DE60326270D1 - Synthese von heteroaryl acetamiden - Google Patents

Synthese von heteroaryl acetamiden

Info

Publication number
DE60326270D1
DE60326270D1 DE60326270T DE60326270T DE60326270D1 DE 60326270 D1 DE60326270 D1 DE 60326270D1 DE 60326270 T DE60326270 T DE 60326270T DE 60326270 T DE60326270 T DE 60326270T DE 60326270 D1 DE60326270 D1 DE 60326270D1
Authority
DE
Germany
Prior art keywords
heteroaryl
alpha
synthesis
hydroxyacetamide
acetamides
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60326270T
Other languages
English (en)
Inventor
Esa T Jarvi
Douglas C Miller
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Mallinckrodt Inc
Original Assignee
Mallinckrodt Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mallinckrodt Inc filed Critical Mallinckrodt Inc
Application granted granted Critical
Publication of DE60326270D1 publication Critical patent/DE60326270D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
DE60326270T 2002-12-18 2003-12-16 Synthese von heteroaryl acetamiden Expired - Lifetime DE60326270D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43576302P 2002-12-18 2002-12-18
PCT/US2003/039951 WO2004058758A1 (en) 2002-12-18 2003-12-16 Synthesis of heteroaryl acetamides

Publications (1)

Publication Number Publication Date
DE60326270D1 true DE60326270D1 (de) 2009-04-02

Family

ID=32682277

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60326270T Expired - Lifetime DE60326270D1 (de) 2002-12-18 2003-12-16 Synthese von heteroaryl acetamiden

Country Status (12)

Country Link
US (1) US7385056B2 (de)
EP (1) EP1575952B1 (de)
JP (1) JP2006516139A (de)
CN (1) CN100398539C (de)
AT (1) ATE423116T1 (de)
AU (1) AU2003297153B2 (de)
CA (1) CA2509561A1 (de)
DE (1) DE60326270D1 (de)
DK (1) DK1575952T3 (de)
ES (1) ES2320758T3 (de)
MX (1) MXPA05006438A (de)
WO (1) WO2004058758A1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2571491A1 (en) 2004-06-22 2006-01-19 Mallinckrodt, Inc. Synthesis of heteroaryl acetamides from reaction mixtures having reduced water content
PT2001892E (pt) 2006-03-17 2013-07-04 Ambit Biosciences Corp Compostos de imidazolotiazole para o tratamento de doenças proliferativas
EP1845098A1 (de) * 2006-03-29 2007-10-17 Ferrer Internacional, S.A. Imidazo[1,2-b]pyridazinen, deren Herstellungverfahren und ihre Verwendung als GABA Rezeptor Liganden
US20080145425A1 (en) * 2006-12-15 2008-06-19 Pliva Research & Development Limited Pharmaceutical composition of zolpidem
WO2009038757A2 (en) 2007-09-19 2009-03-26 Ambit Biosciences Corporation Solid forms comprising n-(5-tert-butyl-isoxazol-3-yl)-n'-{4-[7-(2-morpholin-4-yl-ethoxy)imidazo[2,1-b][1,3]benzothiazol-2-yl]phenyl}urea, compositions thereof, and uses therewith
UA103918C2 (en) 2009-03-02 2013-12-10 Айерем Элелси N-(hetero)aryl, 2-(hetero)aryl-substituted acetamides for use as wnt signaling modulators
CN103360387B (zh) * 2012-03-28 2016-12-14 江苏豪森药业集团有限公司 一种制备化合物唑吡坦的方法

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492382A1 (fr) * 1980-10-22 1982-04-23 Synthelabo Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique
US4675323A (en) 1985-08-06 1987-06-23 Synthelabo Imidazo(1,2-a)quinoline derivatives useful as anxiolytic agents
FR2593179B1 (fr) 1986-01-22 1988-04-01 Synthelabo Derives d'imidazo(1,2-a)quinoleines, leur preparation et leur application en therapeutique
FR2600650B1 (fr) * 1986-06-27 1988-09-09 Synthelabo Procede de preparation d'imidazopyridines et composes intermediaires
FR2606410B1 (fr) * 1986-11-07 1989-02-24 Synthelabo Imidazopyridines, leur preparation et leur application en therapeutique
EP0289371B1 (de) * 1987-03-27 1991-09-25 Synthelabo Imidazopyridinderivate, ihre Herstellung und therapeutische Verwendung
EP0524055A1 (de) * 1991-07-19 1993-01-20 Synthelabo Imidazo(2,1-b)benzothiazolderivate, Verfahren zu ihrer Herstellung und ihre therapeutische Verwendung
EP0607076A1 (de) * 1993-01-15 1994-07-20 Synthelabo 9H-Imidazo 1,2-a benzimidazolderivate mit GABA wirkung
FR2700546B1 (fr) 1993-01-15 1995-02-17 Synthelabo Dérivés d'imidazo[2,1-b]benzoxazole-3-acétamide, leur préparation et leur application en thérapeutique.
FR2719843B1 (fr) * 1994-05-10 1996-06-07 Synthelabo Dérivés de 5,6-dihydro-4h-imidazo [2',1':2,3] imidazo-[4,5,1-ij] quinoléine et de 4,5-dihydroimidazo [1,2-a] pyrrolo-[1,2,3-cd] benzimidazole, leur préparation et leur application en thérapeutique.
FR2741073B1 (fr) 1995-11-09 1997-12-12 Synthelabo Derives de 4,5-dihydroimidazo(1,2-a)pyrrolo(1,2,3-cd) benzimidazole, leur preparation et leur application en therapeutique
ES2151834B1 (es) 1998-08-06 2001-08-16 Sint Quimica Sa Procedimiento para preparar n,n,6-trimetil-2-(4-metilfenil)-imidazo-(1,2-a)-piridina-3-acetamida y sus sales.
DK1038875T3 (da) 1999-03-25 2003-09-29 Synthon Bv Imidazopyridine- derivativer og fremgangsmåde til fremstilling deraf
CN1227252C (zh) 1999-11-22 2005-11-16 埃吉斯药物工厂 制备6－甲基－2－(4－甲基－苯基)－咪唑并[1,2－a]吡啶－3－(N,N－二甲基－乙酰胺)和中间体的方法
EP1292304B1 (de) 2000-04-24 2005-11-02 Teva Pharmaceutical Industries Ltd. Zolpidem hemitartrat
IT1318624B1 (it) 2000-07-14 2003-08-27 Dinamite Dipharma S P A In For Processo per la preparazione di 2-fenil-imidazo (1,2-a)piridin-3-acetammidi.
AU2000264428A1 (en) 2000-08-17 2002-02-25 Cilag A.G. Process for the preparation of imidazopyridines
US6921839B2 (en) 2000-08-29 2005-07-26 Ranbaxy Laboratories Limited Synthesis of N,N-dimethyl-3-(4-methyl) benzoyl propionamide a key intermediate of zolpidem
CN100408577C (zh) * 2002-07-15 2008-08-06 台湾神隆股份有限公司 咪唑并(1,2-a)吡啶-3-乙酰胺类的制备方法
CA2571491A1 (en) * 2004-06-22 2006-01-19 Mallinckrodt, Inc. Synthesis of heteroaryl acetamides from reaction mixtures having reduced water content

Also Published As

Publication number Publication date
US7385056B2 (en) 2008-06-10
AU2003297153A1 (en) 2004-07-22
ES2320758T3 (es) 2009-05-28
AU2003297153B2 (en) 2010-06-10
MXPA05006438A (es) 2005-09-08
CN1729188A (zh) 2006-02-01
EP1575952B1 (de) 2009-02-18
ATE423116T1 (de) 2009-03-15
DK1575952T3 (da) 2009-05-25
CN100398539C (zh) 2008-07-02
CA2509561A1 (en) 2004-07-15
WO2004058758A1 (en) 2004-07-15
US20060025588A1 (en) 2006-02-02
EP1575952A1 (de) 2005-09-21
JP2006516139A (ja) 2006-06-22

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