DK1575952T3 - Syntese af heteroarylacetamider - Google Patents

Syntese af heteroarylacetamider

Info

Publication number
DK1575952T3
DK1575952T3 DK03814010T DK03814010T DK1575952T3 DK 1575952 T3 DK1575952 T3 DK 1575952T3 DK 03814010 T DK03814010 T DK 03814010T DK 03814010 T DK03814010 T DK 03814010T DK 1575952 T3 DK1575952 T3 DK 1575952T3
Authority
DK
Denmark
Prior art keywords
heteroaryl
alpha
synthesis
hydroxyacetamide
acetamides
Prior art date
Application number
DK03814010T
Other languages
English (en)
Inventor
Esa T Jarvi
Douglas C Miller
Original Assignee
Mallinckrodt Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mallinckrodt Inc filed Critical Mallinckrodt Inc
Application granted granted Critical
Publication of DK1575952T3 publication Critical patent/DK1575952T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
DK03814010T 2002-12-18 2003-12-16 Syntese af heteroarylacetamider DK1575952T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43576302P 2002-12-18 2002-12-18
PCT/US2003/039951 WO2004058758A1 (en) 2002-12-18 2003-12-16 Synthesis of heteroaryl acetamides

Publications (1)

Publication Number Publication Date
DK1575952T3 true DK1575952T3 (da) 2009-05-25

Family

ID=32682277

Family Applications (1)

Application Number Title Priority Date Filing Date
DK03814010T DK1575952T3 (da) 2002-12-18 2003-12-16 Syntese af heteroarylacetamider

Country Status (12)

Country Link
US (1) US7385056B2 (da)
EP (1) EP1575952B1 (da)
JP (1) JP2006516139A (da)
CN (1) CN100398539C (da)
AT (1) ATE423116T1 (da)
AU (1) AU2003297153B2 (da)
CA (1) CA2509561A1 (da)
DE (1) DE60326270D1 (da)
DK (1) DK1575952T3 (da)
ES (1) ES2320758T3 (da)
MX (1) MXPA05006438A (da)
WO (1) WO2004058758A1 (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7498439B2 (en) 2004-06-22 2009-03-03 Mallinckrodt Inc. Synthesis of heteroaryl acetamides from reaction mixtures having reduced water content
WO2007109120A2 (en) 2006-03-17 2007-09-27 Ambit Biosciences Corporation Imidazolothiazole compounds for the treatment of disease
EP1845098A1 (en) * 2006-03-29 2007-10-17 Ferrer Internacional, S.A. Imidazo[1,2-b]pyridazines, their processes of preparation and their use as GABA receptor ligands
US20080145425A1 (en) * 2006-12-15 2008-06-19 Pliva Research & Development Limited Pharmaceutical composition of zolpidem
PL2201018T3 (pl) 2007-09-19 2016-11-30 STAŁE POSTACIE ZAWIERAJĄCE N-(5-TERT-BUTYLOIZOKSAZOL-3-ILO)-N'-{4--[7-(2-MORFOLIN-4-YLOETOKSY)IMIDAZO[2,1-b][1,3]BENZOTIAZOL-2-ILO]FENYLO}MOCZNIK, ICH KOMPOZYCJE ORAZ ICH ZASTOSOWANIA
UA103918C2 (en) 2009-03-02 2013-12-10 Айерем Элелси N-(hetero)aryl, 2-(hetero)aryl-substituted acetamides for use as wnt signaling modulators
CN103360387B (zh) * 2012-03-28 2016-12-14 江苏豪森药业集团有限公司 一种制备化合物唑吡坦的方法

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492382A1 (fr) 1980-10-22 1982-04-23 Synthelabo Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique
US4675323A (en) 1985-08-06 1987-06-23 Synthelabo Imidazo(1,2-a)quinoline derivatives useful as anxiolytic agents
FR2593179B1 (fr) * 1986-01-22 1988-04-01 Synthelabo Derives d'imidazo(1,2-a)quinoleines, leur preparation et leur application en therapeutique
FR2600650B1 (fr) 1986-06-27 1988-09-09 Synthelabo Procede de preparation d'imidazopyridines et composes intermediaires
FR2606410B1 (fr) * 1986-11-07 1989-02-24 Synthelabo Imidazopyridines, leur preparation et leur application en therapeutique
EP0289371B1 (fr) * 1987-03-27 1991-09-25 Synthelabo Dérivés d'imidazopyridines, leur préparation et leur application en thérapeutique
EP0524055A1 (fr) * 1991-07-19 1993-01-20 Synthelabo Dérivés d'imidazo[2,1-b]benzothiazole-3-acétamide, leur préparation et leur application en thérapeutique
FR2700546B1 (fr) 1993-01-15 1995-02-17 Synthelabo Dérivés d'imidazo[2,1-b]benzoxazole-3-acétamide, leur préparation et leur application en thérapeutique.
EP0607076A1 (fr) * 1993-01-15 1994-07-20 Synthelabo Dérivés de 9h-imidazo 1,2-a benzimidazole-3-acétamide à activité GABA
FR2719843B1 (fr) * 1994-05-10 1996-06-07 Synthelabo Dérivés de 5,6-dihydro-4h-imidazo [2',1':2,3] imidazo-[4,5,1-ij] quinoléine et de 4,5-dihydroimidazo [1,2-a] pyrrolo-[1,2,3-cd] benzimidazole, leur préparation et leur application en thérapeutique.
FR2741073B1 (fr) 1995-11-09 1997-12-12 Synthelabo Derives de 4,5-dihydroimidazo(1,2-a)pyrrolo(1,2,3-cd) benzimidazole, leur preparation et leur application en therapeutique
ES2151834B1 (es) 1998-08-06 2001-08-16 Sint Quimica Sa Procedimiento para preparar n,n,6-trimetil-2-(4-metilfenil)-imidazo-(1,2-a)-piridina-3-acetamida y sus sales.
ES2195510T3 (es) 1999-03-25 2003-12-01 Synthon Bv Derivados de imidazopiridina y procedimiento para prepararlos.
ES2248154T3 (es) 1999-11-22 2006-03-16 Egis Gyogyszergyar Rt. Procedimiento para la preparacion de 6-metil-2-(4-metil-fenil)-imidazo(1,2-a)-piridina-3-(n,n-dimetil-acetamida) y productos intermedios.
DE20122435U1 (de) 2000-04-24 2005-10-06 Teva Pharmaceutical Industries Ltd. Mikronisiertes Zolpidem-Hemitartrat
IT1318624B1 (it) 2000-07-14 2003-08-27 Dinamite Dipharma S P A In For Processo per la preparazione di 2-fenil-imidazo (1,2-a)piridin-3-acetammidi.
WO2002014306A1 (en) 2000-08-17 2002-02-21 Cilag Ag Process for the preparation of imidazopyridines
US6921839B2 (en) 2000-08-29 2005-07-26 Ranbaxy Laboratories Limited Synthesis of N,N-dimethyl-3-(4-methyl) benzoyl propionamide a key intermediate of zolpidem
ATE394398T1 (de) * 2002-07-15 2008-05-15 Scinopharm Taiwan Ltd Verfahren zur herstellung von imidazo(1,2- a)pyridin-3-acetamiden
US7498439B2 (en) * 2004-06-22 2009-03-03 Mallinckrodt Inc. Synthesis of heteroaryl acetamides from reaction mixtures having reduced water content

Also Published As

Publication number Publication date
ES2320758T3 (es) 2009-05-28
AU2003297153A1 (en) 2004-07-22
WO2004058758A1 (en) 2004-07-15
JP2006516139A (ja) 2006-06-22
DE60326270D1 (de) 2009-04-02
CN100398539C (zh) 2008-07-02
CN1729188A (zh) 2006-02-01
ATE423116T1 (de) 2009-03-15
US7385056B2 (en) 2008-06-10
EP1575952A1 (en) 2005-09-21
EP1575952B1 (en) 2009-02-18
MXPA05006438A (es) 2005-09-08
CA2509561A1 (en) 2004-07-15
US20060025588A1 (en) 2006-02-02
AU2003297153B2 (en) 2010-06-10

Similar Documents

Publication Publication Date Title
DE60100534D1 (de) Vorrichtung für den Ruf-Betrieb in Mobilfunksystemen
DE60226098D1 (de) Lautsprechersystem, Mobilendgerät und elektronische Vorrichtung
ATE483752T1 (de) Wässrige dispersion, herstellungsverfahren dafür und verwendung davon
NL1021362A1 (nl) Katalysator- en oplosmiddelsamenstelling en katalysewerkwijzen waarbij deze samenstelling wordt toegepast.
DE60333589D1 (de) Kommunikationssystem and kommunikationsverfahren
EE05015B1 (et) Makseterminaliseade mgipunktiseadme hendamiseks, maksessteem ja makseprotseduuri teostamise meetod
DE60020726D1 (de) Biaryletherderivate, die als inhibitoren der monoamin-wiederaufnahme nützlich sind
DE60330400D1 (de) Sprachsynthesesystem, Sprachsyntheseverfahren und Rechnerprogramm
FI20055668A0 (fi) Antennimoduuli ja sitä käyttävä elektroninen laite
MX225920B (es) Dispersion polimerica termoendurecedora.
DE60222227D1 (de) Kommunikationssystem, drahtlose Kommunikationsvorrichtung und Kommunikationsverfahren
ATE343569T1 (de) Aromatische hydroxamsäurederivate, die sich als hdac inhibitoren eignen
DE60231842D1 (de) Kleine multimodeantenne und diese verwendendes hochfrequenzmodul
DE60239546D1 (de) Kommunikationsverfahren, kommunikationssystem und ausgabevorrichtung
DK1282663T3 (da) Gel af et poly-a-1,4-glucan og stivelse
DE60332724D1 (de) Kommunikationsgerät, kommunikationssystem, kommunikationsverfahren und programm dafür
DE60204304D1 (de) Katalysatoraktivierungsverfahren
DE60200136D1 (de) Einweg-Roaming von ANS-41 zu GSM Systemen
DE602004016901D1 (de) Informationsverarbeitungsgerät, Informationsausgabegerät, tragbares Endgerät und Informationsausgabeverfahren
DK1575952T3 (da) Syntese af heteroarylacetamider
NO20044448L (no) Nye forbindelser
DE60223706D1 (de) Kommunikationsunterstützungsverfahren, kommunikationsserver dieses umfassend und kommunikationsunterstützungssystem
DE50210349D1 (de) Hochfrequenz Verbindungsvorrichtung
BR0202786B1 (pt) processo de sìntese de uréia.
ITMI20020202A0 (it) Dispositivo atto al trattamento di gas di scarico comprendente un catalizzatore accumulatore