DK1385823T3 - Guanidinoforbindelser som melanocortin-4-receptor- (MC4-R) -agonister - Google Patents
Guanidinoforbindelser som melanocortin-4-receptor- (MC4-R) -agonisterInfo
- Publication number
- DK1385823T3 DK1385823T3 DK02719463T DK02719463T DK1385823T3 DK 1385823 T3 DK1385823 T3 DK 1385823T3 DK 02719463 T DK02719463 T DK 02719463T DK 02719463 T DK02719463 T DK 02719463T DK 1385823 T3 DK1385823 T3 DK 1385823T3
- Authority
- DK
- Denmark
- Prior art keywords
- melanocortin
- agonists
- receptor
- group
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/46—Iso-indoles; Hydrogenated iso-indoles with an oxygen atom in position 1
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/24—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/08—Radicals containing only hydrogen and carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/10—Radicals substituted by halogen atoms or nitro radicals
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Child & Adolescent Psychology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Cosmetics (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US28284701P | 2001-04-09 | 2001-04-09 | |
PCT/US2002/010965 WO2002081443A1 (en) | 2001-04-09 | 2002-04-08 | Novel guanidino compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
DK1385823T3 true DK1385823T3 (da) | 2007-03-26 |
Family
ID=23083379
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK02719463T DK1385823T3 (da) | 2001-04-09 | 2002-04-08 | Guanidinoforbindelser som melanocortin-4-receptor- (MC4-R) -agonister |
Country Status (10)
Country | Link |
---|---|
US (4) | US7456183B2 (ja) |
EP (2) | EP1767525A1 (ja) |
JP (1) | JP4172541B2 (ja) |
AT (1) | ATE348097T1 (ja) |
CY (1) | CY1107442T1 (ja) |
DE (1) | DE60216747T2 (ja) |
DK (1) | DK1385823T3 (ja) |
ES (1) | ES2278016T3 (ja) |
PT (1) | PT1385823E (ja) |
WO (1) | WO2002081443A1 (ja) |
Families Citing this family (75)
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US20030195187A1 (en) * | 2002-02-04 | 2003-10-16 | Chiron Corporation | Guanidino compounds |
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US20050124652A1 (en) * | 2002-02-04 | 2005-06-09 | Rustum Boyce | Guanidino compounds |
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DE19831710A1 (de) | 1998-07-15 | 2000-01-20 | Merck Patent Gmbh | Diacylhydrazinderivate |
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EP1767525A1 (en) | 2001-04-09 | 2007-03-28 | Novartis Vaccines and Diagnostics, Inc. | Guanidino compounds as melanocortin-4 receptor (MC4-R) agonists |
MXPA04011557A (es) | 2002-05-23 | 2005-07-05 | Chiron Corp | Compuestos de quinazolinona sustituida. |
US6638297B1 (en) * | 2002-05-30 | 2003-10-28 | Ethicon Endo-Surgery, Inc. | Surgical staple |
-
2002
- 2002-04-08 EP EP06025693A patent/EP1767525A1/en not_active Withdrawn
- 2002-04-08 DE DE60216747T patent/DE60216747T2/de not_active Expired - Lifetime
- 2002-04-08 PT PT02719463T patent/PT1385823E/pt unknown
- 2002-04-08 WO PCT/US2002/010965 patent/WO2002081443A1/en active IP Right Grant
- 2002-04-08 JP JP2002579431A patent/JP4172541B2/ja not_active Expired - Fee Related
- 2002-04-08 US US10/474,331 patent/US7456183B2/en not_active Expired - Fee Related
- 2002-04-08 US US10/118,730 patent/US6716840B2/en not_active Expired - Fee Related
- 2002-04-08 DK DK02719463T patent/DK1385823T3/da active
- 2002-04-08 ES ES02719463T patent/ES2278016T3/es not_active Expired - Lifetime
- 2002-04-08 EP EP02719463A patent/EP1385823B1/en not_active Expired - Lifetime
- 2002-04-08 AT AT02719463T patent/ATE348097T1/de not_active IP Right Cessation
-
2003
- 2003-04-30 US US10/426,937 patent/US6960582B2/en not_active Expired - Fee Related
-
2004
- 2004-04-05 US US10/818,187 patent/US7189727B2/en not_active Expired - Fee Related
-
2007
- 2007-02-15 CY CY20071100208T patent/CY1107442T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
US20040024211A1 (en) | 2004-02-05 |
US6960582B2 (en) | 2005-11-01 |
EP1767525A1 (en) | 2007-03-28 |
EP1385823A4 (en) | 2005-02-16 |
ES2278016T3 (es) | 2007-08-01 |
DE60216747T2 (de) | 2007-10-04 |
ATE348097T1 (de) | 2007-01-15 |
US6716840B2 (en) | 2004-04-06 |
US7456183B2 (en) | 2008-11-25 |
US20040248895A1 (en) | 2004-12-09 |
DE60216747D1 (de) | 2007-01-25 |
JP4172541B2 (ja) | 2008-10-29 |
EP1385823B1 (en) | 2006-12-13 |
US7189727B2 (en) | 2007-03-13 |
WO2002081443A1 (en) | 2002-10-17 |
EP1385823A1 (en) | 2004-02-04 |
US20020193595A1 (en) | 2002-12-19 |
US20050038027A1 (en) | 2005-02-17 |
PT1385823E (pt) | 2007-01-31 |
JP2004535378A (ja) | 2004-11-25 |
CY1107442T1 (el) | 2012-12-19 |
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