DK1456189T3 - Benzothia(dia)zin-derivater og deres anvendelse som AMPA-modulatorer - Google Patents
Benzothia(dia)zin-derivater og deres anvendelse som AMPA-modulatorerInfo
- Publication number
- DK1456189T3 DK1456189T3 DK02805407T DK02805407T DK1456189T3 DK 1456189 T3 DK1456189 T3 DK 1456189T3 DK 02805407 T DK02805407 T DK 02805407T DK 02805407 T DK02805407 T DK 02805407T DK 1456189 T3 DK1456189 T3 DK 1456189T3
- Authority
- DK
- Denmark
- Prior art keywords
- benzothia
- zin
- dia
- derivatives
- ampa modulators
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/15—Six-membered rings
- C07D285/16—Thiadiazines; Hydrogenated thiadiazines
- C07D285/18—1,2,4-Thiadiazines; Hydrogenated 1,2,4-thiadiazines
- C07D285/20—1,2,4-Thiadiazines; Hydrogenated 1,2,4-thiadiazines condensed with carbocyclic rings or ring systems
- C07D285/22—1,2,4-Thiadiazines; Hydrogenated 1,2,4-thiadiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D285/24—1,2,4-Thiadiazines; Hydrogenated 1,2,4-thiadiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with oxygen atoms directly attached to the ring sulfur atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0116622A FR2833950B1 (fr) | 2001-12-21 | 2001-12-21 | Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| PCT/FR2002/004484 WO2003053947A1 (fr) | 2001-12-21 | 2002-12-20 | Derives de benzothia(dia)zine et leur utilisation comme modulateurs ampa |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1456189T3 true DK1456189T3 (da) | 2007-11-05 |
Family
ID=8870810
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK02805407T DK1456189T3 (da) | 2001-12-21 | 2002-12-20 | Benzothia(dia)zin-derivater og deres anvendelse som AMPA-modulatorer |
Country Status (26)
| Country | Link |
|---|---|
| US (1) | US7250411B2 (ru) |
| EP (1) | EP1456189B1 (ru) |
| JP (1) | JP2005517668A (ru) |
| KR (1) | KR100606606B1 (ru) |
| CN (1) | CN1606550A (ru) |
| AR (1) | AR038029A1 (ru) |
| AT (1) | ATE366245T1 (ru) |
| AU (1) | AU2002365017B2 (ru) |
| BR (1) | BR0215145A (ru) |
| CA (1) | CA2471057A1 (ru) |
| DE (1) | DE60221041T2 (ru) |
| DK (1) | DK1456189T3 (ru) |
| EA (1) | EA007271B1 (ru) |
| ES (1) | ES2289182T3 (ru) |
| FR (1) | FR2833950B1 (ru) |
| GE (1) | GEP20063758B (ru) |
| HU (1) | HUP0402584A2 (ru) |
| MA (1) | MA27089A1 (ru) |
| MX (1) | MXPA04005838A (ru) |
| NO (1) | NO20042684L (ru) |
| NZ (1) | NZ533330A (ru) |
| PL (1) | PL369767A1 (ru) |
| PT (1) | PT1456189E (ru) |
| UA (1) | UA78743C2 (ru) |
| WO (1) | WO2003053947A1 (ru) |
| ZA (1) | ZA200404296B (ru) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2856065B1 (fr) * | 2003-06-13 | 2005-08-19 | Servier Lab | Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| FR2856064B1 (fr) * | 2003-06-13 | 2005-08-19 | Servier Lab | Nouveaux derives de benzothiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| FR2865474B1 (fr) * | 2004-01-26 | 2008-06-13 | Servier Lab | Nouveaux derives de benzothiazines fluorees, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| FR2877342B1 (fr) * | 2004-11-03 | 2007-01-26 | Servier Lab | Nouveaux derives de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| FR2877338B1 (fr) * | 2004-11-03 | 2007-01-26 | Servier Lab | Nouveaux derives de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| FR2879201B1 (fr) * | 2004-12-10 | 2007-02-16 | Servier Lab | Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| GB0724625D0 (en) * | 2007-12-18 | 2008-01-30 | Glaxo Group Ltd | Novel compounds |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU3957093A (en) * | 1992-04-15 | 1993-11-18 | Rhone-Poulenc Rorer S.A. | 3,4-dihydro-2H-1,2,4-benzothiadiazine-1,1-dioxide-3-carboxyl ic acid derivatives, preparation thereof and drugs containing same |
| WO1998012185A1 (en) * | 1996-09-17 | 1998-03-26 | The Regents Of The University Of California | Benzothiadiazide derivatives and their use as allosteric up-modulators of the ampa receptor |
| HUP0101280A3 (en) * | 1998-02-18 | 2003-02-28 | Neurosearch As | Positive ampa receptor modulator compounds and their use |
| FR2801587B1 (fr) * | 1999-11-30 | 2002-01-11 | Adir | Nouveaux derives de benzothiadiazines, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
-
2001
- 2001-12-21 FR FR0116622A patent/FR2833950B1/fr not_active Expired - Fee Related
-
2002
- 2002-12-18 AR ARP020104933A patent/AR038029A1/es unknown
- 2002-12-20 ES ES02805407T patent/ES2289182T3/es not_active Expired - Lifetime
- 2002-12-20 NZ NZ533330A patent/NZ533330A/en unknown
- 2002-12-20 DK DK02805407T patent/DK1456189T3/da active
- 2002-12-20 DE DE60221041T patent/DE60221041T2/de not_active Expired - Fee Related
- 2002-12-20 AT AT02805407T patent/ATE366245T1/de not_active IP Right Cessation
- 2002-12-20 UA UA20040706010A patent/UA78743C2/uk unknown
- 2002-12-20 AU AU2002365017A patent/AU2002365017B2/en not_active Ceased
- 2002-12-20 KR KR1020047009303A patent/KR100606606B1/ko not_active IP Right Cessation
- 2002-12-20 PT PT02805407T patent/PT1456189E/pt unknown
- 2002-12-20 MX MXPA04005838A patent/MXPA04005838A/es active IP Right Grant
- 2002-12-20 CN CNA028258142A patent/CN1606550A/zh active Pending
- 2002-12-20 HU HU0402584A patent/HUP0402584A2/hu unknown
- 2002-12-20 EP EP02805407A patent/EP1456189B1/fr not_active Expired - Lifetime
- 2002-12-20 WO PCT/FR2002/004484 patent/WO2003053947A1/fr active IP Right Grant
- 2002-12-20 CA CA002471057A patent/CA2471057A1/fr not_active Abandoned
- 2002-12-20 PL PL02369767A patent/PL369767A1/xx not_active Application Discontinuation
- 2002-12-20 BR BR0215145-6A patent/BR0215145A/pt not_active IP Right Cessation
- 2002-12-20 US US10/499,082 patent/US7250411B2/en not_active Expired - Fee Related
- 2002-12-20 JP JP2003554663A patent/JP2005517668A/ja active Pending
- 2002-12-20 GE GE5644A patent/GEP20063758B/en unknown
- 2002-12-20 EA EA200400756A patent/EA007271B1/ru not_active IP Right Cessation
-
2004
- 2004-06-01 ZA ZA200404296A patent/ZA200404296B/en unknown
- 2004-06-04 MA MA27718A patent/MA27089A1/fr unknown
- 2004-06-25 NO NO20042684A patent/NO20042684L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US7250411B2 (en) | 2007-07-31 |
| KR100606606B1 (ko) | 2006-08-01 |
| US20050014744A1 (en) | 2005-01-20 |
| KR20040065276A (ko) | 2004-07-21 |
| MXPA04005838A (es) | 2004-09-10 |
| PL369767A1 (en) | 2005-05-02 |
| ZA200404296B (en) | 2005-06-01 |
| EA007271B1 (ru) | 2006-08-25 |
| ATE366245T1 (de) | 2007-07-15 |
| MA27089A1 (fr) | 2004-12-20 |
| DE60221041T2 (de) | 2008-04-10 |
| WO2003053947A1 (fr) | 2003-07-03 |
| EP1456189A1 (fr) | 2004-09-15 |
| FR2833950A1 (fr) | 2003-06-27 |
| CN1606550A (zh) | 2005-04-13 |
| JP2005517668A (ja) | 2005-06-16 |
| EP1456189B1 (fr) | 2007-07-04 |
| FR2833950B1 (fr) | 2005-12-16 |
| ES2289182T3 (es) | 2008-02-01 |
| CA2471057A1 (fr) | 2003-07-03 |
| DE60221041D1 (de) | 2007-08-16 |
| AU2002365017B2 (en) | 2007-12-13 |
| GEP20063758B (en) | 2006-02-27 |
| EA200400756A1 (ru) | 2004-10-28 |
| BR0215145A (pt) | 2004-10-19 |
| NZ533330A (en) | 2006-05-26 |
| AU2002365017A1 (en) | 2003-07-09 |
| NO20042684L (no) | 2004-06-25 |
| PT1456189E (pt) | 2007-09-20 |
| HUP0402584A2 (hu) | 2005-04-28 |
| AR038029A1 (es) | 2004-12-22 |
| UA78743C2 (en) | 2007-04-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK1539712T3 (da) | Pyrimidinderivater og deres anvendelse som CB2-modulatorer | |
| DK1240164T3 (da) | Benzazolderivater og deres anvendelse som JNK-modulatorer | |
| DK1478629T3 (da) | N-aryl-2-oxazolidinon-5-carboxamider og deres derivater og deres anvendelse som antibakterielle midler | |
| NO20034439L (no) | Benzamidinderivater | |
| NO20035766L (no) | Aminonikotinatderivater som glukokinase (GLK) modulatorer | |
| DK1455785T3 (da) | Substituerede 2-thio-3,5-dicyano-4-phenyl-6-aminopyridiner og deres anvendelse | |
| DK1133477T3 (da) | Substituerede benzimidazoler og deres anvendelse som parpinhibitorer | |
| DK1204649T3 (da) | Arylmethylcarbonylaminothiazolderivater og deres anvendelse som antitumormidler | |
| DK1498413T3 (da) | 4-aminopicolinater og deres anvendelse som herbicider | |
| DK1282611T3 (da) | Substituerede phenylacetatamider og anvendelse deraf som glucokinaseaktivatorer | |
| NO20024742D0 (no) | Heterocykliske forbindelser, deres fremstilling og anvendelse | |
| IS6934A (is) | Nýjar spírótrísýklískar afleiður og notkun þeirrasem fosfódíesterasa-7-hindrar | |
| DK1956004T3 (da) | Quinolinderivater og deres anvendelse som 5-HT6-ligander | |
| ATE376831T1 (de) | Nicotin- oder isonicotin benzothiazole derivaten | |
| NO20021253L (no) | Kinolylpropylpiperidinderivater og deres anvendelse som antibakterielle midler | |
| NO20025150D0 (no) | 2-acylindolderivater og deres anvendelse som antitumormidler | |
| NO20042719L (no) | Substituerte 2-amino-cykloalkankarboksamider og deres anvendelse som protease-inhibitorer | |
| DK1603915T3 (da) | Substituerede 8-pyridinyl-dihydrospiro-cycloalkyl-pyrimido- 1,2-a-pyrimidin-6-on og 8-pyrimidinyl-dihydrospiro-cycloalkyl-pyrimido-1,2-a-pyrimidin-6-on-derivater og deres anvendelse mod neurogenerative sygdomme | |
| NO20044665L (no) | Renzoksazin-derivater som 5-HT6-modulatorer og anvendelser derav | |
| ATE459598T1 (de) | Sulfonamidderivate | |
| NO20031838D0 (no) | Benzokazinonderivater, deres fremstilling og anvendelse | |
| DK1387838T3 (da) | Cyanoanthranylamid-derivater og deres anvendelse som lægemidler | |
| NO20040210L (no) | Fenylacetamido-tiazolderivater, fremgangsmate for deres fremstilling og deres anvendelse som antitumormidler | |
| DK1456189T3 (da) | Benzothia(dia)zin-derivater og deres anvendelse som AMPA-modulatorer | |
| NO20043173L (no) | Benzotiazol- og benzoksazol-4,7-dionderivater og deres anvendelse som CDC25-fosfataseinhibitorer |