DK1605932T3 - Intranasal formulering af rotigotin - Google Patents

Intranasal formulering af rotigotin

Info

Publication number
DK1605932T3
DK1605932T3 DK04804221T DK04804221T DK1605932T3 DK 1605932 T3 DK1605932 T3 DK 1605932T3 DK 04804221 T DK04804221 T DK 04804221T DK 04804221 T DK04804221 T DK 04804221T DK 1605932 T3 DK1605932 T3 DK 1605932T3
Authority
DK
Denmark
Prior art keywords
rotigotine
intranasal formulation
cyclodextrin
alpha
viscosity
Prior art date
Application number
DK04804221T
Other languages
Danish (da)
English (en)
Inventor
Robert Kraemer
Original Assignee
Sanol Arznei Schwarz Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanol Arznei Schwarz Gmbh filed Critical Sanol Arznei Schwarz Gmbh
Application granted granted Critical
Publication of DK1605932T3 publication Critical patent/DK1605932T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK04804221T 2003-12-23 2004-12-22 Intranasal formulering af rotigotin DK1605932T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP03029680A EP1547592A1 (de) 2003-12-23 2003-12-23 Intranasale formulierung enthaltend

Publications (1)

Publication Number Publication Date
DK1605932T3 true DK1605932T3 (da) 2006-09-18

Family

ID=34530709

Family Applications (1)

Application Number Title Priority Date Filing Date
DK04804221T DK1605932T3 (da) 2003-12-23 2004-12-22 Intranasal formulering af rotigotin

Country Status (28)

Country Link
US (1) US7683040B2 (de)
EP (2) EP1547592A1 (de)
JP (1) JP4430067B2 (de)
KR (1) KR100718760B1 (de)
CN (1) CN100374112C (de)
AT (1) ATE326961T1 (de)
AU (1) AU2004308641B2 (de)
BR (1) BRPI0407845A (de)
CA (1) CA2516400C (de)
CY (1) CY1105131T1 (de)
DE (1) DE602004000982T2 (de)
DK (1) DK1605932T3 (de)
EA (1) EA008005B1 (de)
ES (1) ES2262122T3 (de)
HK (1) HK1083596A1 (de)
HR (1) HRP20060240T3 (de)
IL (1) IL170297A (de)
IS (1) IS2310B (de)
MX (1) MXPA05008909A (de)
NO (1) NO20054018L (de)
NZ (1) NZ541875A (de)
PL (1) PL1605932T3 (de)
PT (1) PT1605932E (de)
RS (1) RS50534B (de)
SI (1) SI1605932T1 (de)
UA (1) UA79196C2 (de)
WO (1) WO2005063236A1 (de)
ZA (1) ZA200506550B (de)

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US8211462B2 (en) * 2002-07-30 2012-07-03 Ucb Pharma Gmbh Hot-melt TTS for administering rotigotine
US8246979B2 (en) * 2002-07-30 2012-08-21 Ucb Pharma Gmbh Transdermal delivery system for the administration of rotigotine
US8246980B2 (en) 2002-07-30 2012-08-21 Ucb Pharma Gmbh Transdermal delivery system
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DE10334188B4 (de) * 2003-07-26 2007-07-05 Schwarz Pharma Ag Verwendung von Rotigotin zur Behandlung von Depressionen
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EP1547592A1 (de) 2003-12-23 2005-06-29 Schwarz Pharma Ag Intranasale formulierung enthaltend
DE10361258A1 (de) * 2003-12-24 2005-07-28 Schwarz Pharma Ag Verwendung von substituierten 2-Aminotetralinen zur vorbeugenden Behandlung von Morbus Parkinson
US20050197385A1 (en) * 2004-02-20 2005-09-08 Schwarz Pharma Ag Use of rotigotine for treatment or prevention of dopaminergic neuron loss
DE102004014841B4 (de) * 2004-03-24 2006-07-06 Schwarz Pharma Ag Verwendung von Rotigotin zur Behandlung und Prävention des Parkinson-Plus-Syndroms
TWI392670B (zh) * 2006-06-22 2013-04-11 Ucb Pharma Gmbh 經取代的２-胺基萘滿之於製造用於預防、減緩及／或治療各種類型疼痛之藥物上的用途
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EP2215072B1 (de) * 2007-11-28 2015-09-02 UCB Pharma GmbH Polymorphe rotigotin-form
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EP3257504B1 (de) 2009-12-22 2024-06-19 UCB Biopharma SRL Polyvinylpyrrolidon zur stabilisierung einer feststoffdispersion der nichtkristallinen form von rotigotin
EP2559435A1 (de) 2011-08-19 2013-02-20 UCB Pharma GmbH Rotigotin in der Behandlung von Hemineglekt, Schlaganfall und Defiziten nach einem Schlaganfall
DE102012013439A1 (de) 2012-07-03 2014-01-23 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Transdermales therapeutisches System umfassend Rotigotin und Kristallisationsinhibitor
DE102012013421A1 (de) 2012-07-03 2014-01-09 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Transdermales therapeutisches System (TTS) mit Rotigotin
WO2013075822A1 (en) 2011-11-22 2013-05-30 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Transdermal therapeutic system (tts) with rotigotine
CN103768043B (zh) * 2012-10-22 2015-12-09 苏州药明康德新药开发股份有限公司 采用羟丙基-β-环糊精配制四氢化萘类化合物均一稳定溶液的方法
TW201431570A (zh) 2012-11-22 2014-08-16 Ucb Pharma Gmbh 用於經皮投服羅替戈汀（Ｒｏｔｉｇｏｔｉｎｅ）之多天式貼片
BR112015032929B1 (pt) 2013-07-03 2022-08-23 Lts Lohmann Therapie-Systeme Ag Sistema terapêutico transdérmico com componente eletrônico e métodos de produção de um sistema terapêutico transdérmico
CN106233141B (zh) 2014-02-18 2018-08-21 罗伯特·I·汉金 用于诊断和治疗味觉或嗅觉的损失和/或失真的方法和组合物
CN106456568B (zh) 2014-05-20 2020-03-27 Lts勒曼治疗系统股份公司 包含界面调节剂的经皮递送系统
JP6573913B2 (ja) 2014-05-20 2019-09-11 エルテーエス ローマン テラピー−ジステーメ アーゲー ロチゴチンを含む経皮送達システム
JP6895755B2 (ja) 2014-05-20 2021-06-30 エルテーエス ローマン テラピー−ジステーメ アーゲー 経皮送達システムにおける活性薬剤の放出を調節するための方法
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Also Published As

Publication number Publication date
IS8487A (is) 2006-05-26
EA008005B1 (ru) 2007-02-27
NO20054018L (no) 2005-08-30
IL170297A (en) 2010-06-30
HK1083596A1 (en) 2006-07-07
RS50534B (sr) 2010-05-07
EP1605932A1 (de) 2005-12-21
EP1605932B1 (de) 2006-05-24
PT1605932E (pt) 2006-08-31
DE602004000982T2 (de) 2007-05-10
JP2006526004A (ja) 2006-11-16
IS2310B (is) 2007-11-15
CN100374112C (zh) 2008-03-12
PL1605932T3 (pl) 2006-09-29
CN1777422A (zh) 2006-05-24
SI1605932T1 (sl) 2006-08-31
ZA200506550B (en) 2006-05-31
WO2005063236A1 (en) 2005-07-14
CY1105131T1 (el) 2009-11-04
ES2262122T3 (es) 2006-11-16
EP1547592A1 (de) 2005-06-29
KR20060040578A (ko) 2006-05-10
NZ541875A (en) 2008-08-29
MXPA05008909A (es) 2005-10-05
KR100718760B1 (ko) 2007-05-15
AU2004308641A1 (en) 2005-07-14
DE602004000982D1 (de) 2006-06-29
HRP20060240T3 (en) 2007-05-31
US7683040B2 (en) 2010-03-23
BRPI0407845A (pt) 2006-02-14
AU2004308641B2 (en) 2006-10-26
CA2516400C (en) 2009-10-27
UA79196C2 (en) 2007-05-25
JP4430067B2 (ja) 2010-03-10
EA200501159A1 (ru) 2006-02-24
ATE326961T1 (de) 2006-06-15
CA2516400A1 (en) 2005-07-14
US20070191308A1 (en) 2007-08-16

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