DK141846B - Analogifremgangsmåde til fremstilling af 1-oxo- eller 1-thioxo-s-triazolo(4,3-a)(1,4)benzodiazepinderivater. - Google Patents

Analogifremgangsmåde til fremstilling af 1-oxo- eller 1-thioxo-s-triazolo(4,3-a)(1,4)benzodiazepinderivater. Download PDF

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Publication number
DK141846B
DK141846B DK582970AA DK582970A DK141846B DK 141846 B DK141846 B DK 141846B DK 582970A A DK582970A A DK 582970AA DK 582970 A DK582970 A DK 582970A DK 141846 B DK141846 B DK 141846B
Authority
DK
Denmark
Prior art keywords
benzodiazepine
phenyl
chloro
parts
compound
Prior art date
Application number
DK582970AA
Other languages
Danish (da)
English (en)
Other versions
DK141846C (xx
Inventor
Kanji Meguro
Yutaka Kuwada
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of DK141846B publication Critical patent/DK141846B/da
Application granted granted Critical
Publication of DK141846C publication Critical patent/DK141846C/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK582970AA 1969-11-18 1970-11-17 Analogifremgangsmåde til fremstilling af 1-oxo- eller 1-thioxo-s-triazolo(4,3-a)(1,4)benzodiazepinderivater. DK141846B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP44092366A JPS4910958B1 (xx) 1969-11-18 1969-11-18
JP9236669 1969-11-18

Publications (2)

Publication Number Publication Date
DK141846B true DK141846B (da) 1980-06-30
DK141846C DK141846C (xx) 1980-11-24

Family

ID=14052400

Family Applications (1)

Application Number Title Priority Date Filing Date
DK582970AA DK141846B (da) 1969-11-18 1970-11-17 Analogifremgangsmåde til fremstilling af 1-oxo- eller 1-thioxo-s-triazolo(4,3-a)(1,4)benzodiazepinderivater.

Country Status (15)

Country Link
JP (2) JPS5010659B1 (xx)
AT (2) AT300816B (xx)
BE (1) BE759099A (xx)
CH (2) CH549588A (xx)
DE (2) DE2064926A1 (xx)
DK (1) DK141846B (xx)
ES (1) ES385641A1 (xx)
FI (1) FI51701C (xx)
FR (1) FR2073379B1 (xx)
GB (2) GB1337736A (xx)
NL (1) NL167697C (xx)
NO (1) NO126085B (xx)
SE (1) SE363111B (xx)
YU (1) YU34898B (xx)
ZA (1) ZA707644B (xx)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA713364B (en) * 1970-06-18 1972-01-26 Upjohn Co Prganic compounds and process
JPS494470B1 (xx) * 1970-08-26 1974-02-01
CH545302A (de) * 1971-04-08 1974-01-13 Ciba Geigy Ag Verfahren zur Herstellung von neuen Triazolo-benzodiazepinderivaten
US3751426A (en) * 1971-04-28 1973-08-07 Upjohn Co 1-substituted-6-phenyl-4h-s-triazolo(4,3-a)(1,6)benzodiazepine compounds
GB1377230A (en) * 1971-09-13 1974-12-11 Upjohn Co 4h-s-triazolo -4,3-a- 1,4-benzodiazepines
BE790356A (fr) * 1971-10-21 1973-04-20 Takeda Chemical Industries Ltd Derives de benzodiazepine
JPS5418280B2 (xx) * 1971-10-30 1979-07-06
BE793629A (fr) * 1972-01-03 1973-07-03 Upjohn Co Nouveaux derives de benzodiazepines et leur preparation
DE3021107A1 (de) * 1980-06-04 1981-12-17 Hoechst Ag, 6000 Frankfurt Carbamoyloxyamino-1,4-benzodiazepine, verfahren zu irer herstellung und diese enthaltende arzneimittel
CA1211437A (en) * 1981-08-12 1986-09-16 Rene Borer Benzazepines
CN111533745A (zh) * 2020-05-20 2020-08-14 成都药明康德新药开发有限公司 叔丁基-3-(氨基甲基)二氢-5h-三唑并二氮杂卓-8(9h)-甲酸基酯制法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI50981C (fi) * 1968-11-05 1976-09-10 Takeda Chemical Industries Ltd Menetelmä unilääkkeinä ja rauhoittavina lääkkeinä vaikuttavien s-triat solo-(4,3-a)(1,4)-bentsodiatsepiinien valmistamiseksi.
US3987052A (en) * 1969-03-17 1976-10-19 The Upjohn Company 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines

Also Published As

Publication number Publication date
ES385641A1 (es) 1973-10-01
DE2064926A1 (de) 1971-07-22
DE2056174A1 (de) 1971-06-24
JPS5010659B1 (xx) 1975-04-23
AT311993B (de) 1973-12-10
DK141846C (xx) 1980-11-24
GB1337737A (en) 1973-11-21
NL167697C (nl) 1982-01-18
BE759099A (fr) 1971-04-30
JPS4910958B1 (xx) 1974-03-13
NO126085B (xx) 1972-12-18
SE363111B (xx) 1974-01-07
ZA707644B (en) 1971-08-25
AT300816B (de) 1972-08-10
CH551432A (de) 1974-07-15
NL7016848A (xx) 1971-05-21
GB1337736A (en) 1973-11-21
FI51701C (fi) 1977-03-10
FI51701B (xx) 1976-11-30
CH549588A (de) 1974-05-31
NL167697B (nl) 1981-08-17
FR2073379A1 (xx) 1971-10-01
FR2073379B1 (xx) 1974-08-23
YU34898B (en) 1980-04-30
YU282770A (en) 1979-10-31

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