DK142319B - Analogifremgangsmåde til fremstilling af 3-quinolincarboxylsyrederivater. - Google Patents

Analogifremgangsmåde til fremstilling af 3-quinolincarboxylsyrederivater. Download PDF

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Publication number
DK142319B
DK142319B DK366175AA DK366175A DK142319B DK 142319 B DK142319 B DK 142319B DK 366175A A DK366175A A DK 366175AA DK 366175 A DK366175 A DK 366175A DK 142319 B DK142319 B DK 142319B
Authority
DK
Denmark
Prior art keywords
hydroxy
carboxylic acid
acid
quinoline carboxylic
quinoline
Prior art date
Application number
DK366175AA
Other languages
Danish (da)
English (en)
Other versions
DK366175A (el
DK142319C (el
Inventor
Francois Clemence
Roger Deraedt
Odile Le Martret
Andre Allais
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK366175A publication Critical patent/DK366175A/da
Publication of DK142319B publication Critical patent/DK142319B/da
Application granted granted Critical
Publication of DK142319C publication Critical patent/DK142319C/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK366175AA 1974-08-13 1975-08-13 Analogifremgangsmåde til fremstilling af 3-quinolincarboxylsyrederivater. DK142319B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7428038 1974-08-13
FR7428038A FR2281761A1 (fr) 1974-08-13 1974-08-13 Nouveaux derives de l'acide 3-quinoleine carboxylique, leur procede de preparation et leur application comme medicament

Publications (3)

Publication Number Publication Date
DK366175A DK366175A (el) 1976-02-14
DK142319B true DK142319B (da) 1980-10-13
DK142319C DK142319C (el) 1981-03-02

Family

ID=9142372

Family Applications (1)

Application Number Title Priority Date Filing Date
DK366175AA DK142319B (da) 1974-08-13 1975-08-13 Analogifremgangsmåde til fremstilling af 3-quinolincarboxylsyrederivater.

Country Status (21)

Country Link
US (1) US3992540A (el)
JP (1) JPS5925793B2 (el)
AR (1) AR208323A1 (el)
AT (1) AT340928B (el)
BE (1) BE832332A (el)
CA (1) CA1055499A (el)
CH (1) CH614953A5 (el)
DD (1) DD122972A5 (el)
DE (1) DE2536206C2 (el)
DK (1) DK142319B (el)
ES (1) ES440079A1 (el)
FR (1) FR2281761A1 (el)
GB (1) GB1484787A (el)
HU (1) HU170060B (el)
IE (1) IE41841B1 (el)
IL (1) IL47820A (el)
LU (1) LU73193A1 (el)
NL (1) NL7509625A (el)
SE (1) SE425244B (el)
SU (1) SU566522A3 (el)
ZA (1) ZA754905B (el)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2340735A1 (fr) * 1976-02-11 1977-09-09 Roussel Uclaf Nouveaux derives de l'acide 3-quinoleine carboxylique, leur procede de preparation et leur application comme medicament
FR2443467A1 (fr) * 1978-12-08 1980-07-04 Roussel Uclaf Nouveaux derives de l'acide 3-quinoleine carboxylique, leur procede de preparation et leur application comme medicament
FR2482596A1 (fr) * 1980-05-19 1981-11-20 Roussel Uclaf Nouveaux derives de l'acide 4-hydroxy 3-quinoleine carboxylique substitues en 2, leur procede de preparation et leur application comme medicament
IE52670B1 (en) * 1981-03-03 1988-01-20 Leo Ab Heterocyclic carboxamides,compositions containing such compounds,and processes for their preparation
HU190796B (en) * 1981-06-12 1986-11-28 Roussel Uclaf,Fr Process for producing n-dihydrothiazolyl-3-quinoline-carboxamide derivatives
FR2507602A1 (fr) * 1981-06-12 1982-12-17 Roussel Uclaf Nouveau derive dihydrothiazole de la quinoleine, ses sels, procede de preparation, application a titre de medicaments et compositions les renfermant
FR2523130A1 (fr) * 1982-03-15 1983-09-16 Roussel Uclaf Nouveaux derives de la n-dihydrothiazolyl-3-quinoleine carboxamide, leurs sels, procede de preparation, application a titre de medicaments et compositions les renfermant
FR2509728A1 (fr) * 1981-07-17 1983-01-21 Roussel Uclaf Nouveaux derives de la quinoleine, leurs sels, procede de preparation, application a titre de medicaments et compositions les renfermant
FR2537140B1 (fr) * 1982-12-07 1986-07-18 Roussel Uclaf Nouveaux derives de la 4-hydroxy-3-quinoleine carboxamide, leur sels, procede de preparation, application a titre de medicaments, et compositions les renfermant
FR2566405B1 (fr) * 1984-06-25 1986-09-26 Roussel Uclaf Nouveaux derives de l'acide 4-hydroxy 3-quinoleine carboxylique substitues en 2 par une fonction aminee, leur preparation, leur application comme medicaments, les compositions les renfermant et les intermediaires nouveaux obtenus
US4602014A (en) * 1984-07-09 1986-07-22 Ciba-Geigy Corporation Ring-fused pyrazolo[3,4-d]-pyridin-3-one derivatives as benzodiazepine receptor modulators
US4990533A (en) * 1985-12-20 1991-02-05 Warner-Lambert Co. Benzoic acid and benzoic acid ester derivatives having anti-inflammatory and analgesic activity
US4689182A (en) * 1985-12-20 1987-08-25 Warner-Lambert Company Benzoic acid and benzoic acid ester derivatives having anti-inflammatory and analgesic activity
US20100074949A1 (en) 2008-08-13 2010-03-25 William Rowe Pharmaceutical composition and administration thereof
DK2489659T3 (en) * 2004-06-24 2018-02-12 Vertex Pharma Modulators of ATP binding cassette conveyors
US8354427B2 (en) * 2004-06-24 2013-01-15 Vertex Pharmaceutical Incorporated Modulators of ATP-binding cassette transporters
AU2006331614A1 (en) * 2005-12-24 2007-07-05 Vertex Pharmaceuticals Incorporated Quinolin- 4 - one derivatives as modulators of ABC transporters
DK3219705T3 (da) 2005-12-28 2020-04-14 Vertex Pharma Farmaceutiske sammensætninger af den amorfe form af n-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinolin-3-carboxamid
SG193156A1 (en) 2009-03-20 2013-09-30 Vertex Pharma Process for making modulators of cystic fibrosis transmembrane conductance regulator
US8802700B2 (en) 2010-12-10 2014-08-12 Vertex Pharmaceuticals Incorporated Modulators of ATP-Binding Cassette transporters
US20130224293A1 (en) 2012-02-27 2013-08-29 Vertex Pharmaceuticals Incorporated Pharmaceutical composition and administrations thereof
MX370450B (es) 2014-10-07 2019-12-13 Vertex Pharma Co-cristales de moduladores de regulador de conductancia de transmembrana en fibrosis quistica.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH71A (de) * 1888-11-15 1889-06-13 Th Hunziker Apparat zum Absticken verlängerter Nädlinge für Handstickmaschinen
US2798070A (en) * 1954-02-04 1957-07-02 Mcneilab Inc Quaternary quinoline carboxamide salts and method of preparing same
JPS4323948Y1 (el) * 1965-03-06 1968-10-09
US3524858A (en) * 1967-05-18 1970-08-18 Warner Lambert Pharmaceutical 1,4 - dihydro-1-substituted alkyl-6,7-methylenedioxy - 4 - oxoquinoline-3-carboxylic acid
US3496184A (en) * 1969-03-18 1970-02-17 Ciba Geigy Corp Cyclopropylmethoxy-3-quinoline carboxylic acids and esters

Also Published As

Publication number Publication date
FR2281761A1 (fr) 1976-03-12
US3992540A (en) 1976-11-16
DK366175A (el) 1976-02-14
ZA754905B (en) 1976-08-25
IE41841L (en) 1976-02-13
IL47820A (en) 1978-10-31
JPS5925793B2 (ja) 1984-06-21
SE425244B (sv) 1982-09-13
CH614953A5 (el) 1979-12-28
CA1055499A (en) 1979-05-29
JPS5141366A (en) 1976-04-07
BE832332A (fr) 1976-02-12
AR208323A1 (es) 1976-12-20
IE41841B1 (en) 1980-04-09
LU73193A1 (el) 1976-08-13
AT340928B (de) 1978-01-10
DE2536206A1 (de) 1976-03-04
AU8340875A (en) 1977-01-27
ATA630875A (de) 1977-05-15
ES440079A1 (es) 1977-02-16
GB1484787A (en) 1977-09-08
SE7508332L (sv) 1976-02-16
NL7509625A (nl) 1976-02-17
DK142319C (el) 1981-03-02
DD122972A5 (de) 1976-11-12
HU170060B (el) 1977-03-28
IL47820A0 (en) 1975-10-15
SU566522A3 (ru) 1977-07-25
DE2536206C2 (de) 1984-07-19
FR2281761B1 (el) 1978-07-28

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