DK142701B - Analogifremgangsmåde til fremstilling af indol- eller azaindolforbindelser eller tautomere forbindelser eller syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af indol- eller azaindolforbindelser eller tautomere forbindelser eller syreadditionssalte deraf. Download PDF

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Publication number
DK142701B
DK142701B DK316674AA DK316674A DK142701B DK 142701 B DK142701 B DK 142701B DK 316674A A DK316674A A DK 316674AA DK 316674 A DK316674 A DK 316674A DK 142701 B DK142701 B DK 142701B
Authority
DK
Denmark
Prior art keywords
methanol
indole
solution
compounds
tetrahydro
Prior art date
Application number
DK316674AA
Other languages
Danish (da)
English (en)
Other versions
DK142701C (de
DK316674A (de
Inventor
Vishwa Prakash Arya
Kuppuswamy Nagarajan
Original Assignee
Ciba Geigy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy filed Critical Ciba Geigy
Publication of DK316674A publication Critical patent/DK316674A/da
Publication of DK142701B publication Critical patent/DK142701B/da
Application granted granted Critical
Publication of DK142701C publication Critical patent/DK142701C/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/06Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D239/08Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
    • C07D239/10Oxygen or sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK316674AA 1973-06-14 1974-06-13 Analogifremgangsmåde til fremstilling af indol- eller azaindolforbindelser eller tautomere forbindelser eller syreadditionssalte deraf. DK142701B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH860973 1973-06-14
CH860973A CH574441A5 (de) 1973-06-14 1973-06-14

Publications (3)

Publication Number Publication Date
DK316674A DK316674A (de) 1975-02-17
DK142701B true DK142701B (da) 1980-12-22
DK142701C DK142701C (de) 1981-09-21

Family

ID=4342576

Family Applications (1)

Application Number Title Priority Date Filing Date
DK316674AA DK142701B (da) 1973-06-14 1974-06-13 Analogifremgangsmåde til fremstilling af indol- eller azaindolforbindelser eller tautomere forbindelser eller syreadditionssalte deraf.

Country Status (17)

Country Link
US (1) US3954757A (de)
JP (1) JPS5849557B2 (de)
AT (1) AT333267B (de)
BE (1) BE816262A (de)
CH (1) CH574441A5 (de)
DD (1) DD112132A5 (de)
DE (1) DE2427207A1 (de)
DK (1) DK142701B (de)
ES (1) ES427269A1 (de)
FR (1) FR2233047B1 (de)
IE (1) IE39495B1 (de)
IL (1) IL44876A (de)
LU (1) LU70309A1 (de)
MC (1) MC1036A1 (de)
NL (1) NL7407614A (de)
SE (1) SE408709B (de)
YU (1) YU164774A (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5038759B2 (de) * 1971-12-20 1975-12-11
US4055647A (en) * 1973-06-14 1977-10-25 Ciba-Geigy Corporation Condensed pyrrole mercapto compounds having hypotensive and decongestant properties
BE503170A (de) * 1975-09-02
US3996218A (en) * 1975-09-08 1976-12-07 E. R. Squibb & Sons, Inc. Oxopyridazinylthiomethyl derivatives of ureidocephalosporins
US4171367A (en) * 1977-02-18 1979-10-16 Abbott Laboratories Pyrazolyl amino imidazolines
US5486525A (en) * 1993-12-16 1996-01-23 Abbott Laboratories Platelet activating factor antagonists: imidazopyridine indoles
US7582651B2 (en) * 2002-07-11 2009-09-01 Takeda Pharmaceutical Company Limited Pyrrolopyridine derivative and use thereof
EP2566481A4 (de) * 2010-05-06 2014-01-22 Merck Sharp & Dohme Als faah-modulatoren geeignete aza-indol-derivate

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1141949A (en) * 1966-02-23 1969-02-05 Sterling Drug Inc 7-azaindole derivatives
US3377247A (en) * 1967-04-28 1968-04-09 Dow Chemical Co Antidepressant method
US3586695A (en) * 1968-01-26 1971-06-22 Dow Chemical Co Substituted imidazolinyl indoles

Also Published As

Publication number Publication date
ES427269A1 (es) 1976-07-01
NL7407614A (de) 1974-12-17
AT333267B (de) 1976-11-10
IE39495B1 (en) 1978-10-25
DD112132A5 (de) 1975-03-20
IL44876A0 (en) 1974-07-31
DK142701C (de) 1981-09-21
JPS5035160A (de) 1975-04-03
SE408709B (sv) 1979-07-02
FR2233047A1 (de) 1975-01-10
MC1036A1 (fr) 1975-05-30
YU164774A (en) 1982-08-31
DE2427207A1 (de) 1975-01-09
JPS5849557B2 (ja) 1983-11-05
IE39495L (en) 1974-12-14
LU70309A1 (de) 1976-04-13
ATA484774A (de) 1976-03-15
DK316674A (de) 1975-02-17
IL44876A (en) 1978-01-31
SE7407175L (de) 1974-12-16
CH574441A5 (de) 1976-04-15
FR2233047B1 (de) 1977-11-04
BE816262A (fr) 1974-12-13
US3954757A (en) 1976-05-04

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PBP Patent lapsed