DK142813B - Analogifremgangsmåde til fremstilling af 1-thiazolinyl- og 1-thiazinyl-benzimidazolestere. - Google Patents
Analogifremgangsmåde til fremstilling af 1-thiazolinyl- og 1-thiazinyl-benzimidazolestere. Download PDFInfo
- Publication number
- DK142813B DK142813B DK386276AA DK386276A DK142813B DK 142813 B DK142813 B DK 142813B DK 386276A A DK386276A A DK 386276AA DK 386276 A DK386276 A DK 386276A DK 142813 B DK142813 B DK 142813B
- Authority
- DK
- Denmark
- Prior art keywords
- benzimidazole
- amino
- give
- thiazolinyl
- carbon atoms
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
- C07C205/57—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Virology (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/633,203 US4008243A (en) | 1975-11-19 | 1975-11-19 | Antiviral thiazolinyl or thiazinyl benzimidazole esters |
| US63320375 | 1975-11-19 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK386276A DK386276A (es) | 1977-05-20 |
| DK142813B true DK142813B (da) | 1981-02-02 |
| DK142813C DK142813C (es) | 1981-09-21 |
Family
ID=24538665
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK386276AA DK142813B (da) | 1975-11-19 | 1976-08-26 | Analogifremgangsmåde til fremstilling af 1-thiazolinyl- og 1-thiazinyl-benzimidazolestere. |
Country Status (30)
| Country | Link |
|---|---|
| US (1) | US4008243A (es) |
| JP (1) | JPS5265269A (es) |
| AR (1) | AR218228A1 (es) |
| AT (1) | AT358029B (es) |
| AU (1) | AU498521B2 (es) |
| BE (1) | BE845643A (es) |
| BG (1) | BG27550A3 (es) |
| CA (1) | CA1059510A (es) |
| CH (1) | CH623052A5 (es) |
| CS (1) | CS199280B2 (es) |
| DD (1) | DD128675A5 (es) |
| DE (1) | DE2638552A1 (es) |
| DK (1) | DK142813B (es) |
| ES (2) | ES451020A1 (es) |
| FR (1) | FR2332011A1 (es) |
| GB (1) | GB1561481A (es) |
| GR (1) | GR61722B (es) |
| HU (1) | HU172633B (es) |
| IE (1) | IE43618B1 (es) |
| IL (1) | IL50294A (es) |
| MX (1) | MX4067E (es) |
| NL (1) | NL7609415A (es) |
| NZ (1) | NZ181788A (es) |
| PH (1) | PH13615A (es) |
| PL (2) | PL105486B1 (es) |
| PT (1) | PT65488B (es) |
| RO (1) | RO72653A (es) |
| SU (1) | SU721003A3 (es) |
| YU (1) | YU203576A (es) |
| ZA (1) | ZA765143B (es) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1076582A (en) * | 1975-10-28 | 1980-04-29 | Charles J. Paget | Antiviral thiazolinyl or thiazinyl ketobenzimidazoles |
| US4293558A (en) * | 1975-10-28 | 1981-10-06 | Eli Lilly And Company | Antiviral thiazolinyl benzimidazoles and derivatives |
| US4191832A (en) * | 1979-03-12 | 1980-03-04 | Eli Lilly And Company | Separation of syn and anti oximes of 1-sulfonyl-2-aminobenzimidazoles |
| US4338315A (en) * | 1979-11-14 | 1982-07-06 | Eli Lilly And Company | Antiviral method employing thiazinyl benzimidazole derivatives |
| US4401817A (en) * | 1981-04-20 | 1983-08-30 | Eli Lilly And Company | Carbonyl-substituted 1-sulfonylbenzimidazoles |
| US4434288A (en) * | 1982-04-08 | 1984-02-28 | Eli Lilly And Company | Preparation of substituted 1-thiazinyl or 1-thiazolyl-2-aminobenzimidazoles |
| US4463181A (en) * | 1982-04-08 | 1984-07-31 | Eli Lilly And Company | Process for removing sulfonyl groups from benzimidazole isomers |
| US4420479A (en) * | 1982-04-08 | 1983-12-13 | Eli Lilly And Company | Olefinic benzimidazoles, formulations, and antiviral methods |
| IL68297A (en) * | 1982-04-08 | 1986-09-30 | Lilly Co Eli | Process for removing 1-sulfonyl groups from 2-amino-5(6)-substituted benzimidazoles |
| US4492708A (en) * | 1982-09-27 | 1985-01-08 | Eli Lilly And Company | Antiviral benzimidazoles |
| US5508594A (en) * | 1994-06-10 | 1996-04-16 | Westinghouse Electric Corp | Electric vehicle chassis controller |
| US6358971B1 (en) | 1998-05-20 | 2002-03-19 | Eli Lilly And Company | Anti-viral compounds |
| US7652018B2 (en) * | 2006-08-15 | 2010-01-26 | Wyeth Llc | Imidazolidin-2-one derivatives useful as PR modulators |
| US7649007B2 (en) * | 2006-08-15 | 2010-01-19 | Wyeth Llc | Oxazolidine derivatives as PR modulators |
| WO2008021338A2 (en) * | 2006-08-15 | 2008-02-21 | Wyeth | Tricyclic oxazolidone derivatives useful as pr modulators |
| TW200815428A (en) * | 2006-08-15 | 2008-04-01 | Wyeth Corp | Oxazolidone derivatives as PR modulators |
| US7538107B2 (en) | 2006-08-15 | 2009-05-26 | Wyeth | Oxazinan-2-one derivatives useful as PR modulators |
| US20080045560A1 (en) * | 2006-08-15 | 2008-02-21 | Wyeth | Pyrrolidine and related derivatives useful as PR modulators |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3749717A (en) * | 1971-05-04 | 1973-07-31 | Squibb & Sons Inc | Thiazolinyl and thiazinyl derivatives of benzimidazoles |
| US3825537A (en) * | 1972-02-28 | 1974-07-23 | Squibb & Sons Inc | 1-thiazolin-2-yl(or thiazin-2-yl)-2-aminobenzimidazoles and derivatives thereof |
| US3833574A (en) * | 1972-07-31 | 1974-09-03 | Squibb & Sons Inc | Benzimidazolinone compounds |
-
1975
- 1975-11-19 US US05/633,203 patent/US4008243A/en not_active Expired - Lifetime
-
1976
- 1976-08-17 NZ NZ181788A patent/NZ181788A/xx unknown
- 1976-08-17 PT PT65488A patent/PT65488B/pt unknown
- 1976-08-17 GR GR51490A patent/GR61722B/el unknown
- 1976-08-17 MX MX763669U patent/MX4067E/es unknown
- 1976-08-18 HU HU76EI00000693A patent/HU172633B/hu unknown
- 1976-08-18 IL IL50294A patent/IL50294A/xx unknown
- 1976-08-19 YU YU02035/76A patent/YU203576A/xx unknown
- 1976-08-19 CA CA259,393A patent/CA1059510A/en not_active Expired
- 1976-08-19 AU AU16984/76A patent/AU498521B2/en not_active Expired
- 1976-08-19 AR AR264379A patent/AR218228A1/es active
- 1976-08-20 PH PH18822A patent/PH13615A/en unknown
- 1976-08-24 GB GB35092/76A patent/GB1561481A/en not_active Expired
- 1976-08-24 IE IE1883/76A patent/IE43618B1/en unknown
- 1976-08-24 NL NL7609415A patent/NL7609415A/xx not_active Application Discontinuation
- 1976-08-24 CS CS765494A patent/CS199280B2/cs unknown
- 1976-08-25 RO RO7687361A patent/RO72653A/ro unknown
- 1976-08-26 AT AT636576A patent/AT358029B/de not_active IP Right Cessation
- 1976-08-26 ES ES451020A patent/ES451020A1/es not_active Expired
- 1976-08-26 DE DE19762638552 patent/DE2638552A1/de not_active Withdrawn
- 1976-08-26 CH CH1085676A patent/CH623052A5/de not_active IP Right Cessation
- 1976-08-26 BG BG7634082A patent/BG27550A3/xx unknown
- 1976-08-26 SU SU762390302A patent/SU721003A3/ru active
- 1976-08-26 DK DK386276AA patent/DK142813B/da not_active IP Right Cessation
- 1976-08-27 DD DD7600194504A patent/DD128675A5/xx unknown
- 1976-08-27 FR FR7626028A patent/FR2332011A1/fr active Granted
- 1976-08-27 ZA ZA00765143A patent/ZA765143B/xx unknown
- 1976-08-27 BE BE1007588A patent/BE845643A/xx not_active IP Right Cessation
- 1976-09-14 PL PL1976192395A patent/PL105486B1/pl unknown
- 1976-09-14 PL PL1976210940A patent/PL110781B1/pl unknown
- 1976-11-17 JP JP51139043A patent/JPS5265269A/ja active Pending
-
1977
- 1977-08-16 ES ES461632A patent/ES461632A1/es not_active Expired
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PBP | Patent lapsed |