DK1448235T3 - Orale, farmaceutiske sammensætninger af 5,8,14-triaza-tetracyclo[10.3.1.0(2,11).0(4.9)]-hexadeca-2(11),3,5,7,9-pentaen med kontrolleret frigivelse - Google Patents

Orale, farmaceutiske sammensætninger af 5,8,14-triaza-tetracyclo[10.3.1.0(2,11).0(4.9)]-hexadeca-2(11),3,5,7,9-pentaen med kontrolleret frigivelse

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Publication number
DK1448235T3
DK1448235T3 DK02785718T DK02785718T DK1448235T3 DK 1448235 T3 DK1448235 T3 DK 1448235T3 DK 02785718 T DK02785718 T DK 02785718T DK 02785718 T DK02785718 T DK 02785718T DK 1448235 T3 DK1448235 T3 DK 1448235T3
Authority
DK
Denmark
Prior art keywords
pentaene
hexadeca
tetracyclo
triaza
pharmaceutical compositions
Prior art date
Application number
DK02785718T
Other languages
Danish (da)
English (en)
Inventor
Ende Mary Tanya Am
Michael Christopher Roy
Scott Wendell Smith
Kenneth Craig Waterman
Sara Kristen Moses
Ernest Shing Quan
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DK1448235T3 publication Critical patent/DK1448235T3/da

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
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    • A61K9/2022—Organic macromolecular compounds
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    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
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  • Inorganic Chemistry (AREA)
  • Immunology (AREA)
  • Psychology (AREA)
  • Diabetes (AREA)
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  • Anesthesiology (AREA)
  • Rheumatology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK02785718T 2001-11-30 2002-11-04 Orale, farmaceutiske sammensætninger af 5,8,14-triaza-tetracyclo[10.3.1.0(2,11).0(4.9)]-hexadeca-2(11),3,5,7,9-pentaen med kontrolleret frigivelse DK1448235T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US33465201P 2001-11-30 2001-11-30
PCT/IB2002/004612 WO2003045437A1 (en) 2001-11-30 2002-11-04 Pharmaceutical compositions of 5,7,14-triazatetracyclo[10.3.1.0(2,11).0(4,9)]-hexadeca-2(11)3,5,7,9-pentaene

Publications (1)

Publication Number Publication Date
DK1448235T3 true DK1448235T3 (da) 2007-07-02

Family

ID=23308160

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02785718T DK1448235T3 (da) 2001-11-30 2002-11-04 Orale, farmaceutiske sammensætninger af 5,8,14-triaza-tetracyclo[10.3.1.0(2,11).0(4.9)]-hexadeca-2(11),3,5,7,9-pentaen med kontrolleret frigivelse

Country Status (30)

Country Link
US (1) US7771748B2 (zh)
EP (1) EP1448235B1 (zh)
JP (2) JP2005528330A (zh)
KR (2) KR20040063975A (zh)
CN (2) CN1864663A (zh)
AR (1) AR037592A1 (zh)
AT (1) ATE356625T1 (zh)
AU (1) AU2002351008B2 (zh)
BR (1) BR0214806A (zh)
CA (1) CA2467490C (zh)
DE (1) DE60218885T2 (zh)
DK (1) DK1448235T3 (zh)
ES (1) ES2282492T3 (zh)
GT (1) GT200200247A (zh)
IL (1) IL161857A0 (zh)
MX (1) MXPA04003807A (zh)
MY (1) MY130619A (zh)
NO (1) NO20042739L (zh)
NZ (1) NZ532435A (zh)
PA (1) PA8559501A1 (zh)
PE (1) PE20040121A1 (zh)
PL (1) PL208080B1 (zh)
PT (1) PT1448235E (zh)
RU (2) RU2272629C2 (zh)
SI (1) SI1448235T1 (zh)
SV (1) SV2004001418A (zh)
TW (1) TWI327471B (zh)
UY (1) UY27553A1 (zh)
WO (1) WO2003045437A1 (zh)
ZA (1) ZA200403068B (zh)

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SE521512C2 (sv) * 2001-06-25 2003-11-11 Niconovum Ab Anordning för administrering av en substans till främre delen av en individs munhåla
KR20040063975A (ko) 2001-11-30 2004-07-15 화이자 프로덕츠 인크. 5,8,14-트리아자테트라시클로[10.3.1.0(2,11).0(4,9)]-헥사데카-2(11)3,5,7,9-펜타엔의 약학 조성물
EP3473251B1 (en) * 2002-12-20 2023-12-13 NicoNovum AB A nicotine-cellulose combination
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EP1942875B1 (en) * 2005-08-24 2015-08-12 Rubicon Research Private Limited Controlled release formulation
WO2007104573A2 (en) 2006-03-16 2007-09-20 Niconovum Ab Improved snuff composition
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WO2009143347A2 (en) 2008-05-22 2009-11-26 Teva Pharmaceutical Industries Ltd. Varenicline tosylate, an intermediate in the preparation process of varenicline l-tartrate
WO2009155403A2 (en) * 2008-06-19 2009-12-23 Teva Pharmaceutical Industries Ltd. Processes for the preparation of varenicline and intermediates thereof
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CN102427782A (zh) * 2009-05-21 2012-04-25 比奥内克斯制药有限公司 双层和单层剂型
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