DK149111C - Analogifremgangsmaade til fremstilling af histidinderivater eller syreadditionssalte deraf - Google Patents
Analogifremgangsmaade til fremstilling af histidinderivater eller syreadditionssalte derafInfo
- Publication number
- DK149111C DK149111C DK119577A DK119577A DK149111C DK 149111 C DK149111 C DK 149111C DK 119577 A DK119577 A DK 119577A DK 119577 A DK119577 A DK 119577A DK 149111 C DK149111 C DK 149111C
- Authority
- DK
- Denmark
- Prior art keywords
- histidin
- analogue
- derivatives
- preparation
- acid addition
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/26—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D307/30—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/32—Oxygen atoms
- C07D307/33—Oxygen atoms in position 2, the oxygen atom being in its keto or unsubstituted enol form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
- C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Biophysics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Molecular Biology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Genetics & Genomics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biochemistry (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP3217076 | 1976-03-23 | ||
| JP51032170A JPS5944308B2 (ja) | 1976-03-23 | 1976-03-23 | ペプタイド |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK119577A DK119577A (da) | 1977-09-24 |
| DK149111B DK149111B (da) | 1986-01-27 |
| DK149111C true DK149111C (da) | 1986-06-09 |
Family
ID=12351453
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK119577A DK149111C (da) | 1976-03-23 | 1977-03-18 | Analogifremgangsmaade til fremstilling af histidinderivater eller syreadditionssalte deraf |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US4100152A (es) |
| JP (1) | JPS5944308B2 (es) |
| AT (1) | AT360674B (es) |
| AU (1) | AU508387B2 (es) |
| BE (1) | BE852740A (es) |
| CA (1) | CA1060435A (es) |
| CH (1) | CH634548A5 (es) |
| DE (1) | DE2712086C2 (es) |
| DK (1) | DK149111C (es) |
| FR (1) | FR2345448A1 (es) |
| GB (1) | GB1579264A (es) |
| GR (1) | GR62565B (es) |
| HK (1) | HK27584A (es) |
| HU (1) | HU177515B (es) |
| MY (1) | MY8500264A (es) |
| NL (1) | NL188412C (es) |
| SE (1) | SE430601B (es) |
| SG (1) | SG76083G (es) |
| ZA (1) | ZA771495B (es) |
Families Citing this family (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU180926B (en) * | 1979-06-28 | 1983-05-30 | Richter Gedeon Vegyeszet | Process for preparing trh analogues,tripeptide amides infectives on the central nerve sysrhem |
| US4591648A (en) * | 1981-04-01 | 1986-05-27 | National Research Development Corp. | Histidine protection |
| US4426378A (en) | 1981-04-09 | 1984-01-17 | The United States Of America As Represented By The Secretary Of The Army | Thyrotropin releasing hormone in therapy of shock and as a central nervous system stimulant |
| JPS5849313A (ja) * | 1981-09-16 | 1983-03-23 | Takeda Chem Ind Ltd | 抗てんかん剤 |
| US4659696A (en) * | 1982-04-30 | 1987-04-21 | Takeda Chemical Industries, Ltd. | Pharmaceutical composition and its nasal or vaginal use |
| GB2146026A (en) * | 1983-09-07 | 1985-04-11 | Tanabe Seiyaku Co | Peptides and process for preparing the same |
| JPS60190795A (ja) * | 1984-03-09 | 1985-09-28 | Takeda Chem Ind Ltd | ペプタイド |
| US4608365A (en) * | 1984-03-30 | 1986-08-26 | University Of Southern California | Treatment of neurologic functions |
| IL75641A (en) * | 1984-07-10 | 1990-11-05 | Tanabe Seiyaku Co | 1-methyl-4,5-dihydro-orotyl-histidyl-prolinamide,its preparation and pharmaceutical compositions comprising it |
| GB2171101A (en) * | 1985-02-20 | 1986-08-20 | Tanabe Seiyaku Co | Peptide and processes for preparation of the same |
| FR2585709B1 (fr) * | 1985-08-05 | 1987-10-02 | Adir | Nouveaux derives peptidiques a structure lactonique ou cycloamidique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| JP2526589B2 (ja) * | 1986-08-08 | 1996-08-21 | 武田薬品工業株式会社 | ペプチド含有マイクロカプセルおよびその製造法 |
| US5686420A (en) * | 1987-06-05 | 1997-11-11 | Georgetown University | Thyrotropin-releasing hormone analogs and method of use |
| JPS63316724A (ja) * | 1987-06-19 | 1988-12-26 | Nippon Shinyaku Co Ltd | 抗けいれん剤 |
| US5151497A (en) * | 1989-02-21 | 1992-09-29 | Japan Tobacco Inc. | Histidyl peptide derivatives |
| CA2050425A1 (en) | 1990-09-03 | 1992-03-04 | Yoshiaki Uda | Pharmaceutical composition and its mucous use |
| NZ240214A (en) | 1990-10-16 | 1993-02-25 | Takeda Chemical Industries Ltd | Polymer compositions comprising a polylactic acid and a copolymer of glycolic acid and a hydroxycarboxylic acid; use as carrier for prolonged release pharmaceutical compositions of water soluble drugs |
| US5416071A (en) * | 1991-03-12 | 1995-05-16 | Takeda Chemical Industries, Ltd. | Water-soluble composition for sustained-release containing epo and hyaluronic acid |
| ATE161716T1 (de) | 1992-08-07 | 1998-01-15 | Takeda Chemical Industries Ltd | Herstellung von mikrokapseln, die wasserlösliche arzneimittel enthalten |
| US6117455A (en) * | 1994-09-30 | 2000-09-12 | Takeda Chemical Industries, Ltd. | Sustained-release microcapsule of amorphous water-soluble pharmaceutical active agent |
| US5837281A (en) | 1995-03-17 | 1998-11-17 | Takeda Chemical Industries, Ltd. | Stabilized interface for iontophoresis |
| JPH11515014A (ja) * | 1995-10-24 | 1999-12-21 | グルーエネンタール ゲゼルシャフト ミット ベシュレンクテル ハフツング | 哺乳類の概日リズムの調整方法 |
| CA2192782C (en) | 1995-12-15 | 2008-10-14 | Nobuyuki Takechi | Production of microspheres |
| EP0813887A3 (en) * | 1996-06-20 | 1999-11-03 | Hisamitsu Pharmaceutical Co. Inc. | A device structure for iontophoresis |
| AU713133B2 (en) * | 1996-08-28 | 1999-11-25 | Shionogi & Co., Ltd. | Novel peptide derivatives having thiazolyl-alanine residue |
| EP1025089A1 (en) * | 1997-10-22 | 2000-08-09 | Zeneca Limited | Imidazole derivatives and their use as farnesyl protein transferase inhibitors |
| US6342765B1 (en) | 1997-10-22 | 2002-01-29 | Astrazeneca Uk Limited | Imidazole derivatives and their use as farnesyl protein transferase inhibitors |
| US6458790B2 (en) * | 2000-03-23 | 2002-10-01 | Merck & Co., Inc. | Substituted piperidines as melanocortin receptor agonists |
| KR20050105290A (ko) * | 2000-08-31 | 2005-11-03 | 시오노기세이야쿠가부시키가이샤 | 파킨슨씨병 치료제 |
| CA2430934C (en) | 2000-12-01 | 2011-06-21 | Takeda Chemical Industries, Ltd. | A method of producing sustained-release preparations of a bioactive substance using high-pressure gas |
| GB0326632D0 (en) | 2003-11-14 | 2003-12-17 | Jagotec Ag | Dry powder formulations |
| EP2611416B1 (en) | 2010-09-03 | 2015-08-19 | Pharmaterials Ltd. | Pharmaceutical composition suitable for use in a dry powder inhaler |
| JP6224586B2 (ja) | 2012-07-10 | 2017-11-01 | 武田薬品工業株式会社 | 注射用製剤 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3753969A (en) * | 1969-12-22 | 1973-08-21 | K Folkers | Method for synthesizing pyroglutamylhistidyl-prolinamide |
| US3821188A (en) * | 1972-06-14 | 1974-06-28 | American Home Prod | Proline and pyroglutamic acid containing tripeptides |
| US3959248A (en) * | 1974-04-03 | 1976-05-25 | Merck & Co., Inc. | Analogs of thyrotropin-releasing hormone |
| DE2449167C2 (de) * | 1974-10-16 | 1984-05-24 | Grünenthal GmbH, 5190 Stolberg | N-Acyl-L-histidyl-L-prolinamide, Verfahren zu deren Herstellung und diese Verbindungen enthaltende pharmazeutische Zubereitungen |
-
1976
- 1976-03-23 JP JP51032170A patent/JPS5944308B2/ja not_active Expired
-
1977
- 1977-03-11 ZA ZA00771495A patent/ZA771495B/xx unknown
- 1977-03-16 US US05/778,321 patent/US4100152A/en not_active Expired - Lifetime
- 1977-03-18 GR GR53020A patent/GR62565B/el unknown
- 1977-03-18 DK DK119577A patent/DK149111C/da not_active IP Right Cessation
- 1977-03-19 DE DE2712086A patent/DE2712086C2/de not_active Expired
- 1977-03-22 FR FR7708576A patent/FR2345448A1/fr active Granted
- 1977-03-22 CH CH361677A patent/CH634548A5/de not_active IP Right Cessation
- 1977-03-22 SE SE7703283A patent/SE430601B/xx not_active IP Right Cessation
- 1977-03-22 BE BE176000A patent/BE852740A/xx not_active IP Right Cessation
- 1977-03-22 NL NLAANVRAGE7703115,A patent/NL188412C/xx not_active IP Right Cessation
- 1977-03-22 HU HU77TA1428A patent/HU177515B/hu not_active IP Right Cessation
- 1977-03-22 CA CA274,478A patent/CA1060435A/en not_active Expired
- 1977-03-23 AU AU23549/77A patent/AU508387B2/en not_active Expired
- 1977-03-23 GB GB12204/77A patent/GB1579264A/en not_active Expired
- 1977-03-23 AT AT202377A patent/AT360674B/de not_active IP Right Cessation
-
1983
- 1983-12-02 SG SG760/83A patent/SG76083G/en unknown
-
1984
- 1984-03-22 HK HK275/84A patent/HK27584A/xx unknown
-
1985
- 1985-12-30 MY MY264/85A patent/MY8500264A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FR2345448B1 (es) | 1980-06-27 |
| AT360674B (de) | 1981-01-26 |
| GR62565B (en) | 1979-05-10 |
| DK149111B (da) | 1986-01-27 |
| NL188412C (nl) | 1992-06-16 |
| AU2354977A (en) | 1978-09-28 |
| DE2712086C2 (de) | 1986-04-03 |
| NL188412B (nl) | 1992-01-16 |
| SE430601B (sv) | 1983-11-28 |
| NL7703115A (nl) | 1977-09-27 |
| CA1060435A (en) | 1979-08-14 |
| AU508387B2 (en) | 1980-03-20 |
| GB1579264A (en) | 1980-11-19 |
| CH634548A5 (de) | 1983-02-15 |
| DK119577A (da) | 1977-09-24 |
| SG76083G (en) | 1984-08-03 |
| JPS5944308B2 (ja) | 1984-10-29 |
| HK27584A (en) | 1984-03-30 |
| ZA771495B (en) | 1978-02-22 |
| US4100152A (en) | 1978-07-11 |
| MY8500264A (en) | 1985-12-31 |
| ATA202377A (de) | 1980-06-15 |
| HU177515B (en) | 1981-10-28 |
| BE852740A (fr) | 1977-07-18 |
| DE2712086A1 (de) | 1977-09-29 |
| SE7703283L (sv) | 1977-09-24 |
| JPS52116465A (en) | 1977-09-29 |
| FR2345448A1 (fr) | 1977-10-21 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK149111C (da) | Analogifremgangsmaade til fremstilling af histidinderivater eller syreadditionssalte deraf | |
| DK150512C (da) | Analogifremgangsmaade til fremstilling af 3-quino-lincarboxylsyrederivater eller syreadditionssalte deraf | |
| DK144010C (da) | Analogifremgangsmaade til fremstilling af 2-piperazinyl-6,7-dimethoxyquinazoliner eller syreadditionssalte deraf | |
| DK147362C (da) | Analogifremgangsmaade til fremstilling af ergolen- eller ergolin-derivater eller syreadditionssalte deraf | |
| DK462380A (da) | Analogifremgangsmaade til fremstilling af 2,4-diaminoquinazolin-forbindelser eller syreadditionssalte deraf | |
| DK145119C (da) | Analogifremgangsmaade til fremstilling af phenolethere eller syreadditionssalte deraf | |
| DK143275C (da) | Analogifremgangsmaade til fremstilling af 1-(3-dimethylaminopropyl)-phthalanderivater eller syreadditionssalte deraf | |
| DK145260C (da) | Analogifremgangsmaade til fremstilling af 4-acylamino-phenyl-ethanolaminer eller syreadditionssalte heraf | |
| DK147858C (da) | Analogifremgangsmaade til fremstilling af 5'-deoxy-5-fluorcytidin eller 5'-deoxy-5-fluoruridin eller fysiologisk tolerable syreadditionssalte dera | |
| DK146592C (da) | Analogifremgangsmaade til fremstilling af n-substituerede benzensulfonamider eller syreadditionssalte deraf | |
| DK392877A (da) | Fremgangsmaade til fremstilling af phenylethylaminer eller syreadditionssalte heraf | |
| DK413783D0 (da) | Fremgangsmade til fremstilling af 20-amino-macrolidderivater eller syreadditionssalte deraf | |
| DK146281C (da) | Analogifremgangsmaade til fremstilling af 2-brom-6-fluor-n-2-imidazolidinyliden-benzamin eller syreadditionssalte heraf | |
| DK140695B (da) | Analogifremgangsmaade til fremstilling af 2,4-diamo-6,7-dimethoxyquinazolinderivater eller syreadditionssalte heraf | |
| DK159079A (da) | Fremgangsmaade til fremstilling af derivater af 4-amino-2-piperidinoquinazolin eller syreadditionssalte deraf | |
| DK149077C (da) | Analogifremgangsmaade til fremstilling af encephalin-analoge pentapeptidamidderivater eller farmaceutisk acceptable syreadditionssalte deraf | |
| DK58677A (da) | Fremgangsmade til fremstilling af m-trifluormethylphenylpiperidinderivater eller additionssalte deraf | |
| DK148281C (da) | Analogifremgangsmaade til fremstilling af 8a-substituerede 8,8a-desoxy-8,8a-dihydrooleandomycin-forbindelser eller farmaceutiskacceptable syreadditionssalte deraf | |
| DK149628C (da) | Analogifremgangsmaade til fremstilling af 8-substitueret-4ae-amino-makrolider eller syreadditionssalte deraf | |
| DK151629C (da) | Analogifremgangsmaade til fremstilling af 3-amino-1-benzoxepin-5(2h)-on-derivater eller syreadditionssalte deraf | |
| DK146886C (da) | Analogifremgangsmaade til fremstilling af basisk substituerede o-propylerede oximer eller fysiologisk acceptable syreadditionssalte deraf | |
| DK148036C (da) | Analogifremgangsmaade til fremstilling af epimere 4''-amino-erythromycin-forbindelser eller syreadditionssalte deraf | |
| DK148683C (da) | Analogifremgangsmaade til fremstilling af pyridazinylhydrazinderivater eller farmaceutisk acceptable syreadditionssalte deraf | |
| DK142172C (da) | Analogifremgangsmaade til fremstilling af basisk substituerede2-alkylamino-4-phenylimidazoliner eller syreadditionssalte heraf | |
| DK516480A (da) | Fremgangsmaade til fremstilling af 2-amino-ethanol-derivater eller syreadditionssalte deraf |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PBP | Patent lapsed |