DK169676B1 - 4,5,6,7-Tetrahydroisothiazolo[4,5-c]pyridinderivater og farmaceutiske kompositioner deraf - Google Patents

4,5,6,7-Tetrahydroisothiazolo[4,5-c]pyridinderivater og farmaceutiske kompositioner deraf Download PDF

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Publication number
DK169676B1
DK169676B1 DK121789A DK121789A DK169676B1 DK 169676 B1 DK169676 B1 DK 169676B1 DK 121789 A DK121789 A DK 121789A DK 121789 A DK121789 A DK 121789A DK 169676 B1 DK169676 B1 DK 169676B1
Authority
DK
Denmark
Prior art keywords
tetrahydroisothiazolo
pyridine
methyl
propynyloxy
formula
Prior art date
Application number
DK121789A
Other languages
Danish (da)
English (en)
Other versions
DK121789D0 (da
DK121789A (da
Inventor
Povl Krogsgaard-Larsen
Erik Falch
Henrik Pedersen
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB888806013A external-priority patent/GB8806013D0/en
Priority claimed from GB888822564A external-priority patent/GB8822564D0/en
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of DK121789D0 publication Critical patent/DK121789D0/da
Publication of DK121789A publication Critical patent/DK121789A/da
Application granted granted Critical
Publication of DK169676B1 publication Critical patent/DK169676B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK121789A 1988-03-14 1989-03-14 4,5,6,7-Tetrahydroisothiazolo[4,5-c]pyridinderivater og farmaceutiske kompositioner deraf DK169676B1 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8806013 1988-03-14
GB888806013A GB8806013D0 (en) 1988-03-14 1988-03-14 Heterocyclic compounds
GB888822564A GB8822564D0 (en) 1988-09-26 1988-09-26 Heterocyclic compounds
GB8822564 1988-09-26

Publications (3)

Publication Number Publication Date
DK121789D0 DK121789D0 (da) 1989-03-14
DK121789A DK121789A (da) 1989-09-15
DK169676B1 true DK169676B1 (da) 1995-01-09

Family

ID=26293631

Family Applications (1)

Application Number Title Priority Date Filing Date
DK121789A DK169676B1 (da) 1988-03-14 1989-03-14 4,5,6,7-Tetrahydroisothiazolo[4,5-c]pyridinderivater og farmaceutiske kompositioner deraf

Country Status (17)

Country Link
US (1) US4923880A (cs)
EP (1) EP0336555B1 (cs)
JP (1) JPH01275585A (cs)
AT (1) ATE81130T1 (cs)
AU (1) AU630085B2 (cs)
CA (1) CA1337201C (cs)
DE (1) DE68903019T2 (cs)
DK (1) DK169676B1 (cs)
ES (1) ES2052901T3 (cs)
FI (1) FI91411C (cs)
GR (1) GR3006606T3 (cs)
IE (1) IE62782B1 (cs)
IL (1) IL89351A0 (cs)
NO (1) NO177145C (cs)
NZ (1) NZ228182A (cs)
PT (1) PT89992B (cs)
ZA (1) ZA891769B (cs)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2645862B1 (fr) * 1989-04-18 1991-07-12 Esteve Labor Dr Derives d'isothiazolo-pyrydone azetidinyl substitues, leur preparation et leur application en tant que medicaments
US5574028A (en) * 1994-10-31 1996-11-12 Eli Lilly And Company Method for treating anxiety
CZ174698A3 (cs) * 1995-12-07 1998-10-14 Eli Lilly And Company Léčivo pro léčbu bolesti
US20050137222A1 (en) * 2003-12-18 2005-06-23 H. Lundbeck A/S Treatment of insomnia in human patients
US20110098777A1 (en) * 2009-10-23 2011-04-28 Silverstone Leon M Method and apparatus for treatment of neurodegenerative diseases including depression, mild cognitive impairment, and dementia
CN107428776B (zh) 2015-03-24 2020-10-23 H.隆德贝克有限公司 制造4,5,6,7-四氢异噁唑并[5,4-c]吡啶-3-醇
AU2024257614A1 (en) * 2023-04-18 2025-10-02 Vanderbilt University Pyrrolopyridine derivatives as positive allosteric modulators of the muscarinic acetylcholine receptor m4
CN121002030A (zh) 2023-04-18 2025-11-21 范德比尔特大学 作为毒蕈碱型乙酰胆碱受体m4的正向别构调节剂的噻唑并吡啶衍生物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8314391D0 (en) * 1983-05-24 1983-06-29 Kefalas As Heterocyclic compounds
IL87709A (en) * 1987-09-16 1992-11-15 Pfizer Process for preparing haloalkyl thiazoles and some such novel haloalkyl thiazoles
DE3820775A1 (de) * 1988-06-20 1989-12-21 Thomae Gmbh Dr K Neue 4,5,7,8-tetrahydro-6h-thiazolo(5,4,-d)azepine, ihre herstellung und ihre verwendung als arzneimittel
JP3054738B2 (ja) * 1988-07-22 2000-06-19 武田薬品工業株式会社 チアゾロ［５，４―ｂ］アゼピン誘導体

Also Published As

Publication number Publication date
IL89351A0 (en) 1989-09-10
NO177145C (no) 1995-07-26
AU3126289A (en) 1989-09-14
EP0336555A1 (en) 1989-10-11
IE62782B1 (en) 1995-02-22
DK121789D0 (da) 1989-03-14
DE68903019T2 (de) 1993-07-08
PT89992B (pt) 1994-05-31
FI91411B (fi) 1994-03-15
IE890648L (en) 1989-09-14
ATE81130T1 (de) 1992-10-15
FI91411C (fi) 1994-06-27
ZA891769B (en) 1989-12-27
JPH01275585A (ja) 1989-11-06
DK121789A (da) 1989-09-15
US4923880A (en) 1990-05-08
DE68903019D1 (de) 1992-11-05
NO891071D0 (no) 1989-03-13
ES2052901T3 (es) 1994-07-16
GR3006606T3 (cs) 1993-06-30
AU630085B2 (en) 1992-10-22
CA1337201C (en) 1995-10-03
FI891155A7 (fi) 1989-09-15
NO177145B (no) 1995-04-18
NZ228182A (en) 1990-08-28
FI891155A0 (fi) 1989-03-10
PT89992A (pt) 1989-11-10
EP0336555B1 (en) 1992-09-30
NO891071L (no) 1989-09-15

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