DK168159B1 - Fremgangsmåde til fremstilling af med avermectiner og milbemyciner beslægtede forbindelser - Google Patents

Fremgangsmåde til fremstilling af med avermectiner og milbemyciner beslægtede forbindelser Download PDF

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Publication number
DK168159B1
DK168159B1 DK330189A DK330189A DK168159B1 DK 168159 B1 DK168159 B1 DK 168159B1 DK 330189 A DK330189 A DK 330189A DK 330189 A DK330189 A DK 330189A DK 168159 B1 DK168159 B1 DK 168159B1
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DK
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Prior art keywords
formula
compound
prepared
absent
optional bond
Prior art date
Application number
DK330189A
Other languages
Danish (da)
English (en)
Other versions
DK330189D0 (da
DK330189A (da
Inventor
Christopher James Dutton
Stephen Paul Gibson
Nigel Derek Arthur Walshe
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK330189D0 publication Critical patent/DK330189D0/da
Publication of DK330189A publication Critical patent/DK330189A/da
Application granted granted Critical
Publication of DK168159B1 publication Critical patent/DK168159B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23K—FODDER
    • A23K20/00—Accessory food factors for animal feeding-stuffs
    • A23K20/10—Organic substances
    • A23K20/195—Antibiotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/822—Microorganisms using bacteria or actinomycetales
    • Y10S435/886—Streptomyces

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  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Polymers & Plastics (AREA)
  • Zoology (AREA)
  • Genetics & Genomics (AREA)
  • Agronomy & Crop Science (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Animal Husbandry (AREA)
  • Dentistry (AREA)
  • Veterinary Medicine (AREA)
  • Plant Pathology (AREA)
  • Food Science & Technology (AREA)
  • Biochemistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK330189A 1988-07-05 1989-07-04 Fremgangsmåde til fremstilling af med avermectiner og milbemyciner beslægtede forbindelser DK168159B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8815967 1988-07-05
GB888815967A GB8815967D0 (en) 1988-07-05 1988-07-05 Antiparasitic agents

Publications (3)

Publication Number Publication Date
DK330189D0 DK330189D0 (da) 1989-07-04
DK330189A DK330189A (da) 1990-01-08
DK168159B1 true DK168159B1 (da) 1994-02-21

Family

ID=10639888

Family Applications (1)

Application Number Title Priority Date Filing Date
DK330189A DK168159B1 (da) 1988-07-05 1989-07-04 Fremgangsmåde til fremstilling af med avermectiner og milbemyciner beslægtede forbindelser

Country Status (14)

Country Link
US (3) US4980370A (ja)
EP (1) EP0350187B1 (ja)
JP (1) JPH0694466B2 (ja)
AR (1) AR245131A1 (ja)
AT (1) ATE99694T1 (ja)
AU (1) AU603956B2 (ja)
CA (1) CA1339309C (ja)
DE (1) DE68912007T2 (ja)
DK (1) DK168159B1 (ja)
ES (1) ES2061997T3 (ja)
GB (1) GB8815967D0 (ja)
IE (1) IE63621B1 (ja)
NZ (1) NZ229807A (ja)
PT (1) PT91048B (ja)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES8800986A1 (es) * 1985-07-27 1987-12-01 Pfizer Un procedimiento para la produccion de un nuevo derivado de avermectina
US5840704A (en) * 1986-07-16 1998-11-24 Pfizer Inc. Antiparasitic agents and process for their preparation
US5057499A (en) * 1989-06-02 1991-10-15 Merck & Co. Inc. Avermectin derivatives
US5830875A (en) * 1989-10-30 1998-11-03 Merck & Co., Inc. 24-and 25-substituted avermectin and milbemycin derivatives
GB9205007D0 (en) * 1992-03-07 1992-04-22 Pfizer Ltd Antiparasitic agents
GB9316129D0 (en) * 1993-08-04 1993-09-22 Pfizer Ltd Antiprasatic agents
CA2173494C (en) * 1993-10-05 1999-04-13 Thomas C. Crawford Process and antiparasitic intermediates for doramectin
DE4427766A1 (de) * 1994-08-05 1996-02-08 Basf Ag Verfahren zur Herstellung flüssigkristalliner Mischungen
AP1060A (en) 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
GB9825402D0 (en) 1998-11-19 1999-01-13 Pfizer Ltd Antiparasitic formulations
US8636081B2 (en) 2011-12-15 2014-01-28 Milwaukee Electric Tool Corporation Rotary hammer

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4914624A (ja) * 1972-06-08 1974-02-08
SE434277B (sv) * 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
PH15982A (en) * 1977-10-03 1983-05-18 Merck & Co Inc Selective hydrogenation producta of c-076 compounds and derivatives thereof
IL56149A (en) * 1977-12-19 1989-09-28 Merck & Co Inc 13-halo and 13-deoxy derivatives of c-076 compounds,their preparation and method for the treatment of parasitic infections in animals therewith
US4328335A (en) * 1979-08-13 1982-05-04 Merck & Co., Inc. Process for the interconversion of C-076 compounds
US4423209A (en) * 1982-02-26 1983-12-27 Merck & Co., Inc. Processes for the interconversion of avermectin compounds
DK165119C (da) * 1984-06-05 1993-03-01 American Cyanamid Co Antibiotiske forbindelser betegnet ll-f28249alfa, beta, gamma, delta, epsilon, zeta, eta, theta, iota, kappa, my og ny og pharmaceutisk or pharmakologisk acceptable salte deraf samt fremgangsmaade til deres fremstilling
ES8800986A1 (es) * 1985-07-27 1987-12-01 Pfizer Un procedimiento para la produccion de un nuevo derivado de avermectina
GB8606120D0 (en) * 1986-03-12 1986-04-16 Glaxo Group Ltd Process
IN167980B (ja) * 1987-01-23 1991-01-19 Pfizer
GB8726730D0 (en) * 1987-11-14 1987-12-16 Pfizer Ltd Antiparasitic agents
EP0353959A2 (en) * 1988-08-02 1990-02-07 Beecham Group Plc Antihelmintic macrolide antibiotics

Also Published As

Publication number Publication date
US5057498A (en) 1991-10-15
US5112746A (en) 1992-05-12
EP0350187A3 (en) 1991-03-27
DE68912007D1 (de) 1994-02-17
DK330189D0 (da) 1989-07-04
DE68912007T2 (de) 1994-04-28
GB8815967D0 (en) 1988-08-10
NZ229807A (en) 1990-12-21
EP0350187B1 (en) 1994-01-05
IE892158L (en) 1990-01-05
US4980370A (en) 1990-12-25
IE63621B1 (en) 1995-05-17
AU603956B2 (en) 1990-11-29
DK330189A (da) 1990-01-08
ATE99694T1 (de) 1994-01-15
AR245131A1 (es) 1993-12-30
JPH0694466B2 (ja) 1994-11-24
ES2061997T3 (es) 1994-12-16
EP0350187A2 (en) 1990-01-10
PT91048B (pt) 1995-01-31
AU3784089A (en) 1990-05-03
PT91048A (pt) 1990-02-08
CA1339309C (en) 1997-08-19
JPH02288882A (ja) 1990-11-28

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed