DK148826C - Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade - Google Patents

Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade

Info

Publication number
DK148826C
DK148826C DK504881A DK504881A DK148826C DK 148826 C DK148826 C DK 148826C DK 504881 A DK504881 A DK 504881A DK 504881 A DK504881 A DK 504881A DK 148826 C DK148826 C DK 148826C
Authority
DK
Denmark
Prior art keywords
procedure
derivatives
pyrimidide
bases
salts
Prior art date
Application number
DK504881A
Other languages
Danish (da)
English (en)
Other versions
DK504881A (da
DK148826B (da
Inventor
Urs Hengartner
Jean-Claude Muller
Henri Ramuz
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK504881A publication Critical patent/DK504881A/da
Publication of DK148826B publication Critical patent/DK148826B/da
Application granted granted Critical
Publication of DK148826C publication Critical patent/DK148826C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK504881A 1980-12-19 1981-11-13 Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade DK148826C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH941080 1980-12-19
CH941080 1980-12-19
CH635081 1981-10-02
CH635081 1981-10-02

Publications (3)

Publication Number Publication Date
DK504881A DK504881A (da) 1982-06-20
DK148826B DK148826B (da) 1985-10-14
DK148826C true DK148826C (da) 1986-03-24

Family

ID=25699419

Family Applications (1)

Application Number Title Priority Date Filing Date
DK504881A DK148826C (da) 1980-12-19 1981-11-13 Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade

Country Status (23)

Country Link
US (2) US4410698A (no)
EP (1) EP0054866B1 (no)
KR (1) KR880001636B1 (no)
AR (1) AR229169A1 (no)
AT (1) ATE14734T1 (no)
AU (1) AU545324B2 (no)
BR (1) BR8108269A (no)
CA (1) CA1162538A (no)
CS (1) CS226738B2 (no)
DE (1) DE3171744D1 (no)
DK (1) DK148826C (no)
ES (1) ES8304125A1 (no)
FI (1) FI71153C (no)
GR (1) GR76969B (no)
HU (1) HU183744B (no)
IE (1) IE51800B1 (no)
IL (1) IL64524A (no)
MC (1) MC1438A1 (no)
NO (1) NO158422C (no)
NZ (1) NZ199250A (no)
PH (1) PH17300A (no)
PT (1) PT74153B (no)
ZW (1) ZW28581A1 (no)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK148826C (da) * 1980-12-19 1986-03-24 Hoffmann La Roche Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade
CH649291A5 (de) * 1982-03-16 1985-05-15 Hoffmann La Roche Dicarbamate.
EP0187854A4 (en) * 1984-07-13 1987-01-22 Gail S Bazzano SUBSTITUTED PYRIMIDINE OXIDES USEFUL FOR PROMOTING HAIR GROWTH.
LU86959A1 (fr) * 1987-07-31 1989-03-08 Oreal Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie
DE69715869T2 (de) * 1996-07-26 2003-05-28 Vantico Ag, Basel Auf epoxyharzen basierende imidazole enthaltende härtbare mischungen
CN117946133B (zh) * 2024-01-05 2024-08-06 南京理工大学 一种5-(4-氨基-1,2,5-噁二唑-3-基)[1,2,5]噁二唑并[3,4-d]嘧啶-7-胺及其制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH638215A5 (de) * 1977-02-04 1983-09-15 Hoffmann La Roche Oxadiazolopyrimidin-derivate.
CH638216A5 (de) * 1977-02-04 1983-09-15 Hoffmann La Roche Oxadiazolopyrimidin-deriate.
CA1103245A (en) * 1978-07-21 1981-06-16 Jean-Claude Muller Process for the manufacture of novel oxadiazolopyrimidine derivatives
NZ190915A (en) * 1978-07-31 1984-07-31 Hoffmann La Roche Oxadiazolotriazine derivatives and pharmaceutical compositions
DK148826C (da) * 1980-12-19 1986-03-24 Hoffmann La Roche Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade

Also Published As

Publication number Publication date
FI71153B (fi) 1986-08-14
ZW28581A1 (en) 1982-08-11
DK504881A (da) 1982-06-20
AU545324B2 (en) 1985-07-11
FI814048L (fi) 1982-06-20
IL64524A0 (en) 1982-03-31
EP0054866B1 (de) 1985-08-07
NO158422C (no) 1988-09-07
ATE14734T1 (de) 1985-08-15
ES508152A0 (es) 1983-02-16
HU183744B (en) 1984-05-28
AU7846481A (en) 1982-06-24
US4360521A (en) 1982-11-23
FI71153C (fi) 1986-11-24
ES8304125A1 (es) 1983-02-16
DE3171744D1 (en) 1985-09-12
NZ199250A (en) 1984-04-27
EP0054866A3 (en) 1982-09-01
PT74153B (en) 1984-01-05
US4410698A (en) 1983-10-18
IE812990L (en) 1982-06-19
IE51800B1 (en) 1987-04-01
AR229169A1 (es) 1983-06-30
CA1162538A (en) 1984-02-21
IL64524A (en) 1985-05-31
GR76969B (no) 1984-09-04
PT74153A (en) 1982-01-01
DK148826B (da) 1985-10-14
PH17300A (en) 1984-07-18
EP0054866A2 (de) 1982-06-30
CS226738B2 (en) 1984-04-16
BR8108269A (pt) 1982-10-05
NO158422B (no) 1988-05-30
MC1438A1 (fr) 1982-12-06
NO814359L (no) 1982-06-21
KR880001636B1 (ko) 1988-09-03

Similar Documents

Publication Publication Date Title
DK156434C (da) Analogifremgangsmaade til fremstilling af sulfonylurinstoffer eller deres fysiologisk acceptable salte
DK149599C (da) Fremgangsmaade til fremstilling af aminosukkerderivater kaldet trestatina, trestatin b og trestatin c eller salte deraf
DK148260C (da) Analogifremgangsmaade til fremstilling af 1,3,8-trisubstituerede xantinderivater eller salte deraf
DK397387A (da) Carbostyrilderivater og salte deraf samt fremgangsmaade til fremstilling af saadanne forbindelser
DK70083A (da) Fremgangsmaade til fremstilling af pyrroleddikesyreamider eller salte deraf
DK160561C (da) Analogifremgangsmaade til fremstilling af 3-aminopregn-5-enderivater eller salte deraf
DK5976A (da) Fremgangsmade til fremstilling af biphenyloxyderivater eller salte heraf
DK160421C (da) Analogifremgangsmaade til fremstilling af 4-oxo-1,4-dihydronicotinsyrederivater eller salte deraf
DK158658C (da) Analogifremgangsmaade til fremstilling af 9-aminoalkylfluorener eller farmaceutisk acceptable salte deraf
DK27078A (da) Fremgangsmaade til fremstilling af imidazoquinoliner eller salte deraf
DK324979A (da) Fremgangsmaade til fremstilling af imidazoquinoxaliner eller salte deraf
DK157538C (da) Analogifremgangsmaade til fremstilling af heterocycliske phenoxyaminer samt 1-cyclohexenylmethyl-pyrrolidiner til anvendelse som mellemprodukt ved fremgangsmaaden
DK148826C (da) Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade
DK511878A (da) Fremgangsmaade til fremstilling af imidazobenzoazepiner eller salte deraf
DK156066C (da) Analogifremgangsmaade til fremstilling af oxaloamino- eller hydroxyacetylaminobenzopyranderivater eller salte deraf med baser
DK151957C (da) Analogifremgangsmaade til fremstilling af 3-substituerede 2-oxo-1-benzimidazolinalkansyrer eller estere eller amider deraf eller salte deraf med baser
DK127676A (da) Fremgangsmade til fremstilling af 9-alkylamino-erythromyciner eller salte deraf
DK162050C (da) Pyrazolderivater med ergolinskelet eller salte deraf, deres fremstilling, farmaceutiske praeparater indeholdende disse og fremgangsmaade til fremstilling af de farmaceutiske praeparater
DK150206C (da) Analogifremgangsmaade til fremstilling af lrf-analoge nona- eller decapeptidamider eller ikke-toksiske salte deraf og nona- eller decapeptidderivater til anvendelse som udgangsforbindelser ved fremgangsmaaden
DK139677A (da) Fremgangsmade til fremstilling af benzazepiner eller deres salte
DK152491C (da) Analogifremgangsmaade til fremstilling af esterholdige phenoxypropanolaminer eller farmaceutisk anvendelige salte deraf
DK224381A (da) Fremgangsmaade til fremstilling af benzazolderivater eller salte deraf
DK149823C (da) Fremgangsmaade til fremstilling af kijanimicin eller farmaceutisk acceptable salte heraf
DK154021C (da) Analogifremgangsmaade til fremstilling af phenoxy-aminopropanolderivater og epoxider til anvendelse som udgangsmateriale ved denne fremgangsmaade
DK143403C (da) Analogifremgangsmaade til fremstilling af 8-(1h-tetrazol-5-yl)-11h-pyrido(2,1-b)quinazolin-11-oner eller salte deraf

Legal Events

Date Code Title Description
PBP Patent lapsed