Other versions
DK389585A (da
DK389585D0 (da
Inventor
Hansjoerg Urbach
Rainer Henning
Winfried Hertzsch
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Hoechst Ag
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Filing date
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Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of DK389585D0 publication Critical patent/DK389585D0/da
Publication of DK389585A publication Critical patent/DK389585A/da
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Publication of DK170021B1 publication Critical patent/DK170021B1/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/42—Nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK389585A 1984-08-28 1985-08-27 Fremgangsmåde og mellemprodukter til fremstilling af cis,endo-2-azabicycloalkan-3-carboxylsyrederivater DK170021B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3431541A DE3431541A1 (de) 1984-08-28 1984-08-28 Cis,endo-2-azabicycloalkan-3-carbonsaeure-derivate, verfahren zu deren herstellung, deren verwendung sowie zwischenprodukte bei deren herstellung
DE3431541 1984-08-28

Publications (3)

Publication Number Publication Date
DK389585D0 DK389585D0 (da) 1985-08-27
DK389585A DK389585A (da) 1986-03-01
DK170021B1 true DK170021B1 (da) 1995-05-01

Family

ID=6244049

Family Applications (1)

Application Number Title Priority Date Filing Date
DK389585A DK170021B1 (da) 1984-08-28 1985-08-27 Fremgangsmåde og mellemprodukter til fremstilling af cis,endo-2-azabicycloalkan-3-carboxylsyrederivater

Country Status (10)

Country Link
US (2) US4886827A (ja)
EP (1) EP0173199B1 (ja)
JP (2) JPS6160650A (ja)
AT (1) ATE108436T1 (ja)
DE (2) DE3431541A1 (ja)
DK (1) DK170021B1 (ja)
ES (2) ES8607928A1 (ja)
GR (1) GR852048B (ja)
IE (1) IE63525B1 (ja)
PT (1) PT81036B (ja)

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KR101381768B1 (ko) 2006-01-06 2014-04-07 선오비온 파마슈티컬스 인코포레이티드 테트랄론-기재 모노아민 재흡수 저해제
ES2643602T3 (es) 2006-03-31 2017-11-23 Sunovion Pharmaceuticals Inc. Aminas y quirales
US7579370B2 (en) * 2006-06-30 2009-08-25 Sepracor Inc. Fused heterocycles
US7884124B2 (en) 2006-06-30 2011-02-08 Sepracor Inc. Fluoro-substituted inhibitors of D-amino acid oxidase
US20080082066A1 (en) * 2006-10-02 2008-04-03 Weyerhaeuser Co. Crosslinked carboxyalkyl cellulose fibers having non-permanent and temporary crosslinks
US7902252B2 (en) 2007-01-18 2011-03-08 Sepracor, Inc. Inhibitors of D-amino acid oxidase
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CN103936605B (zh) 2007-05-31 2017-09-01 赛诺维信制药公司 苯基取代的环烷胺作为一元胺再摄取抑制剂
WO2010017418A1 (en) * 2008-08-07 2010-02-11 Sepracor Inc. Prodrugs of fused heterocyclic inhibitors of d-amino acid oxidase
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CN111333656B (zh) * 2016-12-15 2023-03-14 豪夫迈·罗氏有限公司 制备btk抑制剂的方法

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DE3322530A1 (de) * 1983-06-23 1985-01-10 Hoechst Ag, 6230 Frankfurt Verfahren zur herstellung von mono-, bi- und tricyclischen aminosaeuren
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DE3639879A1 (de) * 1986-11-21 1988-06-01 Hoechst Ag Verfahren zur herstellung von mono-, bi- und tricyclischen aminosaeuren, zwischenprodukte dieses verfahrens sowie ein verfahren zu deren herstellung
DE3641451A1 (de) * 1986-12-04 1988-06-16 Hoechst Ag Derivate bicyclischer aminocarbonsaeuren, verfahren und zwischenprodukte zu deren herstellung sowie deren verwendung
DE3839127A1 (de) * 1988-11-19 1990-05-23 Hoechst Ag Pyrrolidon-2-carbonsaeure-derivate mit psychotroper wirkung
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Also Published As

Publication number Publication date
GR852048B (ja) 1985-12-18
ES546402A0 (es) 1986-06-01
DK389585A (da) 1986-03-01
IE852108L (en) 1986-02-28
PT81036A (de) 1985-09-01
JPS6160650A (ja) 1986-03-28
JPH06228094A (ja) 1994-08-16
EP0173199A1 (de) 1986-03-05
IE63525B1 (en) 1995-05-03
DE3431541A1 (de) 1986-03-06
ES8707929A1 (es) 1987-09-01
PT81036B (pt) 1987-11-11
ES552317A0 (es) 1987-09-01
US5550255A (en) 1996-08-27
DK389585D0 (da) 1985-08-27
DE3587879D1 (de) 1994-08-18
ATE108436T1 (de) 1994-07-15
EP0173199B1 (de) 1994-07-13
ES8607928A1 (es) 1986-06-01
US4886827A (en) 1989-12-12

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B1 Patent granted (law 1993)
PUP Patent expired